Literature DB >> 36266366

Clinical outcomes of concomitant use of proton pump inhibitors and regorafenib in patients with metastatic colorectal cancer: a multicenter study.

Emre Yekedüz1,2, Mehmet Fatih Özbay3, Dilek Çağlayan4, Atila Yıldırım5, Cihan Erol6, Hasan Çağrı Yıldırım7, Sezai Tunç8, Neslihan Özyurt9, Feyyaz Özdemir5, Mehmet Ali Nahit Şendur6, Abdurrahman Işıkdoğan8, Saadettin Kılıçkap7,10, Yüksel Ürün11,12, Şuayib Yalçın7, Mehmet Artaç4, Hasan Şenol Coşkun3, Güngör Utkan11,12.   

Abstract

AIM: To compare survival outcomes, response rates, and adverse events (AEs) in proton pump inhibitor (PPI) user and non-user patients with metastatic colorectal cancer (mCRC) treated with regorafenib.
METHODS: We included 272 patients with mCRC treated with regorafenib in this study. Patients were divided into two categories according to their status of PPI use. The primary endpoint was overall survival (OS). The secondary endpoints were time to treatment failure (TTF), response rates, and safety. To exclude immortal time bias in survival analyses, we compared PPI non-user patients and all patients.
RESULTS: There were 141 and 131 patients in the PPI non-user and user groups. Baseline characteristics were similar in each group. Pantoprazole was the most used PPI. At the median 35.2 (95% confidence interval (CI): 32.6-37.9) months follow-up, the median OS was similar in PPI non-user and all patients (6.9 months (95% CI: 5.3-8.5) and 7.7 months (95% CI:6.6-8.8), p = 0.913). TTF was also similar in PPI non-user and all patients (3.3 months (95% CI: 2.7-3.9) and 3.5 months (95% CI: 3.0-4.0), p = 0.661). In multivariable analysis, no statistically significant difference was observed between PPI user and non-user groups in OS and TTF (hazard ratio (HR), 0.99; 95% CI, 0.77-1.28; p = 0.963 for OS; HR, 0.93; 0.77-1.20, p = 0.598 for TTF). The objective response rates (ORR) were similar in the PPI non-user and user groups (19.8% and 16.8%, p = 0.455). The rates of any grade AEs were also similar in each group.
CONCLUSION: This study found no worse outcome in the combined use of PPI and regorafenib among patients with mCRC.
© 2022. The Author(s), under exclusive licence to Springer-Verlag GmbH Germany, part of Springer Nature.

Entities:  

Keywords:  Acid suppression; Drug-drug interactions; Regorafenib

Year:  2022        PMID: 36266366     DOI: 10.1007/s00228-022-03403-1

Source DB:  PubMed          Journal:  Eur J Clin Pharmacol        ISSN: 0031-6970            Impact factor:   3.064


  22 in total

Review 1.  Variability in bioavailability of small molecular tyrosine kinase inhibitors.

Authors:  Maikel Herbrink; Bastiaan Nuijen; Jan H M Schellens; Jos H Beijnen
Journal:  Cancer Treat Rev       Date:  2015-03-20       Impact factor: 12.111

Review 2.  Proton Pump Inhibitors in cancer patients: How useful they are? A review of the most common indications for their use.

Authors:  Gianmauro Numico; Vittorio Fusco; Pierfrancesco Franco; Fausto Roila
Journal:  Crit Rev Oncol Hematol       Date:  2017-02-03       Impact factor: 6.312

Review 3.  Indications and safety of proton pump inhibitor drug use in patients with cancer.

Authors:  George Triadafilopoulos; Andrew K Roorda; Junichi Akiyama
Journal:  Expert Opin Drug Saf       Date:  2013-05-07       Impact factor: 4.250

Review 4.  Pharmacokinetic drug-drug interactions of tyrosine kinase inhibitors: A focus on cytochrome P450, transporters, and acid suppression therapy.

Authors:  Caroline Gay; Delphine Toulet; Pascal Le Corre
Journal:  Hematol Oncol       Date:  2016-12-07       Impact factor: 5.271

Review 5.  Regorafenib: A Review of Its Use in Patients with Advanced Gastrointestinal Stromal Tumours.

Authors:  Matt Shirley; Gillian M Keating
Journal:  Drugs       Date:  2015-06       Impact factor: 9.546

Review 6.  Recent Advances in Systemic Therapy for Hepatocellular Carcinoma in an Aging Society: 2020 Update.

Authors:  Masatoshi Kudo
Journal:  Liver Cancer       Date:  2020-11-17       Impact factor: 11.740

Review 7.  Regorafenib: a novel multitargeted tyrosine kinase inhibitor for colorectal cancer and gastrointestinal stromal tumors.

Authors:  Daniel J Crona; Meredith D Keisler; Christine M Walko
Journal:  Ann Pharmacother       Date:  2013-11-01       Impact factor: 3.154

8.  Effects of Proton Pump Inhibitor Coadministration on the Plasma Concentration of Erlotinib in Patients With Non-Small Cell Lung Cancer.

Authors:  Masahiro Ohgami; Takayuki Kaburagi; Atsuhiko Kurosawa; Kosuke Doki; Toshihiro Shiozawa; Nobuyuki Hizawa; Masato Homma
Journal:  Ther Drug Monit       Date:  2018-12       Impact factor: 3.681

9.  Effect of the proton pump inhibitor esomeprazole on the oral absorption and pharmacokinetics of nilotinib.

Authors:  Ophelia Q P Yin; Neil Gallagher; Deirdre Fischer; Eren Demirhan; Wei Zhou; Georg Golor; Horst Schran
Journal:  J Clin Pharmacol       Date:  2010-05-24       Impact factor: 3.126

10.  Tyrosine Kinase Inhibitors and Proton Pump Inhibitors: An Evaluation of Treatment Options.

Authors:  Roelof W F van Leeuwen; Frank G A Jansman; Nicole G Hunfeld; Robert Peric; Anna K L Reyners; Alex L T Imholz; Jacobus R B J Brouwers; Joachim G Aerts; Teun van Gelder; Ron H J Mathijssen
Journal:  Clin Pharmacokinet       Date:  2017-07       Impact factor: 6.447

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