Literature DB >> 36267895

Randomised controlled trial of first-line tyrosine-kinase inhibitor (TKI) versus intercalated TKI with chemotherapy for EGFR-mutated nonsmall cell lung cancer.

Rolof G P Gijtenbeek1, Vincent van der Noort2, Joachim G J V Aerts3, Jeske A Staal-van den Brekel4, Egbert F Smit5, Frans H Krouwels6, Frank A Wilschut7, T Jeroen N Hiltermann8, Wim Timens9, Ed Schuuring9, Joost D J Janssen10, Martijn Goosens11, Paul M van den Berg12, A Joop de Langen13, Jos A Stigt14, Ben E E M van den Borne15, Harry J M Groen8, Wouter H van Geffen1, Anthonie J van der Wekken8.   

Abstract

Introduction: Previous studies have shown interference between epidermal growth factor receptor (EGFR) tyrosine kinase inhibitors and chemotherapy in the cell cycle, thus reducing efficacy. In this randomised controlled trial we investigated whether intercalated erlotinib with chemotherapy was superior compared to erlotinib alone in untreated advanced EGFR-mutated nonsmall cell lung cancer (NSCLC). Materials and methods: Treatment-naïve patients with an activating EGFR mutation, ECOG performance score of 0-3 and adequate organ function were randomly assigned 1:1 to either four cycles of cisplatin-pemetrexed with intercalated erlotinib (day 2-16 out of 21 days per cycle) followed by pemetrexed and erlotinib maintenance (CPE) or erlotinib monotherapy. The primary end-point was progression-free survival (PFS). Secondary end-points were overall survival, objective response rate (ORR) and toxicity.
Results: Between April 2014 and September 2016, 22 patients were randomised equally into both arms; the study was stopped due to slow accrual. Median follow-up was 64 months. Median PFS was 13.7 months (95% CI 5.2-18.8) for CPE and 10.3 months (95% CI 7.1-15.5; hazard ratio (HR) 0.62, 95% CI 0.25-1.57) for erlotinib monotherapy; when compensating for number of days receiving erlotinib, PFS of the CPE arm was superior (HR 0.24, 95% CI 0.07-0.83; p=0.02). ORR was 64% for CPE versus 55% for erlotinib monotherapy. Median overall survival was 31.7 months (95% CI 21.8-61.9 months) for CPE compared to 17.2 months (95% CI 11.5-45.5 months) for erlotinib monotherapy (HR 0.58, 95% CI 0.22-1.41 months). Patients treated with CPE had higher rates of treatment-related fatigue, anorexia, weight loss and renal toxicity.
Conclusion: Intercalating erlotinib with cisplatin-pemetrexed provides a longer PFS compared to erlotinib alone in EGFR-mutated NSCLC at the expense of more toxicity.
Copyright ©The authors 2022.

Entities:  

Year:  2022        PMID: 36267895      PMCID: PMC9574558          DOI: 10.1183/23120541.00239-2022

Source DB:  PubMed          Journal:  ERJ Open Res        ISSN: 2312-0541


  18 in total

1.  Clinical pharmacokinetics of erlotinib in patients with solid tumors and exposure-safety relationship in patients with non-small cell lung cancer.

Authors:  Jian-Feng Lu; Steve M Eppler; Julie Wolf; Marta Hamilton; Ashok Rakhit; Rene Bruno; Bert L Lum
Journal:  Clin Pharmacol Ther       Date:  2006-08       Impact factor: 6.875

2.  TRIBUTE: a phase III trial of erlotinib hydrochloride (OSI-774) combined with carboplatin and paclitaxel chemotherapy in advanced non-small-cell lung cancer.

Authors:  Roy S Herbst; Diane Prager; Robert Hermann; Lou Fehrenbacher; Bruce E Johnson; Alan Sandler; Mark G Kris; Hai T Tran; Pam Klein; Xin Li; David Ramies; David H Johnson; Vincent A Miller
Journal:  J Clin Oncol       Date:  2005-07-25       Impact factor: 44.544

3.  Combined epidermal growth factor receptor (EGFR)-tyrosine kinase inhibitor and chemotherapy in non-small-cell lung cancer: chemo-refractoriness of cells harboring sensitizing-EGFR mutations in the presence of gefitinib.

Authors:  Chun-Ming Tsai; Jen-Ting Chen; Chao-Hua Chiu; Chun-Liang Lai; Shih-Yin Hsiao; Kuo-Ting Chang
Journal:  Lung Cancer       Date:  2013-09-08       Impact factor: 5.705

4.  Gefitinib Versus Gefitinib Plus Pemetrexed and Carboplatin Chemotherapy in EGFR-Mutated Lung Cancer.

Authors:  Vanita Noronha; Vijay Maruti Patil; Amit Joshi; Nandini Menon; Anuradha Chougule; Abhishek Mahajan; Amit Janu; Nilendu Purandare; Rajiv Kumar; Sucheta More; Supriya Goud; Nandkumar Kadam; Nilesh Daware; Atanu Bhattacharjee; Srushti Shah; Akanksha Yadav; Vaishakhi Trivedi; Vichitra Behel; Amit Dutt; Shripad Dinanath Banavali; Kumar Prabhash
Journal:  J Clin Oncol       Date:  2019-08-14       Impact factor: 44.544

5.  Quality of life, symptom status and physical performance in patients with advanced non-small cell lung cancer undergoing chemotherapy: an exploratory analysis of secondary data.

Authors:  Shirin M Shallwani; Maureen J Simmonds; Goulnar Kasymjanova; Jadranka Spahija
Journal:  Lung Cancer       Date:  2016-06-23       Impact factor: 5.705

6.  Randomized Phase II Trial of Gefitinib With and Without Pemetrexed as First-Line Therapy in Patients With Advanced Nonsquamous Non-Small-Cell Lung Cancer With Activating Epidermal Growth Factor Receptor Mutations.

Authors:  Ying Cheng; Haruyasu Murakami; Pan-Chyr Yang; Jianxing He; Kazuhiko Nakagawa; Jin Hyoung Kang; Joo-Hang Kim; Xin Wang; Sotaro Enatsu; Tarun Puri; Mauro Orlando; James Chih-Hsin Yang
Journal:  J Clin Oncol       Date:  2016-08-09       Impact factor: 44.544

7.  Gefitinib in combination with paclitaxel and carboplatin in advanced non-small-cell lung cancer: a phase III trial--INTACT 2.

Authors:  Roy S Herbst; Giuseppe Giaccone; Joan H Schiller; Ronald B Natale; Vincent Miller; Christian Manegold; Giorgio Scagliotti; Rafael Rosell; Ira Oliff; James A Reeves; Michael K Wolf; Annetta D Krebs; Steven D Averbuch; Judith S Ochs; John Grous; Abderrahim Fandi; David H Johnson
Journal:  J Clin Oncol       Date:  2004-03-01       Impact factor: 44.544

8.  Osimertinib plus platinum-pemetrexed in newly diagnosed epidermal growth factor receptor mutation-positive advanced/metastatic non-small-cell lung cancer: safety run-in results from the FLAURA2 study.

Authors:  D Planchard; P-H Feng; N Karaseva; S-W Kim; T M Kim; C K Lee; A Poltoratskiy; N Yanagitani; R Marshall; X Huang; P Howarth; P A Jänne; K Kobayashi
Journal:  ESMO Open       Date:  2021-09-17

9.  Treatment goals and changes over time in older patients with non-curable cancer.

Authors:  M E Stegmann; D Brandenbarg; A K L Reyners; W H van Geffen; T J N Hiltermann; A J Berendsen
Journal:  Support Care Cancer       Date:  2020-12-22       Impact factor: 3.359

Review 10.  Resistance mechanisms to osimertinib in EGFR-mutated non-small cell lung cancer.

Authors:  Alessandro Leonetti; Sugandhi Sharma; Roberta Minari; Paola Perego; Elisa Giovannetti; Marcello Tiseo
Journal:  Br J Cancer       Date:  2019-09-30       Impact factor: 7.640

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