Literature DB >> 34927004

New Drug Modalities in Medicinal Chemistry, Pharmacology, and Translational Science: Joint Virtual Special Issue by Journal of Medicinal Chemistry, ACS Medicinal Chemistry Letters, and ACS Pharmacology & Translational Science.

Christa E Müller, Finn K Hansen, Michael Gütschow, Craig W Lindsley, Dennis Liotta.   

Abstract

Entities:  

Year:  2021        PMID: 34927004      PMCID: PMC8669705          DOI: 10.1021/acsptsci.1c00208

Source DB:  PubMed          Journal:  ACS Pharmacol Transl Sci        ISSN: 2575-9108


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  7 in total

Review 1.  Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings.

Authors:  C A Lipinski; F Lombardo; B W Dominy; P J Feeney
Journal:  Adv Drug Deliv Rev       Date:  2001-03-01       Impact factor: 15.470

Review 2.  New Modalities, Technologies, and Partnerships in Probe and Lead Generation: Enabling a Mode-of-Action Centric Paradigm.

Authors:  Eric Valeur; Patrick Jimonet
Journal:  J Med Chem       Date:  2018-06-13       Impact factor: 7.446

3.  New Chemical Modalities and Strategic Thinking in Early Drug Discovery.

Authors:  Maria-Jesus Blanco; Kevin M Gardinier
Journal:  ACS Med Chem Lett       Date:  2020-01-14       Impact factor: 4.345

4.  Targeted protein degradation: expanding the toolbox.

Authors:  Matthieu Schapira; Matthew F Calabrese; Alex N Bullock; Craig M Crews
Journal:  Nat Rev Drug Discov       Date:  2019-10-30       Impact factor: 84.694

Review 5.  Targeted protein degradation: A promise for undruggable proteins.

Authors:  Kusal T G Samarasinghe; Craig M Crews
Journal:  Cell Chem Biol       Date:  2021-05-17       Impact factor: 9.039

Review 6.  PROTACs: An Emerging Therapeutic Modality in Precision Medicine.

Authors:  Dhanusha A Nalawansha; Craig M Crews
Journal:  Cell Chem Biol       Date:  2020-08-13       Impact factor: 9.039

Review 7.  Designing Chimeric Molecules for Drug Discovery by Leveraging Chemical Biology.

Authors:  Chiara Borsari; Darci J Trader; Annalisa Tait; Maria P Costi
Journal:  J Med Chem       Date:  2020-02-19       Impact factor: 7.446

  7 in total

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