Literature DB >> 35446944

Favipiravir for treatment of outpatients with asymptomatic or uncomplicated COVID-19: a double-blind randomized, placebo-controlled, phase 2 trial.

Marisa Holubar1, Aruna Subramanian1, Natasha Purington2, Haley Hedlin2, Bryan Bunning2, Katharine S Walter1, Hector Bonilla1, Athanasia Boumis3, Michael Chen4, Kimberly Clinton3, Liisa Dewhurst3, Carol Epstein5, Prasanna Jagannathan1,6, Richard H Kaszynski4, Lori Panu3, Julie Parsonnet1,7, Elizabeth L Ponder8, Orlando Quintero1, Elizabeth Sefton8, Upinder Singh1,6, Luke Soberanis3, Henry Truong9, Jason R Andrews1, Manisha Desai2, Chaitan Khosla8,10, Yvonne Maldonado7,11.   

Abstract

BACKGROUND: Favipiravir is an oral, RNA-dependent RNA polymerase inhibitor with in vitro activity against SARS-CoV2. Despite limited data, favipiravir is administered to patients with COVID-19 in several countries.
METHODS: We conducted a phase 2 double-blind randomized controlled outpatient trial of favipiravir in asymptomatic or mildly symptomatic adults with a positive SARS-CoV2 RT-PCR within 72 hours of enrollment. Participants were randomized 1: 1 to receive placebo or favipiravir (1800mg BID Day 1, 800 mg BID Days 2-10). The primary outcome was SARS-CoV-2 shedding cessation in a modified intention-to-treat (mITT) cohort of participants with positive enrollment RT-PCRs. Using SARS-CoV-2 amplicon-based sequencing, we assessed favipiravir's impact on mutagenesis.
RESULTS: From July 8, 2020 - March 23, 2021, we randomized 149 participants with 116 included in the mITT cohort. The participants' mean age was 43 years (SD 12.5) and 57 (49%) were women. We found no difference in time to shedding cessation by treatment arm overall (HR 0.76 favoring placebo, 95% confidence interval [CI] 0.48-1.20) or in sub-group analyses (age, sex, high-risk comorbidities, seropositivity or symptom duration at enrollment). We observed no difference in time to symptom resolution (initial: HR 0.84, 95% CI 0.54-1.29; sustained: HR 0.87, 95% CI 0.52-1.45). We detected no difference in accumulation of transition mutations in the viral genome during treatment.
CONCLUSIONS: Our data do not support favipiravir use at commonly used doses in outpatients with uncomplicated COVID-19. Further research is needed to ascertain if higher doses of favipiravir are effective and safe for patients with COVID-19.
© The Author(s) 2022. Published by Oxford University Press on behalf of the Infectious Diseases Society of America.

Entities:  

Keywords:  COVID-19; SARS-CoV-2; clinical trial; favipiravir

Year:  2022        PMID: 35446944      PMCID: PMC9047233          DOI: 10.1093/cid/ciac312

Source DB:  PubMed          Journal:  Clin Infect Dis        ISSN: 1058-4838            Impact factor:   9.079


  6 in total

1.  Japanese rapid/living recommendations on drug management for COVID-19: updated guidelines (July 2022).

Authors:  Kazuma Yamakawa; Ryo Yamamoto; Takero Terayama; Hideki Hashimoto; Tadashi Ishihara; Go Ishimaru; Haruki Imura; Hiromu Okano; Chihiro Narita; Takuya Mayumi; Hideto Yasuda; Kohei Yamada; Hiroyuki Yamada; Tatsuya Kawasaki; Nobuaki Shime; Kent Doi; Moritoki Egi; Hiroshi Ogura; Morio Aihara; Shigeki Kushimoto; Osamu Nishida
Journal:  Acute Med Surg       Date:  2022-10-19

Review 2.  The efficacy and adverse effects of favipiravir on patients with COVID-19: A systematic review and meta-analysis of published clinical trials and observational studies.

Authors:  Dang The Hung; Suhaib Ghula; Jeza Muhamad Abdul Aziz; Abdelrahman M Makram; Gehad Mohamed Tawfik; Ali Ahmed-Fouad Abozaid; Rohan Andrew Pancharatnam; Amr Mohamed Ibrahim; Muhammad Besher Shabouk; Morgan Turnage; Saloni Nakhare; Zahra Karmally; Basel Kouz; Tran Nhat Le; Suleiman Alhijazeen; Nguyen Quoc Phuong; Alaa Mohamed Ads; Ali Hussein Abdelaal; Nguyen Hai Nam; Tatsuo Iiyama; Kyoshi Kita; Kenji Hirayama; Nguyen Tien Huy
Journal:  Int J Infect Dis       Date:  2022-04-22       Impact factor: 12.074

3.  Antiviral efficacy of favipiravir against Zika and SARS-CoV-2 viruses in non-human primates.

Authors:  Romain Marlin; Delphine Desjardins; Vanessa Contreras; Guillaume Lingas; Caroline Solas; Pierre Roques; Jeremie Guedj; Roger Le Grand; Thibaut Naninck; Quentin Pascal; Sylvie Behillil; Pauline Maisonnasse; Julien Lemaitre; Nidhal Kahlaoui; Benoit Delache; Andrés Pizzorno; Antoine Nougairede; Camille Ludot; Olivier Terrier; Nathalie Dereuddre-Bosquet; Francis Relouzat; Catherine Chapon; Raphael Ho Tsong Fang; Sylvie van der Werf; Manuel Rosa Calatrava; Denis Malvy; Xavier de Lamballerie
Journal:  Nat Commun       Date:  2022-08-30       Impact factor: 17.694

4.  Perspective: repurposed drugs for COVID-19.

Authors:  Kesara Na-Bangchang; Supatra Porasuphatana; Juntra Karbwang
Journal:  Arch Med Sci       Date:  2022-08-30       Impact factor: 3.707

5.  Early immune markers of clinical, virological, and immunological outcomes in patients with COVID-19: a multi-omics study.

Authors:  Zicheng Hu; Kattria van der Ploeg; Saborni Chakraborty; Prabhu S Arunachalam; Diego A M Mori; Karen B Jacobson; Hector Bonilla; Julie Parsonnet; Jason R Andrews; Marisa Holubar; Aruna Subramanian; Chaitan Khosla; Yvonne Maldonado; Haley Hedlin; Lauren de la Parte; Kathleen Press; Maureen Ty; Gene S Tan; Catherine Blish; Saki Takahashi; Isabel Rodriguez-Barraquer; Bryan Greenhouse; Atul J Butte; Upinder Singh; Bali Pulendran; Taia T Wang; Prasanna Jagannathan
Journal:  Elife       Date:  2022-10-14       Impact factor: 8.713

6.  Early treatment of Favipiravir in COVID-19 patients without pneumonia: a multicentre, open-labelled, randomized control study.

Authors:  Rujipas Sirijatuphat; Weerawat Manosuthi; Suvimol Niyomnaitham; Andrew Owen; Katherine Kradangna Copeland; Lantharita Charoenpong; Manoch Rattanasompattikul; Surakameth Mahasirimongkol; Nuanjun Wichukchinda; Kulkanya Chokephaibulkit
Journal:  Emerg Microbes Infect       Date:  2022-12       Impact factor: 19.568

  6 in total

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