Literature DB >> 5654210

Irreversible enzyme inhibitors. CXV. Proteolytic enzymes. V. Active-site-directed irreversible inhibitors of trypsin derived from p-(phenoxyalkoxy) benzamidines with a terminal sulfonyl fluoride.

B R Baker, E H Erickson.   

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Year:  1968        PMID: 5654210     DOI: 10.1021/jm00308a011

Source DB:  PubMed          Journal:  J Med Chem        ISSN: 0022-2623            Impact factor:   7.446


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  5 in total

1.  SuFEx-enabled, agnostic discovery of covalent inhibitors of human neutrophil elastase.

Authors:  Qinheng Zheng; Jordan L Woehl; Seiya Kitamura; Diogo Santos-Martins; Christopher J Smedley; Gencheng Li; Stefano Forli; John E Moses; Dennis W Wolan; K Barry Sharpless
Journal:  Proc Natl Acad Sci U S A       Date:  2019-09-04       Impact factor: 11.205

2.  Arylfluorosulfates Inactivate Intracellular Lipid Binding Protein(s) through Chemoselective SuFEx Reaction with a Binding Site Tyr Residue.

Authors:  Wentao Chen; Jiajia Dong; Lars Plate; David E Mortenson; Gabriel J Brighty; Suhua Li; Yu Liu; Andrea Galmozzi; Peter S Lee; Jonathan J Hulce; Benjamin F Cravatt; Enrique Saez; Evan T Powers; Ian A Wilson; K Barry Sharpless; Jeffery W Kelly
Journal:  J Am Chem Soc       Date:  2016-06-02       Impact factor: 15.419

3.  Studies on ram acrosin. Activation of proacrosin accompanying the isolation of acrosin from spermatozoa, and purification of the enzyme by affinity chromatography.

Authors:  C R Brown; E F Hartree
Journal:  Biochem J       Date:  1978-10-01       Impact factor: 3.857

4.  "Affinity" chromatography of steroid-transforming enzymes with a non-steroidal ligand.

Authors:  A G Renwick; S M Chambers; P Willcox
Journal:  Biochem J       Date:  1979-02-01       Impact factor: 3.857

5.  Affinity chromatography of bovine trypsin. A rapid separation of bovine alpha- and beta-trypsin.

Authors:  G W Jameson; D T Elmore
Journal:  Biochem J       Date:  1974-08       Impact factor: 3.857

  5 in total

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