Literature DB >> 35816198

TAK-242 treatment and its effect on mechanical properties and gene expression associated with IVD degeneration in SPARC-null mice.

Mitchel C Whittal1, Sarah J Poynter2, Kayla Samms2, K Josh Briar1, Sabrina I Sinopoli1, Magali Millecamps3, Laura S Stone3,4, Stephanie J DeWitte-Orr2, Diane E Gregory5,6.   

Abstract

PURPOSE: Intervertebral disc (IVD) degeneration is accompanied by mechanical and gene expression changes to IVDs. SPARC-null mice display accelerated IVD degeneration, and treatment with (toll-like receptor 4 (TLR4) inhibitor) TAK-242 decreases proinflammatory cytokines and pain. This study examined if chronic TAK-242 treatment impacts mechanical properties and gene expression associated with IVD degeneration in SPARC-null mice.
METHODS: Male and female SPARC-null and WT mice aged 7-9 months were given intraperitoneal injections with TAK-242 or an equivalent saline vehicle for 8 weeks (3x/per week, M-W-F). L2-L5 spinal segments were tested in cyclic axial tension and compression. Gene expression analysis (RT-qPCR) was performed on male IVD tissues using Qiagen RT2 PCR arrays.
RESULTS: SPARC-null mice had decreased NZ length (p = 0.001) and increased NZ stiffness (p < 0.001) compared to WT mice. NZ length was not impacted by TAK-242 treatment (p = 0.967) despite increased hysteresis energy (p = 0.024). Tensile stiffness was greater in SPARC-null mice (p = 0.018), and compressive (p < 0.001) stiffness was reduced from TAK-242 treatment in WT but not SPARC-null mice (p = 0.391). Gene expression analysis found upregulation of 13 ECM and 5 inflammatory genes in SPARC-null mice, and downregulation of 2 inflammatory genes after TAK-242 treatment.
CONCLUSIONS: TAK-242 had limited impacts on SPARC-null mechanical properties and did not attenuate NZ mechanical changes associated with IVD degeneration. Expression analysis revealed an increase in ECM and inflammatory gene expression in SPARCnull mice with a reduction in inflammatory expression due to TAK-242 treatment. This study provides insight into the role of TLR4 in SPARC-null mediated IVD degeneration.
© 2022. The Author(s), under exclusive licence to Springer-Verlag GmbH Germany, part of Springer Nature.

Entities:  

Keywords:  Axial loading; Degeneration; Gene expression; Inflammation; Intervertebral disc; TAK- 242

Mesh:

Substances:

Year:  2022        PMID: 35816198     DOI: 10.1007/s00586-022-07310-y

Source DB:  PubMed          Journal:  Eur Spine J        ISSN: 0940-6719            Impact factor:   2.721


  36 in total

1.  Biomechanical evaluation of segmental instability in degenerative lumbar spondylolisthesis.

Authors:  Kazuhiro Hasegewa; Ko Kitahara; Toshiaki Hara; Ko Takano; Haruka Shimoda
Journal:  Eur Spine J       Date:  2008-12-10       Impact factor: 3.134

2.  The Intervertebral Disc: Physiology and Pathology of a Brittle Joint.

Authors:  Aymeric Amelot; Christian Mazel
Journal:  World Neurosurg       Date:  2018-09-12       Impact factor: 2.104

Review 3.  Complexity of danger: the diverse nature of damage-associated molecular patterns.

Authors:  Liliana Schaefer
Journal:  J Biol Chem       Date:  2014-11-12       Impact factor: 5.157

Review 4.  Biomechanics of intervertebral disk degeneration.

Authors:  Nozomu Inoue; Alejandro A Espinoza Orías
Journal:  Orthop Clin North Am       Date:  2011-10       Impact factor: 2.472

Review 5.  What is intervertebral disc degeneration, and what causes it?

Authors:  Michael A Adams; Peter J Roughley
Journal:  Spine (Phila Pa 1976)       Date:  2006-08-15       Impact factor: 3.468

6.  Lumbar intervertebral disc mRNA sequencing identifies the regulatory pathway in patients with disc herniation and spondylolisthesis.

Authors:  Mohamad Bydon; F M Moinuddin; Yagiz U Yolcu; Waseem Wahood; Mohammed Ali Alvi; Anshit Goyal; Mohammed Elminawy; Catalina Galeano-Garces; Amel Dudakovic; Ahmad Nassr; A Noelle Larson; Andre J van Wijnen
Journal:  Gene       Date:  2020-03-30       Impact factor: 3.688

Review 7.  Cellular and molecular mechanisms of pain.

Authors:  Allan I Basbaum; Diana M Bautista; Grégory Scherrer; David Julius
Journal:  Cell       Date:  2009-10-16       Impact factor: 41.582

8.  Expression and regulation of toll-like receptors (TLRs) in human intervertebral disc cells.

Authors:  Marina Klawitter; Michiyuki Hakozaki; Hiroshi Kobayashi; Olga Krupkova; Lilian Quero; Caroline Ospelt; Steffen Gay; Oliver Hausmann; Thomas Liebscher; Ullrich Meier; Miho Sekiguchi; Shin-ichi Konno; Norbert Boos; Stephen J Ferguson; Karin Wuertz
Journal:  Eur Spine J       Date:  2014-07-05       Impact factor: 3.134

9.  Gene expression profile identifies potential biomarkers for human intervertebral disc degeneration.

Authors:  Wei Guo; Bin Zhang; Yan Li; Hui-Quan Duan; Chao Sun; Yun-Qiang Xu; Shi-Qing Feng
Journal:  Mol Med Rep       Date:  2017-10-09       Impact factor: 2.952

10.  Gene expression profile analysis of human intervertebral disc degeneration.

Authors:  Kai Chen; Dajiang Wu; Xiaodong Zhu; Haijian Ni; Xianzhao Wei; Ningfang Mao; Yang Xie; Yunfei Niu; Ming Li
Journal:  Genet Mol Biol       Date:  2013-08-30       Impact factor: 1.771

View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.