Literature DB >> 34949103

Provocation Testing and Therapeutic Response in a Newly Described Channelopathy: RyR2 Calcium Release Deficiency Syndrome.

Julian O M Ormerod1,2, Elizabeth Ormondroyd1, Yanhui Li3,4, John Taylor5, Jinhong Wei3, Wenting Guo3, Ruiwu Wang3, Caroline N S Sarton5, Karen McGuire5, Helene M P Dreau6, Jenny C Taylor7,5, Matthew R Ginks2, Kim Rajappan2, S R Wayne Chen3, Hugh Watkins1,7.   

Abstract

BACKGROUND: A novel familial arrhythmia syndrome, cardiac ryanodine receptor (RyR2) calcium release deficiency syndrome (CRDS), has recently been described. We evaluated a large and well characterized family to assess provocation testing, risk factor stratification and response to therapy in CRDS.
METHODS: We present a family with multiple unheralded sudden cardiac deaths and aborted cardiac arrests, primarily in children and young adults, with no clear phenotype on standard clinical testing.
RESULTS: Genetic analysis, including whole genome sequencing, firmly established that a missense mutation in RYR2, Ala4142Thr, was the underlying cause of disease in the family. Functional study of the variant in a cell model showed RyR2 loss-of-function, indicating that the family was affected by CRDS. EPS (Electrophysiological Study) was undertaken in 9 subjects known to carry the mutation, including a survivor of aborted sudden cardiac death, and the effects of flecainide alone and in combination with metoprolol were tested. There was a clear gradation in inducibility of nonsustained and sustained ventricular arrhythmia between subjects at EPS, with the survivor of aborted sudden cardiac death being the most inducible subject. Administration of flecainide substantially reduced arrhythmia inducibility in this subject and abolished arrhythmia in all others. Finally, the effects of additional metoprolol were tested; it increased inducibility in 4/9 subjects.
CONCLUSIONS: The Ala4142Thr mutation of RYR2 causes the novel heritable arrhythmia syndrome CRDS, which is characterized by familial sudden death in the absence of prior symptoms or a recognizable phenotype on ambulatory monitoring or exercise stress testing. We increase the experience of a specific EPS protocol in human subjects and show that it is helpful in establishing the clinical status of gene carriers, with potential utility for risk stratification. Our data provide evidence that flecainide is protective in human subjects with CRDS, consistent with the effect previously shown in a mouse model.

Entities:  

Keywords:  arrhythmias; calcium; phenotype; ryanodine receptor; young adult

Mesh:

Substances:

Year:  2021        PMID: 34949103     DOI: 10.1161/CIRCGEN.121.003589

Source DB:  PubMed          Journal:  Circ Genom Precis Med        ISSN: 2574-8300


  4 in total

1.  How does flecainide impact RyR2 channel function?

Authors:  Samantha C Salvage; Christopher L-H Huang; James A Fraser; Angela F Dulhunty
Journal:  J Gen Physiol       Date:  2022-06-17       Impact factor: 4.000

Review 2.  Therapeutic Approaches of Ryanodine Receptor-Associated Heart Diseases.

Authors:  Norbert Szentandrássy; Zsuzsanna É Magyar; Judit Hevesi; Tamás Bányász; Péter P Nánási; János Almássy
Journal:  Int J Mol Sci       Date:  2022-04-18       Impact factor: 6.208

Review 3.  The Antiarrhythmic Mechanisms of Flecainide in Catecholaminergic Polymorphic Ventricular Tachycardia.

Authors:  Yukun Li; Xiaodong Peng; Rong Lin; Xuesi Wang; Xinmeng Liu; Rong Bai; Changsheng Ma; Ribo Tang; Yanfei Ruan; Nian Liu
Journal:  Front Physiol       Date:  2022-03-09       Impact factor: 4.566

Review 4.  Molecular, Subcellular, and Arrhythmogenic Mechanisms in Genetic RyR2 Disease.

Authors:  Ewan Douglas Fowler; Spyros Zissimopoulos
Journal:  Biomolecules       Date:  2022-07-26
  4 in total

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