Literature DB >> 35298785

Efficacy and safety of the apolipoprotein C-III inhibitor Volanesorsen: a systematic evaluation and meta-analysis.

Yonglang Cheng1, Tongxi Li1, Peng Tan2, Yichao Du2, Zhiwei Huang1, Hao Shi1, Tianying Cai1, Yifan Chen1, Wenguang Fu3,4.   

Abstract

PURPOSE: Familial celiac disease syndrome (FCS) is a form of hypertriglyceridemia (HTG) caused by the accumulation of celiac particles. Currently, volanesorsen is considered to be used to treat patients with FCS and HTG to improve symptoms. To evaluate the effect of volanesorsen on lipid metabolism in patients with FCS, we performed a systematic evaluation and meta-analysis.
METHODS: A systematic search of PubMed, Embase, ClinicalTrials.gov, and the Cochrane Library was conducted, and the bibliographies of original articles were checked manually. The quality of the studies was assessed using the Cochrane Risk of Bias tool.
RESULTS: Four randomized, controlled trials involving 246 patients were analyzed in this study. Patients treated with volanesorsen showed (MD = -78.85%; 95% CI = -96.04 to -61.65, P = 0.67, I2 = 0%) decrease in TG and (MD = -80.08%; 95% CI = -90.02 to -71.54, P = 0.25, I2 = 29%) decrease in ApoC-III levels compared to patients in the placebo group showing a significant decrease. In addition, HDL-C increased (MD = 46.01% 95% CI = 41.03 to 50.99, P = 0.41, I2 = 0%), NHDL-C decreased (MD = -32.12%; 95% CI = -44.39 to -19.85, P = 0.11, I2 = 55%), VLDL-C decreased (MD = -65.88%; 95% CI = -83.97 to -47.79, P = 0.71, I2 = 0%), apo A1 increased (MD = 13.12%; 95% CI = 7.83 to 18.40, P = 0.72, I2 = 0%), and apoB increased (MD = 7.94 %; 95% CI = -1.90 to 17.78, P = 0.54, I2 = 0%) all suggest that volanesorsen has an overall FCS with a therapeutic effect. However, LDL-C increased (MD = 99.59%; 95% CI = 69.19 to 130.00, P = 0.61, I2 = 0%) and apo B48 decreased (MD = 82.89%; 95% CI = -100.88 to -64.91, P = 0.42, I2 = 0%), showing an inverse effect, suggesting that volanesorsen's did not target all proteins of lipid metabolism.
© 2022. The Author(s), under exclusive licence to Springer Science+Business Media, LLC, part of Springer Nature.

Entities:  

Keywords:  Familial hypercoeliac disease syndrome; Lipid metabolism; Meta-analysis; Volanesorsen; systematic evaluation

Mesh:

Substances:

Year:  2022        PMID: 35298785     DOI: 10.1007/s12020-022-03025-8

Source DB:  PubMed          Journal:  Endocrine        ISSN: 1355-008X            Impact factor:   3.633


  17 in total

1.  Efficacy and safety of volanesorsen in patients with multifactorial chylomicronaemia (COMPASS): a multicentre, double-blind, randomised, placebo-controlled, phase 3 trial.

Authors:  Ioanna Gouni-Berthold; Veronica J Alexander; Qingqing Yang; Eunju Hurh; Elisabeth Steinhagen-Thiessen; Patrick M Moriarty; Stephen G Hughes; Daniel Gaudet; Robert A Hegele; Louis St L O'Dea; Erik S G Stroes; Sotirios Tsimikas; Joseph L Witztum
Journal:  Lancet Diabetes Endocrinol       Date:  2021-03-30       Impact factor: 32.069

2.  Rare variants in triglycerides-related genes increase pancreatitis risk in multifactorial chylomicronemia syndrome.

Authors:  Martine Paquette; Julie Amyot; Manon Fantino; Alexis Baass; Sophie Bernard
Journal:  J Clin Endocrinol Metab       Date:  2021-05-21       Impact factor: 5.958

Review 3.  The Chylomicronemia Syndrome Is Most Often Multifactorial: A Narrative Review of Causes and Treatment.

Authors:  Alan Chait; Robert H Eckel
Journal:  Ann Intern Med       Date:  2019-04-30       Impact factor: 25.391

4.  Volanesorsen and Triglyceride Levels in Familial Chylomicronemia Syndrome.

Authors:  Joseph L Witztum; Daniel Gaudet; Steven D Freedman; Veronica J Alexander; Andres Digenio; Karren R Williams; Qingqing Yang; Steven G Hughes; Richard S Geary; Marcello Arca; Erik S G Stroes; Jean Bergeron; Handrean Soran; Fernando Civeira; Linda Hemphill; Sotirios Tsimikas; Dirk J Blom; Louis O'Dea; Eric Bruckert
Journal:  N Engl J Med       Date:  2019-08-08       Impact factor: 91.245

5.  Antisense Inhibition of Apolipoprotein C-III in Patients with Hypertriglyceridemia.

Authors:  Daniel Gaudet; Veronica J Alexander; Brenda F Baker; Diane Brisson; Karine Tremblay; Walter Singleton; Richard S Geary; Steven G Hughes; Nicholas J Viney; Mark J Graham; Rosanne M Crooke; Joseph L Witztum; John D Brunzell; John J P Kastelein
Journal:  N Engl J Med       Date:  2015-07-30       Impact factor: 91.245

6.  Molecular and functional characterization of familial chylomicronemia syndrome.

Authors:  Ryota Teramoto; Hayato Tada; Masa-Aki Kawashiri; Atsushi Nohara; Takuya Nakahashi; Tetsuo Konno; Akihiro Inazu; Hiroshi Mabuchi; Masakazu Yamagishi; Kenshi Hayashi
Journal:  Atherosclerosis       Date:  2017-11-14       Impact factor: 5.162

7.  Apolipoprotein C-III inhibits triglyceride hydrolysis by GPIHBP1-bound LPL.

Authors:  Mikael Larsson; Christopher M Allan; Rachel S Jung; Patrick J Heizer; Anne P Beigneux; Stephen G Young; Loren G Fong
Journal:  J Lipid Res       Date:  2017-07-10       Impact factor: 5.922

Review 8.  Rare Treatments for Rare Dyslipidemias: New Perspectives in the Treatment of Homozygous Familial Hypercholesterolemia (HoFH) and Familial Chylomicronemia Syndrome (FCS).

Authors:  Laura D'Erasmo; Simone Bini; Marcello Arca
Journal:  Curr Atheroscler Rep       Date:  2021-09-01       Impact factor: 5.113

Review 9.  Targeting apoC-III and ANGPTL3 in the treatment of hypertriglyceridemia.

Authors:  N S Nurmohamed; G M Dallinga-Thie; E S G Stroes
Journal:  Expert Rev Cardiovasc Ther       Date:  2020-06-08
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