Literature DB >> 34016181

Strontium ranelate promotes chondrogenesis through inhibition of the Wnt/β-catenin pathway.

Hao Yu1,2, Yan Liu1,2, Xiangwen Yang1,2, Jiajing He1,2, Fan Zhang2,3, Qun Zhong1,2, Xiaojing Guo4,5.   

Abstract

BACKGROUND: Cartilage regeneration is a key step in functional reconstruction for temporomandibular joint osteoarthritis (TMJ-OA) but is a difficult issue to address. Strontium ranelate (SrR) is an antiosteoporosis drug that has been proven to affect OA in recent years, but its effect on chondrogenesis and the underlying mechanism are still unclear.
METHODS: Bone mesenchymal stem cells (BMSCs) from Sprague-Dawley (SD) rats were induced in chondrogenic differentiation medium with or without SrR, XAV-939, and LiCl. CCK-8 assays were used to examine cell proliferation, and alcian blue staining, toluidine blue staining, immunofluorescence, and PCR analysis were performed. Western blot (WB) analyses were used to assess chondrogenic differentiation of the cells. For an in vivo study, 30 male SD rats with cartilage defects on both femoral condyles were used. The defect sites were not filled, filled with silica nanosphere plus gelatine-methacryloyl (GelMA), or filled with SrR-loaded silica nanosphere plus GelMA. After 3 months of healing, paraffin sections were made, and toluidine blue staining, safranin O/fast green staining, and immunofluorescent or immunohistochemical staining were performed for histological evaluation. The data were analyzed by SPSS 26.0 software.
RESULTS: Low concentrations of SrR did not inhibit cell proliferation, and the cells treated with SrR (0.25 mmol/L) showed stronger chondrogenesis than the control. XAV-939, an inhibitor of β-catenin, significantly promoted chondrogenesis, and SrR did not suppress this effect, while LiCl, an agonist of β-catenin, strongly suppressed chondrogenesis, and SrR reversed this inhibitory effect. In vivo study showed a significantly better cartilage regeneration and a lower activation level of β-catenin by SrR-loaded GelMA than the other treatments.
CONCLUSION: SrR could promote BMSCs chondrogenic differentiation by inhibiting the Wnt/β-catenin signaling pathway and accelerate cartilage regeneration in rat femoral condyle defects.

Entities:  

Keywords:  BMSCs; Cartilage regeneration; Chondrogenesis; Strontium ranelate; Wnt/β-catenin pathway

Year:  2021        PMID: 34016181     DOI: 10.1186/s13287-021-02372-z

Source DB:  PubMed          Journal:  Stem Cell Res Ther        ISSN: 1757-6512            Impact factor:   6.832


  39 in total

1.  Prevalence and clinical signs of degenerative temporomandibular joint changes validated by magnetic resonance imaging in a non-patient group.

Authors:  Olaf Bernhardt; Reiner Biffar; Thomas Kocher; Georg Meyer
Journal:  Ann Anat       Date:  2007       Impact factor: 2.698

2.  Minimally Invasive Approach for Diagnosing TMJ Osteoarthritis.

Authors:  B Shoukri; J C Prieto; A Ruellas; M Yatabe; J Sugai; M Styner; H Zhu; C Huang; B Paniagua; S Aronovich; L Ashman; E Benavides; P de Dumast; N T Ribera; C Mirabel; L Michoud; Z Allohaibi; M Ioshida; L Bittencourt; L Fattori; L R Gomes; L Cevidanes
Journal:  J Dent Res       Date:  2019-07-24       Impact factor: 6.116

3.  Strontium ranelate reduces the urinary level of cartilage degradation biomarker CTX-II in postmenopausal women.

Authors:  Peter Alexandersen; M A Karsdal; Per Qvist; J-Y Reginster; Claus Christiansen
Journal:  Bone       Date:  2006-09-28       Impact factor: 4.398

Review 4.  Strontium ranelate, a promising disease modifying osteoarthritis drug.

Authors:  Weiyu Han; Shicai Fan; Xiaochun Bai; Changhai Ding
Journal:  Expert Opin Investig Drugs       Date:  2017-01-25       Impact factor: 6.206

Review 5.  Current understanding of pathogenesis and treatment of TMJ osteoarthritis.

Authors:  X D Wang; J N Zhang; Y H Gan; Y H Zhou
Journal:  J Dent Res       Date:  2015-03-05       Impact factor: 6.116

Review 6.  Osteoarthritis: an update with relevance for clinical practice.

Authors:  Johannes W J Bijlsma; Francis Berenbaum; Floris P J G Lafeber
Journal:  Lancet       Date:  2011-06-18       Impact factor: 79.321

Review 7.  Stem Cells for Temporomandibular Joint Repair and Regeneration.

Authors:  Shipin Zhang; Adrian U J Yap; Wei Seong Toh
Journal:  Stem Cell Rev Rep       Date:  2015-10       Impact factor: 5.739

8.  Disease-modifying effect of strontium ranelate in a subset of patients from the Phase III knee osteoarthritis study SEKOIA using quantitative MRI: reduction in bone marrow lesions protects against cartilage loss.

Authors:  Jean-Pierre Pelletier; Camille Roubille; Jean-Pierre Raynauld; François Abram; Marc Dorais; Philippe Delorme; Johanne Martel-Pelletier
Journal:  Ann Rheum Dis       Date:  2013-12-02       Impact factor: 19.103

Review 9.  What about strontium ranelate in osteoarthritis? Doubts and securities.

Authors:  Sara Tenti; Sara Cheleschi; Giacomo Maria Guidelli; Mauro Galeazzi; Antonella Fioravanti
Journal:  Mod Rheumatol       Date:  2014-03-19       Impact factor: 3.023

10.  Efficacy and safety of strontium ranelate in the treatment of knee osteoarthritis: results of a double-blind, randomised placebo-controlled trial.

Authors:  Jean-Yves Reginster; Janusz Badurski; Nicholas Bellamy; William Bensen; Roland Chapurlat; Xavier Chevalier; Claus Christiansen; Harry Genant; Federico Navarro; Evgeny Nasonov; Philip N Sambrook; Timothy D Spector; Cyrus Cooper
Journal:  Ann Rheum Dis       Date:  2012-11-01       Impact factor: 19.103

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  5 in total

Review 1.  Strontium Functionalized in Biomaterials for Bone Tissue Engineering: A Prominent Role in Osteoimmunomodulation.

Authors:  Jiaqian You; Yidi Zhang; Yanmin Zhou
Journal:  Front Bioeng Biotechnol       Date:  2022-07-06

2.  Wnt/β-catenin signaling pathway is activated in the progress of mandibular condylar cartilage degeneration and subchondral bone loss induced by overloaded functional orthopedic force (OFOF).

Authors:  Zijing He; Meixi Liu; Qiang Zhang; Yihong Tian; Lingzhi Wang; Xiao Yan; Dapeng Ren; Xiao Yuan
Journal:  Heliyon       Date:  2022-10-01

3.  The anti-inflammation effect of strontium ranelate on rat chondrocytes with or without IL-1β in vitro.

Authors:  Hao Yu; Yan Liu; Xiangwen Yang; Jiajing He; Qun Zhong; Xiaojing Guo
Journal:  Exp Ther Med       Date:  2022-01-07       Impact factor: 2.447

4.  Dickkopf‑3 and β‑catenin play opposite roles in the Wnt/β‑catenin pathway during the abnormal subchondral bone formation of human knee osteoarthritis.

Authors:  Xuegang Liang; Qunhua Jin; Xiaochun Yang; Wenhui Jiang
Journal:  Int J Mol Med       Date:  2022-02-09       Impact factor: 4.101

5.  3D printing polylactic acid polymer-bioactive glass loaded with bone cement for bone defect in weight-bearing area.

Authors:  Yurun Ding; Xiaolin Liu; Jue Zhang; Zhuocheng Lv; Xiangchao Meng; Zhiguo Yuan; Teng Long; You Wang
Journal:  Front Bioeng Biotechnol       Date:  2022-07-25
  5 in total

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