Literature DB >> 34221222

Methimazole in the Treatment of Melasma: A Clinical and Dermascopic Study.

Azza Farag1,2,3,4,5, Mostafa Hammam1,2,3,4,5, Nada Alnaidany1,2,3,4,5, Eman Badr1,2,3,4,5, Mustafa Elshaib1,2,3,4,5, Aliaa El-Swah1,2,3,4,5, Wafaa Shehata1,2,3,4,5.   

Abstract

BACKGROUND: Melasma is a chronic hypermelanotic disorder that is challenging to treat; no single effective therapeutic agent for it has been discovered. Methimazole, an oral antithyroid drug, has a skin depigmenting effect when used topically.
OBJECTIVE: We sought to evaluate the efficacy and safety of methimazole, applied during microneedling sessions and additional topical use in between sessions, for the treatment of melasma.
METHODS: This split-face study included 30 Egyptian patients with melasma, each of whom received 12 microneedling sessions once per week for 12 weeks followed by topical methimazole on the right side of face and placebo on the left side. In between the sessions, topical methimazole 5% cream was applied twice per day on the right side and placebo on the left side. Assessments were performed using the Hemi-melasma Area and Severity Index (hemi-MASI) percentage of improvement, patient satisfaction, dermoscopy, and thyroid-stimulating hormone (TSH) serum levels.
RESULTS: There were significant clinical and dermoscopic improvements; hemi-MASI scores on the methimazole-treated right sides were decreased (p<0.001). The percent of hemi-MASI score improvement was significantly associated with the malar pattern (p=0.031) and epidermal type (p=0.04) of melasma. About 70 percent of our studied patients reported being satisfied with their treatment response (7% excellent, 33% good, 30% fair). No significant local or systemic side effects were observed. Pre- and posttreatment serum TSH levels were within the normal range in all treated cases.
CONCLUSIONS: Methimazole has the potential to be a safe and promising therapeutic agent for the treatment of melasma via dermapen-delivered microneedling sessions with topical use in between sessions.
Copyright © 2021. Matrix Medical Communications. All rights reserved.

Entities:  

Keywords:  Methimazole; melasma; microneedling

Year:  2021        PMID: 34221222      PMCID: PMC8211339     

Source DB:  PubMed          Journal:  J Clin Aesthet Dermatol        ISSN: 1941-2789


  15 in total

1.  Depigmentation of brown Guinea pig skin by topical application of methimazole.

Authors:  Behrooz Kasraee
Journal:  J Invest Dermatol       Date:  2002-01       Impact factor: 8.551

2.  Methimazole is an inhibitor of melanin synthesis in cultured B16 melanocytes.

Authors:  Behrooz Kasraee; Ambros Hügin; Christian Tran; Olivier Sorg; Jean-Hilaire Saurat
Journal:  J Invest Dermatol       Date:  2004-05       Impact factor: 8.551

Review 3.  Clinical review 12: The use and misuse of the sensitive thyrotropin assays.

Authors:  J T Nicoloff; C A Spencer
Journal:  J Clin Endocrinol Metab       Date:  1990-09       Impact factor: 5.958

4.  Effect of methimazole on the activity of mushroom tyrosinase.

Authors:  A Andrawis; V Kahn
Journal:  Biochem J       Date:  1986-04-01       Impact factor: 3.857

5.  The efficacy and safety of topical 5% methimazole vs 4% hydroquinone in the treatment of melasma: A randomized controlled trial.

Authors:  Mehdi Gheisari; Sahar Dadkhahfar; Elham Olamaei; Hamid Reza Moghimi; Nasim Niknejad; Niloufar Najar Nobari
Journal:  J Cosmet Dermatol       Date:  2019-05-17       Impact factor: 2.696

6.  Evaluation of the efficacy and safety of combinations of hydroquinone, glycolic acid, and hyaluronic acid in the treatment of melasma.

Authors:  Zeinab A Ibrahim; Shereen F Gheida; Gamal M El Maghraby; Zeinab E Farag
Journal:  J Cosmet Dermatol       Date:  2015-04-06       Impact factor: 2.696

7.  Localized intradermal microinjection of tranexamic acid for treatment of melasma in Asian patients: a preliminary clinical trial.

Authors:  Ji Ho Lee; Jong Gap Park; Sook Hee Lim; Jo Yong Kim; Kun Young Ahn; Mi-Yeon Kim; Young Min Park
Journal:  Dermatol Surg       Date:  2006-05       Impact factor: 3.398

8.  Safety of topical methimazole for the treatment of melasma. Transdermal absorption, the effect on thyroid function and cutaneous adverse effects.

Authors:  B Kasraee; G H Safaee Ardekani; A Parhizgar; F Handjani; G R Omrani; M Samani; M Nikbakhsh; N Tanideh; A Eshraghian; O Sorg; J H Saurat
Journal:  Skin Pharmacol Physiol       Date:  2008-07-31       Impact factor: 3.479

9.  Therapeutical approaches in melasma.

Authors:  Francesca Prignano; Jean-Paul Ortonne; Gionata Buggiani; Torello Lotti
Journal:  Dermatol Clin       Date:  2007-07       Impact factor: 3.478

10.  A Randomised, Open-label, Comparative Study of Tranexamic Acid Microinjections and Tranexamic Acid with Microneedling in Patients with Melasma.

Authors:  Leelavathy Budamakuntla; Eswari Loganathan; Deepak Hurkudli Suresh; Sharavana Shanmugam; Shwetha Suryanarayan; Aparna Dongare; Lakshmi Dammaningala Venkataramiah; Namitha Prabhu
Journal:  J Cutan Aesthet Surg       Date:  2013-07
View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.