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19 in total

1. Crystallographic and kinetic investigations of the covalent complex formed by a specific tetrapeptide aldehyde and the serine protease from Streptomyces griseus.

Authors: G D Brayer; L T Delbaere; M N James; C A Bauer; R C Thompson
Journal: Proc Natl Acad Sci U S A Date: 1979-01 Impact factor: 11.205

2. Peptidyl inverse esters of p-methoxybenzoic acid: a novel class of potent inactivator of the serine proteases.

Authors: J Lynas; B Walker
Journal: Biochem J Date: 1997-08-01 Impact factor: 3.857

3. Pentavalent Organo-Vanadates as Transition State Analogues for Phosphoryl Transfer Reactions.

Authors: June M Messmore; Ronald T Raines
Journal: J Am Chem Soc Date: 2000-10-18 Impact factor: 15.419

4. Identification of the proteasome inhibitor MG262 as a potent ATP-dependent inhibitor of the Salmonella enterica serovar Typhimurium Lon protease.

Authors: Hilary Frase; Jason Hudak; Irene Lee
Journal: Biochemistry Date: 2006-07-11 Impact factor: 3.162

5. Binding of a possible transition state analogue to the active site of carboxypeptidase A.

Authors: D W Christianson; W N Lipscomb
Journal: Proc Natl Acad Sci U S A Date: 1985-10 Impact factor: 11.205

6. Identification of multiple structurally distinct, nonpeptidic small molecule inhibitors of protein arginine deiminase 3 using a substrate-based fragment method.

Authors: Haya Jamali; Hasan A Khan; Joseph R Stringer; Somenath Chowdhury; Jonathan A Ellman
Journal: J Am Chem Soc Date: 2015-03-05 Impact factor: 15.419

7. Benzyloxycarbonylprolylprolinal, a transition-state analogue for prolyl oligopeptidase, forms a tetrahedral adduct with catalytic serine, not a reactive cysteine.

Authors: A Kahyaoglu; K Haghjoo; F Kraicsovits; F Jordan; L Polgar
Journal: Biochem J Date: 1997-03-15 Impact factor: 3.857

Use of peptide aldehydes to generate transition-state analogs of elastase.