Literature DB >> 35904596

The effectiveness and tolerability of fixed-dose combination netarsudil 0.02%/latanoprost 0.005% at a tertiary glaucoma center.

Jae-Chiang Wong1,2, Eric J Shiuey3, Reza Razeghinejad1,3, Aakriti G Shukla1,3, Natasha N Kolomeyer1,3, Jonathan S Myers1,3, Michael J Pro1,3, Daniel Lee4,5.   

Abstract

PURPOSE: To assess real-world effectiveness and tolerability of fixed-dose combination netarsudil 0.02%/latanoprost 0.005% (FCNL) in management of glaucoma patients in a tertiary eye care center.
METHODS: This retrospective cohort study included glaucoma patients initiated on FCNL from January 2018 to July 2021 with at least 1-month follow-up. Demographic and clinical data were collected at baseline and at follow-up visits through 12 months. Patient-solicited side effects were recorded at each visit. Maximum glaucoma pharmacotherapy was defined as surgery/laser being the next treatment option following an intensive pharmacotherapy regimen, or when pharmacotherapy could not be increased due to allergy/intolerance or all pharmacologic mechanisms already being in use.
RESULTS: Seventy-nine eyes of 47 patients were included. Mean age was 67.7 ± 14.7 years. Baseline IOP was 18.7 ± 4.9 mmHg; mean change in IOP (∆IOP) each study visit compared to baseline ranged from - 1.6 ± 3.5 to - 4.4 ± 4.1 mmHg (all p < 0.05). The eyes on maximum glaucoma pharmacotherapy (73.4%) had similar ∆IOP compared to those on non-maximal therapy at each visit (p > 0.2 for all). Forty-three (54.4%) eyes were switched from a prostaglandin analog alone, producing a 1-month IOP reduction of - 4.7 ± 3.9 mmHg at 1 month which remained significant at each visit for the 12-month study period (all p < 0.05). Across all study visits, conjunctival hyperemia was documented in 26 (32.9%) eyes. Subjective blurry vision was reported in 22 (27.8%) eyes without significant worsening of visual acuity at any visit (all p > 0.05). Six (7.6%) and 7 (8.9%) eyes required further medical or surgical/laser intervention, respectively. Kaplan-Meier analysis revealed no significant difference in the need for subsequent medical or surgical intervention between those on maximum and non-maximal pharmacotherapy (p > 0.4).
CONCLUSION: FCNL was well-tolerated and demonstrated a significant and sustained reduction in IOP, even as last-line therapy before incisional or laser surgery in those on maximum glaucoma pharmacotherapy. FCNL is a viable treatment option for glaucomatous eyes before consideration of surgical intervention.
© 2022. The Author(s), under exclusive licence to Springer-Verlag GmbH Germany, part of Springer Nature.

Entities:  

Keywords:  Fixed dose combination; Glaucoma; Glaucoma drops; Latanoprost; Netarsudil

Year:  2022        PMID: 35904596     DOI: 10.1007/s00417-022-05780-w

Source DB:  PubMed          Journal:  Graefes Arch Clin Exp Ophthalmol        ISSN: 0721-832X            Impact factor:   3.535


  14 in total

1.  Modulation of aqueous humor outflow facility by the Rho kinase-specific inhibitor Y-27632.

Authors:  P V Rao; P F Deng; J Kumar; D L Epstein
Journal:  Invest Ophthalmol Vis Sci       Date:  2001-04       Impact factor: 4.799

2.  Fixed-dose combination of AR-13324 and latanoprost: a double-masked, 28-day, randomised, controlled study in patients with open-angle glaucoma or ocular hypertension.

Authors:  Richard A Lewis; Brian Levy; Nancy Ramirez; Casey C Kopczynski; Dale W Usner; Gary D Novack
Journal:  Br J Ophthalmol       Date:  2015-07-24       Impact factor: 4.638

3.  Discovery of the ROCK inhibitor netarsudil for the treatment of open-angle glaucoma.

Authors:  Jill M Sturdivant; Susan M Royalty; Cheng-Wen Lin; Lori A Moore; Jeffrey D Yingling; Carmen L Laethem; Bryan Sherman; Geoffrey R Heintzelman; Casey C Kopczynski; Mitchell A deLong
Journal:  Bioorg Med Chem Lett       Date:  2016-04-01       Impact factor: 2.823

4.  Double-masked, randomized, dose-response study of AR-13324 versus latanoprost in patients with elevated intraocular pressure.

Authors:  Jason Bacharach; Harvey B Dubiner; Brian Levy; Casey C Kopczynski; Gary D Novack
Journal:  Ophthalmology       Date:  2014-09-27       Impact factor: 12.079

5.  Global data on visual impairment in the year 2002.

Authors:  Serge Resnikoff; Donatella Pascolini; Daniel Etya'ale; Ivo Kocur; Ramachandra Pararajasegaram; Gopal P Pokharel; Silvio P Mariotti
Journal:  Bull World Health Organ       Date:  2004-12-14       Impact factor: 9.408

Review 6.  Collaborative normal tension glaucoma study.

Authors:  Douglas R Anderson
Journal:  Curr Opin Ophthalmol       Date:  2003-04       Impact factor: 3.761

7.  One Year of Netarsudil and Latanoprost Fixed-Dose Combination for Elevated Intraocular Pressure: Phase 3, Randomized MERCURY-1 Study.

Authors:  Jacob W Brubaker; Savak Teymoorian; Richard A Lewis; Dale Usner; Hayley J McKee; Nancy Ramirez; Casey C Kopczynski; Theresa Heah
Journal:  Ophthalmol Glaucoma       Date:  2020-06-04

Review 8.  Rho Kinase Inhibitors as a Novel Treatment for Glaucoma and Ocular Hypertension.

Authors:  Angelo P Tanna; Mark Johnson
Journal:  Ophthalmology       Date:  2018-07-12       Impact factor: 12.079

9.  Two Phase 3 Clinical Trials Comparing the Safety and Efficacy of Netarsudil to Timolol in Patients With Elevated Intraocular Pressure: Rho Kinase Elevated IOP Treatment Trial 1 and 2 (ROCKET-1 and ROCKET-2).

Authors:  Janet B Serle; L Jay Katz; Eugene McLaurin; Theresa Heah; Nancy Ramirez-Davis; Dale W Usner; Gary D Novack; Casey C Kopczynski
Journal:  Am J Ophthalmol       Date:  2017-12-01       Impact factor: 5.258

10.  Fixed-Dose Combination of Netarsudil and Latanoprost in Ocular Hypertension and Open-Angle Glaucoma: Pooled Efficacy/Safety Analysis of Phase 3 MERCURY-1 and -2.

Authors:  Sanjay Asrani; Jason Bacharach; Edward Holland; Hayley McKee; Huan Sheng; Richard A Lewis; Casey C Kopczynski; Theresa Heah
Journal:  Adv Ther       Date:  2020-03-12       Impact factor: 3.845

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