Literature DB >> 34117788

Monoacylglycerol Lipase Inhibition in Tourette Syndrome: A 12-Week, Randomized, Controlled Study.

Kirsten R Müller-Vahl1, Carolin Fremer1, Chan Beals2, Jelena Ivkovic3, Henrik Loft3, Christoph Schindler4.   

Abstract

BACKGROUND: Modulation of the endocannabinoid system via monoacylglycerol lipase inhibition with Lu AG06466 (formerly known as ABX-1431) has previously been shown to reduce tics in patients with Tourette syndrome.
OBJECTIVE: The aim of this study was to evaluate the efficacy and safety of Lu AG06466 in reducing tics, premonitory urges, and comorbidities in patients with Tourette syndrome.
METHODS: This was a 12-week, multicenter, randomized, placebo-controlled, double-blind clinical trial of Lu AG06466 given at two dose levels in 49 adults with Tourette syndrome.
RESULTS: Both treatment groups showed improvement on the Total Tic Score of the Yale Global Tic Severity Scale; the mean (95% CI) treatment difference at week 8 of 3.0 (0.1, 5.9) (P = 0.043) favored placebo. No significant differences were seen for other endpoints assessing changes in tic severity, premonitory urges, quality of life, and common psychiatric comorbidities. Treatment with Lu-AG06466 was generally safe.
CONCLUSIONS: There was no evidence that Lu AG06466 has efficacy in suppressing tics.
© 2021 The Authors. Movement Disorders published by Wiley Periodicals LLC on behalf of International Parkinson and Movement Disorder Society. © 2021 The Authors. Movement Disorders published by Wiley Periodicals LLC on behalf of International Parkinson and Movement Disorder Society.

Entities:  

Keywords:  ABX-1431; Lu AG06466; Tourette syndrome; endocannabinoid modulator; tics

Mesh:

Substances:

Year:  2021        PMID: 34117788     DOI: 10.1002/mds.28681

Source DB:  PubMed          Journal:  Mov Disord        ISSN: 0885-3185            Impact factor:   10.338


  8 in total

1.  Mechanistic Modeling of Monoglyceride Lipase Covalent Modification Elucidates the Role of Leaving Group Expulsion and Discriminates Inhibitors with High and Low Potency.

Authors:  Francesca Galvani; Laura Scalvini; Silvia Rivara; Alessio Lodola; Marco Mor
Journal:  J Chem Inf Model       Date:  2022-05-17       Impact factor: 6.162

2.  Medical Cannabis for Gilles de la Tourette Syndrome: An Open-Label Prospective Study.

Authors:  Saar Anis; Corinne Zalomek; Amos D Korczyn; Alina Rosenberg; Nir Giladi; Tanya Gurevich
Journal:  Behav Neurol       Date:  2022-03-09       Impact factor: 3.342

3.  Endocannabinoid Modulation Using Monoacylglycerol Lipase Inhibition in Tourette Syndrome: A Phase 1 Randomized, Placebo-Controlled Study.

Authors:  Kirsten R Müller-Vahl; Carolin Fremer; Chan Beals; Jelena Ivkovic; Henrik Loft; Christoph Schindler
Journal:  Pharmacopsychiatry       Date:  2021-11-30       Impact factor: 2.544

Review 4.  Tourette syndrome research highlights from 2021.

Authors:  Andreas Hartmann; Per Andrén; Cyril Atkinson-Clement; Virginie Czernecki; Cécile Delorme; Nanette Marinette Debes; Natalia Szejko; Keisuke Ueda; Kevin Black
Journal:  F1000Res       Date:  2022-06-29

5.  A potent and selective inhibitor for the modulation of MAGL activity in the neurovasculature.

Authors:  Alicia M Kemble; Benoit Hornsperger; Iris Ruf; Hans Richter; Jörg Benz; Bernd Kuhn; Dominik Heer; Matthias Wittwer; Britta Engelhardt; Uwe Grether; Ludovic Collin
Journal:  PLoS One       Date:  2022-09-09       Impact factor: 3.752

6.  Cannabinoid signaling modulation through JZL184 restores key phenotypes of a mouse model for Williams-Beuren syndrome.

Authors:  Alba Navarro-Romero; Lorena Galera-López; Paula Ortiz-Romero; Alberto Llorente-Ovejero; Lucía de Los Reyes-Ramírez; Iker Bengoetxea de Tena; Anna Garcia-Elias; Aleksandra Mas-Stachurska; Marina Reixachs-Solé; Antoni Pastor; Rafael de la Torre; Rafael Maldonado; Begoña Benito; Eduardo Eyras; Rafael Rodríguez-Puertas; Victoria Campuzano; Andres Ozaita
Journal:  Elife       Date:  2022-10-11       Impact factor: 8.713

Review 7.  Tourette Syndrome Treatment Updates: a Review and Discussion of the Current and Upcoming Literature.

Authors:  Jessica Frey; Irene A Malaty
Journal:  Curr Neurol Neurosci Rep       Date:  2022-02-02       Impact factor: 6.030

Review 8.  European clinical guidelines for Tourette syndrome and other tic disorders: summary statement.

Authors:  Kirsten R Müller-Vahl; Natalia Szejko; Cara Verdellen; Veit Roessner; Pieter J Hoekstra; Andreas Hartmann; Danielle C Cath
Journal:  Eur Child Adolesc Psychiatry       Date:  2021-07-10       Impact factor: 4.785

  8 in total

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