Literature DB >> 36260199

Long-term delayed emergence after remimazolam-based general anesthesia: a case report.

Tsubasa Takemori1, Yoshimasa Oyama2, Takenori Makino1, Seigo Hidaka1, Takaaki Kitano1.   

Abstract

BACKGROUND: Remimazolam is an ultra-short-acting benzodiazepine anesthetic that is antagonized by flumazenil, and it is typically expected to be applied in anesthesia with the purpose of ensuring early postoperative recovery. We report a case of long-term delayed emergence with re-sedation even after three times of flumazenil administration. CASE
PRESENTATION: A 71-year-old man was scheduled for a robotic-assisted laparoscopic radical prostatectomy for prostate cancer. We used remimazolam for anesthetic induction and maintenance. The intraoperative bispectral index (BIS) was 30-50. Flumazenil was administered as patient emergence was delayed after surgery; however, re-sedation was observed. This finding persisted till 12 h after surgery, and the patient awakened on postoperative day 2.
CONCLUSIONS: Remimazolam is a short-acting anesthetic, but long-term delayed emergence with re-sedation may occur even after flumazenil administration. Anesthesia using remimazolam requires anesthesia management that takes into account the individual differences in sensitivity and metabolism, with BIS as the indicator.
© 2022. The Author(s).

Entities:  

Keywords:  Benzodiazepines; Flumazenil; Prostatectomy; Prostatic neoplasms; Remimazolam

Year:  2022        PMID: 36260199      PMCID: PMC9582068          DOI: 10.1186/s40981-022-00576-7

Source DB:  PubMed          Journal:  JA Clin Rep        ISSN: 2363-9024


  15 in total

1.  A placebo- and midazolam-controlled phase I single ascending-dose study evaluating the safety, pharmacokinetics, and pharmacodynamics of remimazolam (CNS 7056): Part II. Population pharmacokinetic and pharmacodynamic modeling and simulation.

Authors:  Hugh R Wiltshire; Gavin J Kilpatrick; Gary S Tilbrook; Keith M Borkett
Journal:  Anesth Analg       Date:  2012-01-16       Impact factor: 5.108

2.  Bispectral index monitoring during sedation with sevoflurane, midazolam, and propofol.

Authors:  A E Ibrahim; J K Taraday; E D Kharasch
Journal:  Anesthesiology       Date:  2001-11       Impact factor: 7.892

3.  A placebo- and midazolam-controlled phase I single ascending-dose study evaluating the safety, pharmacokinetics, and pharmacodynamics of remimazolam (CNS 7056): Part I. Safety, efficacy, and basic pharmacokinetics.

Authors:  Laurie J Antonik; D Ronald Goldwater; Gavin J Kilpatrick; Gary S Tilbrook; Keith M Borkett
Journal:  Anesth Analg       Date:  2011-12-20       Impact factor: 5.108

4.  Safety and efficacy of remimazolam in induction and maintenance of general anesthesia in high-risk surgical patients (ASA Class III): results of a multicenter, randomized, double-blind, parallel-group comparative trial.

Authors:  Matsuyuki Doi; Naoyuki Hirata; Toshiyasu Suzuki; Hiroshi Morisaki; Hiroshi Morimatsu; Atsuhiro Sakamoto
Journal:  J Anesth       Date:  2020-04-17       Impact factor: 2.078

5.  Pharmacodynamic analysis of intravenous bolus remimazolam for loss of consciousness in patients undergoing general anaesthesia: a randomised, prospective, double-blind study.

Authors:  Dongwoo Chae; Hyun-Chang Kim; Young Song; Young Seo Choi; Dong Woo Han
Journal:  Br J Anaesth       Date:  2022-05-11       Impact factor: 11.719

Review 6.  The role of human carboxylesterases in drug metabolism: have we overlooked their importance?

Authors:  S Casey Laizure; Vanessa Herring; Zheyi Hu; Kevin Witbrodt; Robert B Parker
Journal:  Pharmacotherapy       Date:  2013-02       Impact factor: 4.705

7.  CNS 7056: a novel ultra-short-acting Benzodiazepine.

Authors:  Gavin J Kilpatrick; Margaret S McIntyre; Richard F Cox; Jeffrey A Stafford; Gregory J Pacofsky; Gwyer G Lovell; Robert P Wiard; Paul L Feldman; Holly Collins; Barbara L Waszczak; Gary S Tilbrook
Journal:  Anesthesiology       Date:  2007-07       Impact factor: 7.892

8.  Pharmacokinetic properties of remimazolam in subjects with hepatic or renal impairment.

Authors:  Thomas Stöhr; Pieter J Colin; Joachim Ossig; Marija Pesic; Keith Borkett; Peter Winkle; Michel M R F Struys; Frank Schippers
Journal:  Br J Anaesth       Date:  2021-07-08       Impact factor: 9.166

9.  Structure of a human synaptic GABAA receptor.

Authors:  Shaotong Zhu; Colleen M Noviello; Jinfeng Teng; Richard M Walsh; Jeong Joo Kim; Ryan E Hibbs
Journal:  Nature       Date:  2018-06-27       Impact factor: 49.962

10.  Shared structural mechanisms of general anaesthetics and benzodiazepines.

Authors:  Jeong Joo Kim; Anant Gharpure; Jinfeng Teng; Yuxuan Zhuang; Rebecca J Howard; Shaotong Zhu; Colleen M Noviello; Richard M Walsh; Erik Lindahl; Ryan E Hibbs
Journal:  Nature       Date:  2020-09-02       Impact factor: 49.962

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