Literature DB >> 36267758

Efficacy and safety of apatinib in advanced refractory soft tissue sarcoma and association with histologic subtypes: a multicenter retrospective study.

Xiangling Wang1, Jian Wang1, Baoyong Sun2, Yuping Sun3, Ning Liu4, Xuecai Niu5, Chunhua Li6, Li Li1, Qiang Zhang7, Jing Hao1, Xiuwen Wang1.   

Abstract

Background: Antiangiogenic therapy is a potential strategy against advanced refractory soft tissue sarcoma (STS). This retrospective study aimed to assess the efficacy and safety of apatinib in patients with advanced refractory STS and explore its clinical effect on the different histologic subtypes.
Methods: Patients with pathologically diagnosed and metastatic STS who had failed at least standard chemotherapy and were naive to angiogenesis inhibitors were enrolled in this multicenter respective study. Apatinib was administered orally at a dosage of 250 to 850 mg/day. The primary endpoints were objective response rate (ORR) and disease control rate (DCR). The secondary endpoints were progression free survival (PFS) and overall survival (OS). Tumor assessment was done after the first 4 weeks and every 8 weeks thereafter.
Results: Twenty-six patients were enrolled from seven centers between December 2015 and December 2020, consisting of 9 leiomyosarcomas (LMS), 4 rhabdomyosarcomas (RMS), 3 undifferentiated pleomorphic cell sarcomas (UPS), 3 fibrosarcomas (FS), 3 alveolar soft part sarcomas (ASPS), 2 angiosarcomas (AS) and 2 synovial sarcomas (SS). The median age was 49.0 [26-77] years, 15 females and 11 males. The ORR was 34.62% [9/26, 95% confidence interval (CI): 19.42-53.78%] and DCR was as high as 84.62% (22/26, 95% CI: 66.47-93.85%). The median progression-free survival and overall survival were 6.0 months (95% CI: 2.42-9.58) and 19.3 months (95% CI: 7.31-31.29) respectively. Furthermore, 181 patients from seven studies as well as this trial were included for pooled analysis of apatinib efficacy dependency on histology. In terms of ORR, RMS (41.7%), ASPS (78.6%), and Ewing sarcoma (40.7%) seemed to benefit more than the other histologic subtypes. Common adverse events (AEs) included hand-foot skin reaction (n=13, 50.0%), hypertension (n=12, 46.15%), proteinuria (n=10, 38.46%). Seven patients (7/26, 26.92%) had grade 3 AEs and no grade 4 AEs occurred. 2 patients (2/26, 7.69%) and 15 patients (15/26, 57.69%) experienced dose withdrawal and dose reduction respectively. Conclusions: Apatinib showed promising efficacy and a manageable safety profile in patients with advanced refractory STS. In addition, the response to apatinib in STS seemed to be dependent on histology. 2022 Annals of Translational Medicine. All rights reserved.

Entities:  

Keywords:  Apatinib; advanced refractory soft tissue sarcoma; efficacy; safety

Year:  2022        PMID: 36267758      PMCID: PMC9577742          DOI: 10.21037/atm-22-3250

Source DB:  PubMed          Journal:  Ann Transl Med        ISSN: 2305-5839


  31 in total

1.  Pazopanib for metastatic soft-tissue sarcoma (PALETTE): a randomised, double-blind, placebo-controlled phase 3 trial.

Authors:  Winette T A van der Graaf; Jean-Yves Blay; Sant P Chawla; Dong-Wan Kim; Binh Bui-Nguyen; Paolo G Casali; Patrick Schöffski; Massimo Aglietta; Arthur P Staddon; Yasuo Beppu; Axel Le Cesne; Hans Gelderblom; Ian R Judson; Nobuhito Araki; Monia Ouali; Sandrine Marreaud; Rachel Hodge; Mohammed R Dewji; Corneel Coens; George D Demetri; Christopher D Fletcher; Angelo Paolo Dei Tos; Peter Hohenberger
Journal:  Lancet       Date:  2012-05-16       Impact factor: 79.321

Review 2.  Targeting angiogenesis for the treatment of sarcoma.

Authors:  Lakshmi Balasubramanian; Andrew M Evens
Journal:  Curr Opin Oncol       Date:  2006-07       Impact factor: 3.645

3.  Efficacy and Safety of Trabectedin or Dacarbazine for Metastatic Liposarcoma or Leiomyosarcoma After Failure of Conventional Chemotherapy: Results of a Phase III Randomized Multicenter Clinical Trial.

Authors:  George D Demetri; Margaret von Mehren; Robin L Jones; Martee L Hensley; Scott M Schuetze; Arthur Staddon; Mohammed Milhem; Anthony Elias; Kristen Ganjoo; Hussein Tawbi; Brian A Van Tine; Alexander Spira; Andrew Dean; Nushmia Z Khokhar; Youn Choi Park; Roland E Knoblauch; Trilok V Parekh; Robert G Maki; Shreyaskumar R Patel
Journal:  J Clin Oncol       Date:  2015-09-14       Impact factor: 44.544

4.  The Efficacy and Safety of Apatinib in Advanced Synovial Sarcoma: A Case Series of Twenty-One Patients in One Single Institution.

Authors:  Yitian Wang; Minxun Lu; Yong Zhou; Sisi Zhou; Xinzhu Yu; Fan Tang; Yi Luo; Wenli Zhang; Hong Duan; Li Min; Chongqi Tu
Journal:  Cancer Manag Res       Date:  2020-07-01       Impact factor: 3.989

5.  Apatinib for chemotherapy-refractory advanced metastatic gastric cancer: results from a randomized, placebo-controlled, parallel-arm, phase II trial.

Authors:  Jin Li; Shukui Qin; Jianming Xu; Weijian Guo; Jianping Xiong; Yuxian Bai; Guoping Sun; Yan Yang; Liwei Wang; Nong Xu; Ying Cheng; Zhehai Wang; Leizhen Zheng; Min Tao; Xiaodong Zhu; Dongmei Ji; Xin Liu; Hao Yu
Journal:  J Clin Oncol       Date:  2013-08-05       Impact factor: 44.544

6.  Randomized, Double-Blind, Placebo-Controlled Phase III Trial of Apatinib in Patients With Chemotherapy-Refractory Advanced or Metastatic Adenocarcinoma of the Stomach or Gastroesophageal Junction.

Authors:  Jin Li; Shukui Qin; Jianming Xu; Jianping Xiong; Changping Wu; Yuxian Bai; Wei Liu; Jiandong Tong; Yunpeng Liu; Ruihua Xu; Zhehai Wang; Qiong Wang; Xuenong Ouyang; Yan Yang; Yi Ba; Jun Liang; Xiaoyan Lin; Deyun Luo; Rongsheng Zheng; Xin Wang; Guoping Sun; Liwei Wang; Leizhen Zheng; Hong Guo; Jingbo Wu; Nong Xu; Jianwei Yang; Honggang Zhang; Ying Cheng; Ningju Wang; Lei Chen; Zhining Fan; Piaoyang Sun; Hao Yu
Journal:  J Clin Oncol       Date:  2016-02-16       Impact factor: 44.544

7.  Safety and Efficacy of Anlotinib, a Multikinase Angiogenesis Inhibitor, in Patients with Refractory Metastatic Soft-Tissue Sarcoma.

Authors:  Yihebali Chi; Zhiwei Fang; Xiaonan Hong; Yang Yao; Ping Sun; Guowen Wang; Feng Du; Yongkun Sun; Qiong Wu; Guofan Qu; Shusen Wang; Jianmin Song; Jianchun Yu; Yongkui Lu; Xia Zhu; Xiaohui Niu; Zhiyong He; Jinwan Wang; Hao Yu; Jianqiang Cai
Journal:  Clin Cancer Res       Date:  2018-06-12       Impact factor: 12.531

8.  Significant partial response of metastatic intra-abdominal and pelvic round cell liposarcoma to a small-molecule VEGFR-2 tyrosine kinase inhibitor apatinib: A case report.

Authors:  Min Dong; Jingwang Bi; Xiaohong Liu; Baocheng Wang; Jun Wang
Journal:  Medicine (Baltimore)       Date:  2016-08       Impact factor: 1.889

9.  The clinical outcome of pazopanib treatment in Japanese patients with relapsed soft tissue sarcoma: A Japanese Musculoskeletal Oncology Group (JMOG) study.

Authors:  Tomoki Nakamura; Akihiko Matsumine; Akira Kawai; Nobuhito Araki; Takahiro Goto; Tsukasa Yonemoto; Hideshi Sugiura; Yoshihiro Nishida; Hiroaki Hiraga; Kanya Honoki; Taketoshi Yasuda; Shogen Boku; Akihiro Sudo; Takafumi Ueda
Journal:  Cancer       Date:  2016-03-11       Impact factor: 6.860

10.  Advanced alveolar soft part sarcoma responds to apatinib.

Authors:  Yong Zhou; Fan Tang; Yiying Wang; Li Min; Yi Luo; Wenli Zhang; Rui Shi; Hong Duan; Chongqi Tu
Journal:  Oncotarget       Date:  2017-07-25
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