Literature DB >> 3803564

3,5-Diamino-1,2,6-thiadiazine 1,1-dioxide derivatives: synthesis and antiparasitic activity.

V J Arán, A G Bielsa, P Goya, C Ochoa, J A Páez, M Stud, M Contreras, J A Escario, M I Jiménez, E A Durán.   

Abstract

The synthesis of new 3,5-diamino-1,2,6-thiadiazine 1,1-dioxide derivatives is described and their structures discussed on the basis of 1H and 13C-N.M.R. data. The antiparasitic activity of these and related compounds was evaluated. The bacterial mutagenicity of the parent compound (I) was studied.

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Year:  1986        PMID： 3803564

Source DB:  PubMed          Journal:  Farmaco Sci        ISSN： 0430-0920


  2 in total

1.  Crystal structure, Hirshfeld analysis and a mol-ecular docking study of a new inhibitor of the Hepatitis B virus (HBV): ethyl 5-methyl-1,1-dioxo-2-{[5-(pentan-3-yl)-1,2,4-oxa-diazol-3-yl]meth-yl}-2H-1,2,6-thia-diazine-4-carboxyl-ate.

Authors:  Alexandre V Ivachtchenko; Sergiy M Kovalenko; Dmitry V Kravchenko; Oleg D Mitkin; Vladimir V Ivanov; Thierry Langer
Journal:  Acta Crystallogr E Crystallogr Commun       Date:  2020-01-01

2.  Ethyl 2-(3,5-dimethyl-1,1-dioxo-2H-1λ(6),2,6-thia-diazin-4-yl)benzoate.

Authors:  Nilay Bhatt; Pralav Bhatt; Kartik B Vyas; Kiran Nimavat; Thavendran Govender; Hendrik G Kruger; Glenn E M Maguire
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2012-06-20
  2 in total

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