Literature DB >> 34436928

Veliparib in Combination With Platinum-Based Chemotherapy for First-Line Treatment of Advanced Squamous Cell Lung Cancer: A Randomized, Multicenter Phase III Study.

Suresh S Ramalingam1, Silvia Novello2, Salih Zeki Guclu3,4, Dmitry Bentsion5, Zanete Zvirbule6, Maria Szilasi7, Reyes Bernabe8, Konstantinos Syrigos9, Lauren Averett Byers10, Philip Clingan11, Jair Bar12, Everett E Vokes13, Ramaswamy Govindan14, Martin Dunbar15, Peter Ansell15, Lei He15, Xin Huang15, Vasudha Sehgal15, Jaimee Glasgow15, Bruce A Bach15, Julien Mazieres16.   

Abstract

PURPOSE: Squamous non-small-cell lung cancer (sqNSCLC) is genetically complex with evidence of DNA damage. This phase III study investigated the efficacy and safety of poly (ADP-ribose) polymerase inhibitor veliparib in combination with conventional chemotherapy for advanced sqNSCLC (NCT02106546). PATIENTS AND METHODS: Patients age ≥ 18 years with untreated, advanced sqNSCLC were randomly assigned 1:1 to carboplatin and paclitaxel with veliparib 120 mg twice daily (twice a day) or placebo twice a day for up to six cycles. The primary end point was overall survival (OS) in the veliparib arm versus the control arm in current smokers, based on phase II findings. Archival tumor samples were provided for biomarker analysis using a 52-gene expression histology classifier (LP52).
RESULTS: Overall, 970 patients were randomly assigned to carboplatin and paclitaxel plus either veliparib (n = 486) or placebo (n = 484); 57% were current smokers. There was no significant OS benefit with veliparib in current smokers, with median OS 11.9 versus 11.1 months (hazard ratio [HR], 0.905; 95% CI, 0.744 to 1.101; P = .266). In the overall population, OS favored veliparib; median OS was 12.2 versus 11.2 months (HR, 0.853; 95% CI, 0.747 to 0.974), with no difference in progression-free survival (median 5.6 months per arm). In patients with biomarker-evaluable tumor samples (n = 360), OS favored veliparib in the LP52-positive population (median 14.0 v 9.6 months; HR, 0.66; 95% CI, 0.49 to 0.89), but favored placebo in the LP52-negative population (median 11.0 v 14.4 months; HR, 1.33; 95% CI, 0.95 to 1.86). No new safety signals were observed in the experimental arm.
CONCLUSION: In current smokers with advanced sqNSCLC, there was no therapeutic benefit of adding veliparib to first-line chemotherapy. The LP52 signature may identify a subgroup of patients likely to derive benefit from veliparib with chemotherapy.

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Year:  2021        PMID: 34436928      PMCID: PMC8577684          DOI: 10.1200/JCO.20.03318

Source DB:  PubMed          Journal:  J Clin Oncol        ISSN: 0732-183X            Impact factor:   44.544


  37 in total

1.  Nivolumab plus Ipilimumab in Lung Cancer with a High Tumor Mutational Burden.

Authors:  Matthew D Hellmann; Tudor-Eliade Ciuleanu; Adam Pluzanski; Jong Seok Lee; Gregory A Otterson; Clarisse Audigier-Valette; Elisa Minenza; Helena Linardou; Sjaak Burgers; Pamela Salman; Hossein Borghaei; Suresh S Ramalingam; Julie Brahmer; Martin Reck; Kenneth J O'Byrne; William J Geese; George Green; Han Chang; Joseph Szustakowski; Prabhu Bhagavatheeswaran; Diane Healey; Yali Fu; Faith Nathan; Luis Paz-Ares
Journal:  N Engl J Med       Date:  2018-04-16       Impact factor: 91.245

2.  SRY (sex determining region Y)-box2 (Sox2)/poly ADP-ribose polymerase 1 (Parp1) complexes regulate pluripotency.

Authors:  Yi-Shin Lai; Chia-Wei Chang; Kevin M Pawlik; Dewang Zhou; Matthew B Renfrow; Tim M Townes
Journal:  Proc Natl Acad Sci U S A       Date:  2012-02-23       Impact factor: 11.205

Review 3.  Current and Emergent Therapy Options for Advanced Squamous Cell Lung Cancer.

Authors:  Mark A Socinski; Coleman Obasaju; David Gandara; Fred R Hirsch; Philip Bonomi; Paul A Bunn; Edward S Kim; Corey J Langer; Ronald B Natale; Silvia Novello; Luis Paz-Ares; Maurice Pérol; Martin Reck; Suresh S Ramalingam; Craig H Reynolds; David R Spigel; Heather Wakelee; Nick Thatcher
Journal:  J Thorac Oncol       Date:  2017-11-23       Impact factor: 15.609

4.  PARP inhibitors synergize with gemcitabine by potentiating DNA damage in non-small-cell lung cancer.

Authors:  Yu Jiang; Hui Dai; Yang Li; Jun Yin; Shuliang Guo; Shiaw-Yih Lin; Daniel J McGrail
Journal:  Int J Cancer       Date:  2018-09-24       Impact factor: 7.396

5.  Smoking History Predicts Sensitivity to PARP Inhibitor Veliparib in Patients with Advanced Non-Small Cell Lung Cancer.

Authors:  Martin Reck; Normand Blais; Erzsebet Juhasz; Vera Gorbunova; C Michael Jones; Laszlo Urban; Sergey Orlov; Fabrice Barlesi; Ebenezer Kio; Ulrich Keilholz; Qin Qin; Jiang Qian; Caroline Nickner; Juliann Dziubinski; Hao Xiong; Rajendar K Mittapalli; Martin Dunbar; Peter Ansell; Lei He; Mark McKee; Vincent Giranda; Suresh S Ramalingam
Journal:  J Thorac Oncol       Date:  2017-04-29       Impact factor: 15.609

6.  Randomized, Placebo-Controlled, Phase II Study of Veliparib in Combination with Carboplatin and Paclitaxel for Advanced/Metastatic Non-Small Cell Lung Cancer.

Authors:  Suresh S Ramalingam; Normand Blais; Julien Mazieres; Martin Reck; C Michael Jones; Erzsebet Juhasz; Laszlo Urban; Sergey Orlov; Fabrice Barlesi; Ebenezer Kio; Ulrich Keiholz; Qin Qin; Jiang Qian; Caroline Nickner; Juliann Dziubinski; Hao Xiong; Peter Ansell; Mark McKee; Vincent Giranda; Vera Gorbunova
Journal:  Clin Cancer Res       Date:  2016-10-10       Impact factor: 12.531

Review 7.  The PARP superfamily.

Authors:  Jean-Christophe Amé; Catherine Spenlehauer; Gilbert de Murcia
Journal:  Bioessays       Date:  2004-08       Impact factor: 4.345

8.  A Phase I Clinical Trial of the Poly(ADP-ribose) Polymerase Inhibitor Veliparib and Weekly Topotecan in Patients with Solid Tumors.

Authors:  Andrea E Wahner Hendrickson; Michael E Menefee; Lynn C Hartmann; Harry J Long; Donald W Northfelt; Joel M Reid; Felix Boakye-Agyeman; Olumide Kayode; Karen S Flatten; Maria I Harrell; Elizabeth M Swisher; Guy G Poirier; Daniel Satele; Jake Allred; Janet L Lensing; Alice Chen; Jiuping Ji; Yiping Zang; Charles Erlichman; Paul Haluska; Scott H Kaufmann
Journal:  Clin Cancer Res       Date:  2017-11-14       Impact factor: 12.531

9.  In silico characterization of the family of PARP-like poly(ADP-ribosyl)transferases (pARTs).

Authors:  Helge Otto; Pedro A Reche; Fernando Bazan; Katharina Dittmar; Friedrich Haag; Friedrich Koch-Nolte
Journal:  BMC Genomics       Date:  2005-10-04       Impact factor: 3.969

10.  Genomic and Molecular Landscape of DNA Damage Repair Deficiency across The Cancer Genome Atlas.

Authors:  Theo A Knijnenburg; Linghua Wang; Michael T Zimmermann; Nyasha Chambwe; Galen F Gao; Andrew D Cherniack; Huihui Fan; Hui Shen; Gregory P Way; Casey S Greene; Yuexin Liu; Rehan Akbani; Bin Feng; Lawrence A Donehower; Chase Miller; Yang Shen; Mostafa Karimi; Haoran Chen; Pora Kim; Peilin Jia; Eve Shinbrot; Shaojun Zhang; Jianfang Liu; Hai Hu; Matthew H Bailey; Christina Yau; Denise Wolf; Zhongming Zhao; John N Weinstein; Lei Li; Li Ding; Gordon B Mills; Peter W Laird; David A Wheeler; Ilya Shmulevich; Raymond J Monnat; Yonghong Xiao; Chen Wang
Journal:  Cell Rep       Date:  2018-04-03       Impact factor: 9.423

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  5 in total

1.  Synergistic Effects of A Combined Treatment of Glioblastoma U251 Cells with An Anti-miR-10b-5p Molecule and An AntiCancer Agent Based on 1-(3',4',5'-Trimethoxyphenyl)-2-Aryl-1H-Imidazole Scaffold.

Authors:  Matteo Zurlo; Romeo Romagnoli; Paola Oliva; Jessica Gasparello; Alessia Finotti; Roberto Gambari
Journal:  Int J Mol Sci       Date:  2022-05-26       Impact factor: 6.208

Review 2.  [DNA Damage Repair System and Antineoplastic Agents in Lung Cancer].

Authors:  Linlin Zhang; Fanlu Meng; Diansheng Zhong
Journal:  Zhongguo Fei Ai Za Zhi       Date:  2022-06-20

Review 3.  Application of Approved Cisplatin Derivatives in Combination Therapy against Different Cancer Diseases.

Authors:  Dobrina Tsvetkova; Stefka Ivanova
Journal:  Molecules       Date:  2022-04-11       Impact factor: 4.927

Review 4.  Everything Comes with a Price: The Toxicity Profile of DNA-Damage Response Targeting Agents.

Authors:  Federica Martorana; Leandro Apolinario Da Silva; Cristiana Sessa; Ilaria Colombo
Journal:  Cancers (Basel)       Date:  2022-02-14       Impact factor: 6.639

Review 5.  PARP Inhibitors: Clinical Limitations and Recent Attempts to Overcome Them.

Authors:  Dongha Kim; Hye Jin Nam
Journal:  Int J Mol Sci       Date:  2022-07-29       Impact factor: 6.208

  5 in total

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