Literature DB >> 34074829

Outcomes of Sequential Therapy With Tenofovir Alafenamide After Long-term Entecavir.

Mindie H Nguyen1, Masanori Atsukawa2, Toru Ishikawa3, Satoshi Yasuda4, Keisuke Yokohama5, Huy N Trinh6, Taeang Arai2, Shinya Fukunishi7, Eiichi Ogawa8, Yao-Chun Hsu9, Mayumi Maeda1, Hansen Dang1, Cheng-Hao Tseng9, Hirokazu Takahashi10,11, Dae Won Jun12, Tsunamasa Watanabe13, Makoto Chuma14, Akito Nozaki14, Norifumi Kawada15, Ramsey Cheung1,16, Masaru Enomoto15, Koichi Takaguchi17, Hidenori Toyoda4.   

Abstract

INTRODUCTION: Entecavir (ETV) and tenofovir alafenamide (TAF) are both first-line hepatitis B virus (HBV) therapies, but ETV-to-TAF switch outcome data are limited. We aimed to assess outcomes up to 96 weeks after ETV-to-TAF switch.
METHODS: ETV-treated (≥12 months) chronic hepatitis B patients switched to TAF in routine practice at 15 centers (United States, Korea, Japan, and Taiwan) were included. Primary outcome was complete viral suppression (CVS) rate (HBV DNA <20 IU/mL).
RESULTS: We analyzed 425 eligible patients (mean age 60.7 ± 13.2 years, 60% men, 90.8% Asian, 20.7% with diabetes, 27% with hypertension, 14.8% with cirrhosis, 8.3% with hepatocellular carcinoma, and mean ETV duration before switch 6.16 ± 3.17 years). The mean baseline estimated glomerular filtration rate (eGFR) was 89 ± 19 (chronic kidney disease [CKD] stages: 55.6% stage 1, 35.7% stage 2, and 8.8% stages 3-5). CVS rate increased from 91.90% at switch (from 90.46% 24 weeks before switch) to 95.57% and 97.21% at 48 and 96 weeks after (P = 0.03 and 0.02, respectively). Over the 96 weeks after switch, mean HBV DNA (P < 0.001) but not alanine aminotransferase or CKD stage decreased. Between switch and 96-week follow-up, 11% (26/235) of CKD stage 1 patients migrated to stage 2 and 8% (12/151) of stage 2 patients to stages 3-5, whereas 18% (27/151) from stage 2 to 1, and 19% (7/37) from stages 3-5 to 2. On multivariable generalized estimated equation analysis adjusted for age, sex, hypertension, diabetes, and cirrhosis, baseline eGFR, age (P < 0.001), and CKD stages 2 and 3-5 (vs 1) (both P < 0.001) were associated with lower follow-up eGFR. DISCUSSION: After an average of 6 years on ETV, CVS increased from 91.9% at TAF switch to 97.2% at 96 weeks later.
Copyright © 2021 by The American College of Gastroenterology.

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Year:  2021        PMID: 34074829     DOI: 10.14309/ajg.0000000000001157

Source DB:  PubMed          Journal:  Am J Gastroenterol        ISSN: 0002-9270            Impact factor:   10.864


  3 in total

1.  First-In-Human Study on Pharmacokinetics, Safety, and Tolerability of Single and Multiple Escalating Doses of Hepenofovir, a Novel Hepatic Targeting Prodrug of Tenofovir in Healthy Chinese Subjects.

Authors:  Hong Zhang; Lei Gao; Jinfeng Lou; Min Wu; Hong Chen; Lizhi Yang; Jingrui Liu; Xiaoxue Zhu; Xiaojiao Li; Cuiyun Li; Meng Wang; Chengjiao Liu; Weibo Guo; Yuan Wang; Zhongqiang Gao; Lei Han; Daidi Wang; Weili Jin; Yanhua Ding
Journal:  Front Pharmacol       Date:  2022-05-19       Impact factor: 5.988

Review 2.  Review article: switching patients with chronic hepatitis B to tenofovir alafenamide-a review of current data.

Authors:  Young-Suk Lim; Wai-Kay Seto; Masayuki Kurosaki; Scott Fung; Jia-Horng Kao; Jinlin Hou; Stuart C Gordon; John F Flaherty; Leland J Yee; Yang Zhao; Kosh Agarwal; Pietro Lampertico
Journal:  Aliment Pharmacol Ther       Date:  2022-02-17       Impact factor: 9.524

3.  Switching to tenofovir alafenamide versus continued therapy in chronic hepatitis B patients who were treated with entecavir: A prospective, multicenter, randomized controlled study.

Authors:  Kosuke Sato; Jun Inoue; Takehiro Akahane; Tomoo Kobayashi; Shuichi Sato; Norihiro Kisara; Masashi Ninomiya; Tomoaki Iwata; Akitoshi Sano; Mio Tsuruoka; Masazumi Onuki; Atsushi Masamune
Journal:  Medicine (Baltimore)       Date:  2022-09-30       Impact factor: 1.817

  3 in total

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