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6 in total

1. Synthesis and SARs of novel lincomycin derivatives Part 5: optimization of lincomycin analogs exhibiting potent antibacterial activities by chemical modification at the 6- and 7-positions.

Authors: Yoshinari Wakiyama; Ko Kumura; Eijiro Umemura; Satomi Masaki; Kazutaka Ueda; Yasuo Sato; Yoko Hirai; Yoshio Hayashi; Keiichi Ajito
Journal: J Antibiot (Tokyo) Date: 2017-11-01 Impact factor: 2.649

2. Absolute bioavailability of cis-mirincamycin and trans-mirincamycin in healthy rhesus monkeys and ex vivo antimalarial activity against Plasmodium falciparum.

Authors: Phisit Khemawoot; David Saunders; Maneerat Rasameesoraj; Victor Melendez; Rawiwan Imerbsin; Colin Ohrt; Susan Fracisco; Paktiya Teja-Isavadharm
Journal: Antimicrob Agents Chemother Date: 2011-09-26 Impact factor: 5.191

3. Synthesis and structure-activity relationships of novel lincomycin derivatives. Part 4: synthesis of novel lincomycin analogs modified at the 6- and 7-positions and their potent antibacterial activities.

Authors: Yoshinari Wakiyama; Ko Kumura; Eijiro Umemura; Kazutaka Ueda; Takashi Watanabe; Keiko Yamada; Takafumi Okutomi; Keiichi Ajito
Journal: J Antibiot (Tokyo) Date: 2017-05-31 Impact factor: 2.649

Lincomycin. 14. An improved synthesis and resolution of the antimalarial agent, 1'-demethyl-4'-depropyl-4'-(R)- and -(S)-pentylclindamycin hydrochloride (U-24, 729A).

1. Synthesis and SARs of novel lincomycin derivatives Part 5: optimization of lincomycin analogs exhibiting potent antibacterial activities by chemical modification at the 6- and 7-positions.

2. Absolute bioavailability of cis-mirincamycin and trans-mirincamycin in healthy rhesus monkeys and ex vivo antimalarial activity against Plasmodium falciparum.

3. Synthesis and structure-activity relationships of novel lincomycin derivatives. Part 4: synthesis of novel lincomycin analogs modified at the 6- and 7-positions and their potent antibacterial activities.

Review 4. The evolving role of chemical synthesis in antibacterial drug discovery.

5. In vitro activity of mirincamycin (U24729A) against Plasmodium falciparum isolates from Gabon.

6. Enhancement of the curative activity of primaquine by concomitant administration of mirincamycin.