Literature DB >> 3882966

Pepstatin-derived inhibitors of aspartic proteinases. A close look at an apparent transition-state analogue inhibitor.

D H Rich.   

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Year:  1985        PMID： 3882966     DOI： 10.1021/jm00381a001

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  12 in total

Review 1.  Nonproteinogenic amino acid building blocks for nonribosomal peptide and hybrid polyketide scaffolds.

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Review 2.  Renin inhibitors.

Authors:  W J Greenlee
Journal:  Pharm Res       Date:  1987-10       Impact factor: 4.200

3.  Positions of His-64 and a bound water in human carbonic anhydrase II upon binding three structurally related inhibitors.

Authors:  G M Smith; R S Alexander; D W Christianson; B M McKeever; G S Ponticello; J P Springer; W C Randall; J J Baldwin; C N Habecker
Journal:  Protein Sci       Date:  1994-01       Impact factor: 6.725

4.  Mechanism of action of aspartic proteinases: application of transition-state analogue theory.

Authors:  S Ołdziej; J Ciarkowski
Journal:  J Comput Aided Mol Des       Date:  1996-12       Impact factor: 3.686

5.  P1 and P1' para-fluoro phenyl groups show enhanced binding and favorable predicted pharmacological properties: structure-based virtual screening of extended lopinavir analogs against multi-drug resistant HIV-1 protease.

Authors:  Ravikiran S Yedidi; Zhigang Liu; Iulia A Kovari; Patrick M Woster; Ladislau C Kovari
Journal:  J Mol Graph Model       Date:  2013-11-01       Impact factor: 2.518

6.  Molecular basis for the inhibition of human alpha-thrombin by the macrocyclic peptide cyclotheonamide A.

Authors:  B E Maryanoff; X Qiu; K P Padmanabhan; A Tulinsky; H R Almond; P Andrade-Gordon; M N Greco; J A Kauffman; K C Nicolaou; A Liu
Journal:  Proc Natl Acad Sci U S A       Date:  1993-09-01       Impact factor: 11.205

7.  Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation.

Authors:  Jason C Kwan; Erika A Eksioglu; Chen Liu; Valerie J Paul; Hendrik Luesch
Journal:  J Med Chem       Date:  2009-09-24       Impact factor: 7.446

8.  Kinetics and mechanism of autoprocessing of human immunodeficiency virus type 1 protease from an analog of the Gag-Pol polyprotein.

Authors:  J M Louis; N T Nashed; K D Parris; A R Kimmel; D M Jerina
Journal:  Proc Natl Acad Sci U S A       Date:  1994-08-16       Impact factor: 11.205

9.  Renin inhibitor: relationship between molecular structure and oral absorption.

Authors:  N Hashimoto; T Fujioka; K Hayashi; K Odaguchi; T Toyoda; M Nakamura; K Hirano
Journal:  Pharm Res       Date:  1994-10       Impact factor: 4.200

10.  Inhibition of human immunodeficiency virus 1 protease in vitro: rational design of substrate analogue inhibitors.

Authors:  G B Dreyer; B W Metcalf; T A Tomaszek; T J Carr; A C Chandler; L Hyland; S A Fakhoury; V W Magaard; M L Moore; J E Strickler
Journal:  Proc Natl Acad Sci U S A       Date:  1989-12       Impact factor: 11.205
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