Literature DB >> 500698

Evaluation of methods for estimating the dissociation constant of tight binding enzyme inhibitors.

W R Greco, M T Hakala.   

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Year:  1979        PMID： 500698

Source DB:  PubMed          Journal:  J Biol Chem        ISSN： 0021-9258            Impact factor:   5.157


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  26 in total

1.  A human surfactant peptide-elastase inhibitor construct as a treatment for emphysema.

Authors:  Frank Guarnieri; Jean L Spencer; Edgar C Lucey; Matthew A Nugent; Phillip J Stone
Journal:  Proc Natl Acad Sci U S A       Date:  2010-06-01       Impact factor: 11.205

2.  Progress-curve equations for reversible enzyme-catalysed reactions inhibited by tight-binding inhibitors.

Authors:  S E Szedlacsek; V Ostafe; R G Duggleby; M Serban; M O Vlad
Journal:  Biochem J       Date:  1990-02-01       Impact factor: 3.857

3.  HIV-1 protease inhibitors from inverse design in the substrate envelope exhibit subnanomolar binding to drug-resistant variants.

Authors:  Michael D Altman; Akbar Ali; G S Kiran Kumar Reddy; Madhavi N L Nalam; Saima Ghafoor Anjum; Hong Cao; Sripriya Chellappan; Visvaldas Kairys; Miguel X Fernandes; Michael K Gilson; Celia A Schiffer; Tariq M Rana; Bruce Tidor
Journal:  J Am Chem Soc       Date:  2008-04-16       Impact factor: 15.419

4.  Computation of affinity and selectivity: binding of 2,4-diaminopteridine and 2,4-diaminoquinazoline inhibitors to dihydrofolate reductases.

Authors:  J Marelius; M Graffner-Nordberg; T Hansson; A Hallberg; J Aqvist
Journal:  J Comput Aided Mol Des       Date:  1998-03       Impact factor: 3.686

5.  Effect of temperature and chloride on steady-state inhibition of angiotensin I-converting enzyme by enalaprilat and ramiprilat.

Authors:  A Skoglof; P O Göthe; J Deinum
Journal:  Biochem J       Date:  1990-12-01       Impact factor: 3.857

6.  Ligand characterization of CYP4B1 isoforms modified for high-level expression in Escherichia coli and HepG2 cells.

Authors:  Katharina Roellecke; Vera D Jäger; Veselin H Gyurov; John P Kowalski; Stephanie Mielke; Allan E Rettie; Helmut Hanenberg; Constanze Wiek; Marco Girhard
Journal:  Protein Eng Des Sel       Date:  2017-03-01       Impact factor: 1.650

7.  The role of simulation in biomathematical modeling.

Authors:  W R Greco
Journal:  Bull Math Biol       Date:  1986       Impact factor: 1.758

8.  Slow-tight-binding inhibition of enoyl-acyl carrier protein reductase from Plasmodium falciparum by triclosan.

Authors:  Mili Kapoor; C Chandramouli Reddy; M V Krishnasastry; Namita Surolia; Avadhesha Surolia
Journal:  Biochem J       Date:  2004-08-01       Impact factor: 3.857

9.  ABT-378, a highly potent inhibitor of the human immunodeficiency virus protease.

Authors:  H L Sham; D J Kempf; A Molla; K C Marsh; G N Kumar; C M Chen; W Kati; K Stewart; R Lal; A Hsu; D Betebenner; M Korneyeva; S Vasavanonda; E McDonald; A Saldivar; N Wideburg; X Chen; P Niu; C Park; V Jayanti; B Grabowski; G R Granneman; E Sun; A J Japour; J M Leonard; J J Plattner; D W Norbeck
Journal:  Antimicrob Agents Chemother       Date:  1998-12       Impact factor: 5.191

10.  A family of diverse Kunitz inhibitors from Echinococcus granulosus potentially involved in host-parasite cross-talk.

Authors:  Silvia González; Martín Fló; Mariana Margenat; Rosario Durán; Gualberto González-Sapienza; Martín Graña; John Parkinson; Rick M Maizels; Gustavo Salinas; Beatriz Alvarez; Cecilia Fernández
Journal:  PLoS One       Date:  2009-09-17       Impact factor: 3.240
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