Literature DB >> 34843030

New Antipsychotic Medications in the Last Decade.

Mehak Pahwa1, Ahmad Sleem2, Omar H Elsayed2, Megan Elizabeth Good2, Rif S El-Mallakh3.   

Abstract

PURPOSE OF REVIEW: Over the last ten years, the treatment of psychosis has seen a near explosion of creative development in both novel agents and new delivery modalities. The current review summarizes these developments over the past decade (2011-2020). We performed a systematic review utilizing PubMed and PsychInfo with the aim of identifying all the RCT and related analyses in adults with psychosis (schizophrenia and mania). RECENT
FINDINGS: We identified 11 significant developments: the introduction of new antipsychotics cariprazine, brexpiprazole, lumateperone, and pimavanserin; introduction of new delivery methods: subcutaneous long-acting risperidone, aripiprazole lauroxil, transdermal asenapine, and inhaled loxapine; and the introduction of new approaches such as olanzapine/samidorphan for olanzapine-associated weight gain, examination of the TAAR1 agonist SEP 363,856 as a test of concept, and the combination of Xanomeline/Trospium, an M1 and M4 muscarinic receptor agonist in conjunction with a peripheral anticholinergic. Last decade has seen a tremendous development in second-generation antipsychotics which provides unprecedented treatment options for clinicians in treating psychosis.
© 2021. The Author(s), under exclusive licence to Springer Science+Business Media, LLC, part of Springer Nature.

Entities:  

Keywords:  Aripiprazole lauroxil; Brexpiprazole; Cariprazine; Inhaled loxapine; Lumateperone; New antipsychotics; Olanzapine/samidorphan; Pimavanserin; SEP-363856; Subcutaneous risperidone; Transdermal asenapine; Xanomeline/trospium

Mesh:

Substances:

Year:  2021        PMID: 34843030     DOI: 10.1007/s11920-021-01298-w

Source DB:  PubMed          Journal:  Curr Psychiatry Rep        ISSN: 1523-3812            Impact factor:   5.285


  165 in total

1.  Discovery of cariprazine (RGH-188): a novel antipsychotic acting on dopamine D3/D2 receptors.

Authors:  Eva Agai-Csongor; György Domány; Katalin Nógrádi; János Galambos; István Vágó; György Miklós Keserű; István Greiner; István Laszlovszky; Anikó Gere; Eva Schmidt; Béla Kiss; Mónika Vastag; Károly Tihanyi; Katalin Sághy; Judit Laszy; István Gyertyán; Mária Zájer-Balázs; Larisza Gémesi; Margit Kapás; Zsolt Szombathelyi
Journal:  Bioorg Med Chem Lett       Date:  2012-04-04       Impact factor: 2.823

2.  Cariprazine: First Global Approval.

Authors:  Paul L McCormack
Journal:  Drugs       Date:  2015-11       Impact factor: 9.546

3.  An evaluation of the safety and efficacy of cariprazine in patients with acute exacerbation of schizophrenia: a phase II, randomized clinical trial.

Authors:  Suresh Durgam; Anju Starace; Dayong Li; Raffaele Migliore; Adam Ruth; György Németh; István Laszlovszky
Journal:  Schizophr Res       Date:  2014-01-10       Impact factor: 4.939

4.  Cariprazine in acute exacerbation of schizophrenia: a fixed-dose, phase 3, randomized, double-blind, placebo- and active-controlled trial.

Authors:  Suresh Durgam; Andrew J Cutler; Kaifeng Lu; Raffaele Migliore; Adam Ruth; István Laszlovszky; György Németh; Herbert Y Meltzer
Journal:  J Clin Psychiatry       Date:  2015-12       Impact factor: 4.384

5.  Brain uptake and distribution of the dopamine D3 /D2 receptor partial agonist [11 C]cariprazine: an in vivo positron emission tomography study in nonhuman primates.

Authors:  Miklós Tóth; Andrea Varrone; Carsten Steiger; István Laszlovszky; Attila Horváth; Béla Kiss; István Gyertyán; Nika Adham; Christer Halldin; Balázs Gulyás
Journal:  Synapse       Date:  2013-02-08       Impact factor: 2.562

6.  Occupancy of dopamine D₂ and D₃ and serotonin 5-HT₁A receptors by the novel antipsychotic drug candidate, cariprazine (RGH-188), in monkey brain measured using positron emission tomography.

Authors:  Nicholas Seneca; Sjoerd J Finnema; István Laszlovszky; Béla Kiss; Attila Horváth; Gabriella Pásztor; Margó Kapás; István Gyertyán; Sándor Farkas; Robert B Innis; Christer Halldin; Balázs Gulyás
Journal:  Psychopharmacology (Berl)       Date:  2011-05-28       Impact factor: 4.530

7.  Mechanism of action of cariprazine.

Authors:  Stephen M Stahl
Journal:  CNS Spectr       Date:  2016-03-09       Impact factor: 3.790

8.  Cariprazine (RGH-188), a dopamine D(3) receptor-preferring, D(3)/D(2) dopamine receptor antagonist-partial agonist antipsychotic candidate: in vitro and neurochemical profile.

Authors:  Béla Kiss; Attila Horváth; Zsolt Némethy; Eva Schmidt; István Laszlovszky; Gyula Bugovics; Károly Fazekas; Katalin Hornok; Szabolcs Orosz; István Gyertyán; Eva Agai-Csongor; György Domány; Károly Tihanyi; Nika Adham; Zsolt Szombathelyi
Journal:  J Pharmacol Exp Ther       Date:  2010-01-21       Impact factor: 4.030

9.  Cariprazine in the treatment of schizophrenia: a proof-of-concept trial.

Authors:  Suresh Durgam; Robert E Litman; Kelly Papadakis; Dayong Li; György Németh; István Laszlovszky
Journal:  Int Clin Psychopharmacol       Date:  2016-03       Impact factor: 1.659

10.  Clinical pharmacology study of cariprazine (MP-214) in patients with schizophrenia (12-week treatment).

Authors:  Tadakatsu Nakamura; Tomoko Kubota; Atsushi Iwakaji; Masayoshi Imada; Margit Kapás; Yasunori Morio
Journal:  Drug Des Devel Ther       Date:  2016-01-14       Impact factor: 4.162

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  2 in total

Review 1.  Risk of Drug-induced Movement Disorders with Newer Antipsychotic Agents.

Authors:  George T Kannarkat; Stanley N Caroff; James F Morley
Journal:  Tremor Other Hyperkinet Mov (N Y)       Date:  2022-06-08

2.  Potentially inappropriate medications according to PRISCUS list and FORTA (Fit fOR The Aged) classification in geriatric psychiatry: a cross-sectional study.

Authors:  Martin Schulze Westhoff; Adrian Groh; Sebastian Schröder; Phileas Johannes Proskynitopoulos; Kirsten Jahn; Martin Klietz; Benjamin Krichevsky; Dirk O Stichtenoth; Felix Wedegärtner; Stefan Bleich; Helge Frieling; Johannes Heck
Journal:  J Neural Transm (Vienna)       Date:  2022-09-02       Impact factor: 3.850

  2 in total

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