Literature DB >> 36272052

The Role of the Non-Steroidal Mineralocorticoid Antagonist Finerenone in Cardiorenal Management.

Craig J Beavers1.   

Abstract

PURPOSE OF REVIEW: Finerenone is a novel, non-steroidal mineralocorticoid receptor antagonist (MRAs) that has been investigated for the management of cardiorenal conditions. This article provides an overview of recent evidence of benefits on cardiovascular (CV) outcomes. RECENT
FINDINGS: The recently published phase III FIDELIO-DKD and FIGARO-DKD, alone and pooled, in patients with CKD and diabetes demonstrate that finerenone reduces the composite of CV death, non-fatal myocardial infarction, nonfatal stroke, and hospitalization for heart failure (HF) with hospitalization for HF being the primary driver of this composite. Finerenone is indicated to reduce renal and CV outcomes in patients with CKD and diabetes. Future investigations of this agent include patients with non-diabetic CKD, HF with preserved ejection fraction, and with the use of sodium-glucose transporter type 2 inhibitors.
© 2022. The Author(s), under exclusive licence to Springer Science+Business Media, LLC, part of Springer Nature.

Entities:  

Keywords:  Cardiovascular disease; Chronic kidney disease; Finerenone; Heart failure; Mineralocorticoid antagonist; Type 2 diabetes mellitus

Year:  2022        PMID: 36272052     DOI: 10.1007/s11886-022-01795-1

Source DB:  PubMed          Journal:  Curr Cardiol Rep        ISSN: 1523-3782            Impact factor:   3.955


  25 in total

1.  Cardiorenal Syndrome: Classification, Pathophysiology, Diagnosis, and Treatment Strategies: A Scientific Statement From the American Heart Association.

Authors:  Janani Rangaswami; Vivek Bhalla; John E A Blair; Tara I Chang; Salvatore Costa; Krista L Lentine; Edgar V Lerma; Kenechukwu Mezue; Mark Molitch; Wilfried Mullens; Claudio Ronco; W H Wilson Tang; Peter A McCullough
Journal:  Circulation       Date:  2019-04-16       Impact factor: 29.690

2.  Direct and Indirect Mineralocorticoid Effects Determine Distal Salt Transport.

Authors:  Andrew S Terker; Bethzaida Yarbrough; Mohammed Z Ferdaus; Rebecca A Lazelle; Kayla J Erspamer; Nicholas P Meermeier; Hae J Park; James A McCormick; Chao-Ling Yang; David H Ellison
Journal:  J Am Soc Nephrol       Date:  2015-12-28       Impact factor: 10.121

Review 3.  Mechanisms of ligand specificity of the mineralocorticoid receptor.

Authors:  Peter J Fuller; Yizou Yao; Jun Yang; Morag J Young
Journal:  J Endocrinol       Date:  2011-12-12       Impact factor: 4.286

Review 4.  Nonsteroidal mineralocorticoid receptor antagonism for cardiovascular and renal disorders - New perspectives for combination therapy.

Authors:  Peter Kolkhof; Amer Joseph; Ulrich Kintscher
Journal:  Pharmacol Res       Date:  2021-08-28       Impact factor: 7.658

5.  Non-steroidal mineralocorticoid receptor antagonists in cardiorenal disease.

Authors:  Arjun K Pandey; Deepak L Bhatt; Francesco Cosentino; Nikolaus Marx; Ori Rotstein; Bertram Pitt; Ambarish Pandey; Javed Butler; Subodh Verma
Journal:  Eur Heart J       Date:  2022-08-14       Impact factor: 35.855

Review 6.  Novel non-steroidal mineralocorticoid receptor antagonists in cardiorenal disease.

Authors:  Ulrich Kintscher; George L Bakris; Peter Kolkhof
Journal:  Br J Pharmacol       Date:  2022-01-13       Impact factor: 9.473

Review 7.  Contribution of aldosterone to cardiovascular and renal inflammation and fibrosis.

Authors:  Nancy J Brown
Journal:  Nat Rev Nephrol       Date:  2013-06-18       Impact factor: 28.314

Review 8.  Approaches towards tissue-selective pharmacology of the mineralocorticoid receptor.

Authors:  Dorien Clarisse; Lisa Deng; Karolien de Bosscher; Achim Lother
Journal:  Br J Pharmacol       Date:  2021-12-16       Impact factor: 9.473

Review 9.  30 YEARS OF THE MINERALOCORTICOID RECEPTOR: Mineralocorticoid receptor antagonists: 60 years of research and development.

Authors:  Peter Kolkhof; Lars Bärfacker
Journal:  J Endocrinol       Date:  2017-07       Impact factor: 4.286

10.  Steroidal and non-steroidal mineralocorticoid receptor antagonists in cardiorenal medicine.

Authors:  Rajiv Agarwal; Peter Kolkhof; George Bakris; Johann Bauersachs; Hermann Haller; Takashi Wada; Faiez Zannad
Journal:  Eur Heart J       Date:  2021-01-07       Impact factor: 29.983

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