Literature DB >> 34088513

Pazopanib based oral metronomic therapy for platinum resistant/refractory epithelial ovarian cancer: A phase II, open label, randomized, controlled trial.

Aparna Sharma1, Mayank Singh1, Ravi Chauhan1, Prabhat Singh Malik1, Sachin Khurana1, Sandeep Mathur2, Sunesh Kumar3, Vishnubhatla Sreenivas4, Lalit Kumar5.   

Abstract

BACKGROUND: Treatment of patients with platinum resistant/refractory epithelial ovarian cancer (EOC) is an unmet need. We evaluated the role of oral metronomic therapy in this setting. PATIENTS AND METHODS: Between October 2017 and September 2019 seventy five patients with platinum resistant/refractory EOC were enrolled. Patients received oral etoposide (50 mg, day 1 to 14, cyclophosphamide 50 mg, day 1 to 28, every 4 weeks (Arm A, n = 38). Patients in Arm- B (n = 37) received Pazopanib (400 mg once daily) in addition to etoposide and cyclophosphamide. Quality of life (QoL) was evaluated using the EORTC questionnaire. Serum VEGF and PDGF were estimated at baseline, after 3rd and 6th cycle. The primary endpoint was progression free survival (PFS). Secondary endpoints were overall survival (OS), toxicity and QoL.
RESULTS: Patients characteristics were well matched. Median PFS was higher in arm B, 5.1 months (95% CI 3.13 to10.33) compared to 3.4 months (95% CI 3.0 to 6.53) in arm A, p = 0.045. Median OS has 'not reached' in Arm B compared to 11.2 months (95% CI, 5.66 - not reached) in arm A, p = 0.032. Therapy was tolerated well; oral mucositis (p = 0.36) and fatigue (p = 0.08) being more in arm B. QoL assessment revealed modest improvement in 'symptom scales' in Arm B. Serum VEGF and PDGF levels decreased with therapy in both arms (Arm A-p < 0.0001, Arm B-p < 0.016).
CONCLUSION: Addition of pazopanib to etoposide and cyclophosphamide could be a novel oral combination for metronomic therapy for platinum resistant/refractory EOC. TRIAL REGISTRATION: CTRI/2017/10/010219.
Copyright © 2021 Elsevier Inc. All rights reserved.

Entities:  

Keywords:  Adverse effects; PDGF; Pazopanib; Progression free survival; Quality of life; VEGF

Mesh:

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Year:  2021        PMID: 34088513     DOI: 10.1016/j.ygyno.2021.05.025

Source DB:  PubMed          Journal:  Gynecol Oncol        ISSN: 0090-8258            Impact factor:   5.482


  3 in total

1.  Effectiveness and toxicity of metronomic oral cyclophosphamide for recurrent or platinum-refractory ovarian cancer: A meta-analysis.

Authors:  Lili Huang; Ting Jiang; Pengcheng Li; Jie Zhang; Xing Luo; Fang Yang; Tao Ren; Ke Xu
Journal:  Heliyon       Date:  2022-08-24

2.  Pazopanib restricts small cell lung cancer proliferation via reactive oxygen species-mediated endoplasmic reticulum stress.

Authors:  Yue Li; Chen Chen; Hai-Lin Liu; Chen-Guang Li; Zhen-Fa Zhang; Chang-Li Wang
Journal:  Thorac Cancer       Date:  2022-07-21       Impact factor: 3.223

3.  Phase II study of sodium valproate in combination with oral etoposide in platinum-resistant ovarian cancer.

Authors:  Thejeswar Nakka; Luxitaa Goenka; Biswajit Dubashi; Smita Kayal; Jayanthi Mathaiyan; Deepak Barathi; Narendran Krishnamoorthy; Divya Bala Thumaty; Sindhu Dahagama; Prasanth Ganesan
Journal:  Med Oncol       Date:  2022-09-29       Impact factor: 3.738

  3 in total

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