Literature DB >> 33977088

What Can Be Done to Solve the Unmet Clinical Need of Hepatocellular Carcinoma Patients following Lenvatinib Failure?

Atsushi Hiraoka1, Takashi Kumada2, Toshifumi Tada3, Kazuya Kariyama4, Joji Tani5, Shinya Fukunishi6, Masanori Atsukawa7, Masashi Hirooka8, Kunihiko Tsuji9, Toru Ishikawa10, Koichi Takaguchi11, Ei Itobayashi12, Kazuto Tajiri13, Noritomo Shimada14, Hiroshi Shibata15, Hironori Ochi16, Kazuhito Kawata17, Satoshi Yasuda18, Hidenori Toyoda18, Hideko Ohama6, Kazuhiro Nouso4, Akemi Tsutsui11, Takuya Nagano11, Norio Itokawa7, Korenobu Hayama7, Taeang Arai7, Michitaka Imai10, Yohei Koizumi8, Shinichiro Nakamura3, Kouji Joko16, Kojiro Michitaka1, Yoichi Hiasa8, Masatoshi Kudo19.   

Abstract

BACKGROUND/AIM: An effective postprogression treatment of lenvatinib (LEN) against unresectable hepatocellular carcinoma (u-HCC) has not been established. We aimed to elucidate the clinical role of continuing LEN beyond progression of disease (PD).
METHODS: From March 2018 to October 2020, 99 u-HCC patients, in whom PD was confirmed (male:female = 78:21, median age 72 years, Child-Pugh A = 99, Barcelona Clinic Liver Cancer stage A:B:C = 2:43:54, LEN as first-line = 55), were enrolled (stopped LEN at PD [A group], n = 26; continued LEN beyond PD [B group], n = 73). Radiological response was evaluated with RECIST 1.1. Clinical features and prognostic factors for overall survival (OS) were retrospectively investigated using inverse probability weighting (IPW) calculated by propensity score.
RESULTS: Median time to progression, best response, and modified albumin-bilirubin grade (mALBI) at both baseline and PD did not show significant difference between the groups. Postprogression treatment in the A group was best supportive care in 17, sorafenib in 4, regorafenib in 3, ramucirumab in 1, and hepatic arterial infusion chemotherapy in 1. After adjusting with IPW, the B group showed better prognosis in regard to OS after PD and OS after introducing LEN than the A group (10.8/19.6 vs. 5.8/11.2 months, p < 0.001, respectively). In IPW-adjusted Cox hazard multivariate analysis, significant prognostic factors for OS after PD were mALBI 2b/3 at PD (HR 1.983, p = 0.021), decline of Eastern Cooperative Oncology Group performance status (ECOG PS) from baseline at PD (HR 3.180, p < 0.001), elevated alpha-fetoprotein (≥100 ng/mL) at introducing LEN (HR 2.511, p = 0.004), appearance of new extrahepatic metastasis (HR 2.396, p = 0.006), positive for hand-foot skin reaction (HFSR) before PD (any grade) (HR 0.292, p < 0.001), and continuing LEN beyond PD (HR 0.297, p < 0.001).
CONCLUSION: When ECOG PS and hepatic reserve function permit, continuing LEN treatment beyond PD, especially in u-HCC patients showed HFSR during LEN treatment, might be a good therapeutic option, at least until a more effective drug as a postprogression treatment after LEN failure is developed.
Copyright © 2021 by S. Karger AG, Basel.

Entities:  

Keywords:  Beyond progression of disease; Hand-foot skin reaction; Hepatocellular carcinoma; Lenvatinib; Postprogression treatment

Year:  2021        PMID: 33977088      PMCID: PMC8077500          DOI: 10.1159/000513355

Source DB:  PubMed          Journal:  Liver Cancer        ISSN: 1664-5553            Impact factor:   11.740


  45 in total

1.  Intraindividual comparison of gadoxetate disodium-enhanced MR imaging and 64-section multidetector CT in the Detection of hepatocellular carcinoma in patients with cirrhosis.

Authors:  Michele Di Martino; Daniele Marin; Antonino Guerrisi; Mahbubeh Baski; Francesca Galati; Massimo Rossi; Stefania Brozzetti; Raffaele Masciangelo; Roberto Passariello; Carlo Catalano
Journal:  Radiology       Date:  2010-09       Impact factor: 11.105

2.  Adjusted Kaplan-Meier estimator and log-rank test with inverse probability of treatment weighting for survival data.

Authors:  Jun Xie; Chaofeng Liu
Journal:  Stat Med       Date:  2005-10-30       Impact factor: 2.373

Review 3.  General Rules for the Clinical and Pathological Study of Primary Liver Cancer, Nationwide Follow-Up Survey and Clinical Practice Guidelines: The Outstanding Achievements of the Liver Cancer Study Group of Japan.

Authors:  Masatoshi Kudo; Masayuki Kitano; Toshiharu Sakurai; Naoshi Nishida
Journal:  Dig Dis       Date:  2015-10-21       Impact factor: 2.404

4.  Transection of the oesophagus for bleeding oesophageal varices.

Authors:  R N Pugh; I M Murray-Lyon; J L Dawson; M C Pietroni; R Williams
Journal:  Br J Surg       Date:  1973-08       Impact factor: 6.939

5.  Important Clinical Factors in Sequential Therapy Including Lenvatinib against Unresectable Hepatocellular Carcinoma.

Authors:  Atsushi Hiraoka; Takashi Kumada; Masanori Atsukawa; Masashi Hirooka; Kunihiko Tsuji; Toru Ishikawa; Koichi Takaguchi; Kazuya Kariyama; Ei Itobayashi; Kazuto Tajiri; Noritomo Shimada; Hiroshi Shibata; Hironori Ochi; Toshifumi Tada; Hidenori Toyoda; Kazuhiro Nouso; Akemi Tsutsui; Takuya Nagano; Norio Itokawa; Korenobu Hayama; Michitaka Imai; Kouji Joko; Hironori Tanaka; Tsutomu Tamai; Yohei Koizumi; Yoichi Hiasa; Kojiro Michitaka; Masatoshi Kudo
Journal:  Oncology       Date:  2019-07-15       Impact factor: 2.935

6.  Usefulness of albumin-bilirubin grade for evaluation of prognosis of 2584 Japanese patients with hepatocellular carcinoma.

Authors:  Atsushi Hiraoka; Takashi Kumada; Kojiro Michitaka; Hidenori Toyoda; Toshifumi Tada; Hidetaro Ueki; Miho Kaneto; Toshihiko Aibiki; Tomonari Okudaira; Takamasa Kawakami; Tomoe Kawamura; Hiroka Yamago; Yoshifumi Suga; Yuji Miyamoto; Hideomi Tomida; Nobuaki Azemoto; Kenichiro Mori; Hideki Miyata; Tomoyuki Ninomiya; Hideki Kawasaki
Journal:  J Gastroenterol Hepatol       Date:  2016-05       Impact factor: 4.029

7.  Regorafenib for patients with hepatocellular carcinoma who progressed on sorafenib treatment (RESORCE): a randomised, double-blind, placebo-controlled, phase 3 trial.

Authors:  Jordi Bruix; Shukui Qin; Philippe Merle; Alessandro Granito; Yi-Hsiang Huang; György Bodoky; Marc Pracht; Osamu Yokosuka; Olivier Rosmorduc; Valeriy Breder; René Gerolami; Gianluca Masi; Paul J Ross; Tianqiang Song; Jean-Pierre Bronowicki; Isabelle Ollivier-Hourmand; Masatoshi Kudo; Ann-Lii Cheng; Josep M Llovet; Richard S Finn; Marie-Aude LeBerre; Annette Baumhauer; Gerold Meinhardt; Guohong Han
Journal:  Lancet       Date:  2016-12-06       Impact factor: 79.321

8.  Sorafenib in advanced hepatocellular carcinoma.

Authors:  Josep M Llovet; Sergio Ricci; Vincenzo Mazzaferro; Philip Hilgard; Edward Gane; Jean-Frédéric Blanc; Andre Cosme de Oliveira; Armando Santoro; Jean-Luc Raoul; Alejandro Forner; Myron Schwartz; Camillo Porta; Stefan Zeuzem; Luigi Bolondi; Tim F Greten; Peter R Galle; Jean-François Seitz; Ivan Borbath; Dieter Häussinger; Tom Giannaris; Minghua Shan; Marius Moscovici; Dimitris Voliotis; Jordi Bruix
Journal:  N Engl J Med       Date:  2008-07-24       Impact factor: 91.245

9.  Validation and Potential of Albumin-Bilirubin Grade and Prognostication in a Nationwide Survey of 46,681 Hepatocellular Carcinoma Patients in Japan: The Need for a More Detailed Evaluation of Hepatic Function.

Authors:  Atsushi Hiraoka; Kojiro Michitaka; Takashi Kumada; Namiki Izumi; Masumi Kadoya; Norihiro Kokudo; Shoji Kubo; Yutaka Matsuyama; Osamu Nakashima; Michiie Sakamoto; Tadatoshi Takayama; Takashi Kokudo; Kosuke Kashiwabara; Masatoshi Kudo
Journal:  Liver Cancer       Date:  2017-09-22       Impact factor: 11.740

10.  Therapeutic efficacy of lenvatinib for patients with unresectable hepatocellular carcinoma based on the middle-term outcome.

Authors:  Akira Fuchigami; Yukinori Imai; Yoshihito Uchida; Hiroshi Uchiya; Yohei Fujii; Manabu Nakazawa; Satsuki Ando; Kayoko Sugawara; Nobuaki Nakayama; Tomoaki Tomiya; Satoshi Mochida
Journal:  PLoS One       Date:  2020-04-10       Impact factor: 3.240

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  5 in total

1.  Lenvatinib with or without Concurrent Drug-Eluting Beads Transarterial Chemoembolization in Patients with Unresectable, Advanced Hepatocellular Carcinoma: A Real-World, Multicenter, Retrospective Study.

Authors:  Dongdong Xia; Wei Bai; Enxin Wang; Jiaping Li; Xiaoming Chen; Zhexuan Wang; Mingsheng Huang; Ming Huang; Junhui Sun; Weizhu Yang; Zhengyu Lin; Jianbing Wu; Zixiang Li; Shufa Yang; Xu Zhu; Zaizhong Chen; Yanfang Zhang; Wenzhe Fan; Qicong Mai; Rong Ding; Chunhui Nie; Long Feng; Xueda Li; Wukui Huang; Jun Sun; Qiuhe Wang; Yong Lv; Xiaomei Li; Bohan Luo; Zhengyu Wang; Jie Yuan; Wengang Guo; Kai Li; Bing Li; Ruijun Li; Zhanxin Yin; Jielai Xia; Guohong Han
Journal:  Liver Cancer       Date:  2022-03-09       Impact factor: 12.430

2.  m7G Methylation-Related Genes as Biomarkers for Predicting Overall Survival Outcomes for Hepatocellular Carcinoma.

Authors:  Xin-Yu Li; Zhi-Jie Zhao; Jing-Bing Wang; Yu-Hao Shao; Jian-Xiong You; Xi-Tao Yang
Journal:  Front Bioeng Biotechnol       Date:  2022-05-10

Review 3.  New treatment paradigm with systemic therapy in intermediate-stage hepatocellular carcinoma.

Authors:  Masatoshi Kudo
Journal:  Int J Clin Oncol       Date:  2022-05-08       Impact factor: 3.850

4.  Analysis of Survival and Response to Lenvatinib in Unresectable Hepatocellular Carcinoma.

Authors:  Kei Amioka; Tomokazu Kawaoka; Masanari Kosaka; Yusuke Johira; Yuki Shirane; Ryoichi Miura; Serami Murakami; Shigeki Yano; Kensuke Naruto; Yuwa Ando; Yumi Kosaka; Yasutoshi Fujii; Kenichiro Kodama; Shinsuke Uchikawa; Hatsue Fujino; Atsushi Ono; Takashi Nakahara; Eisuke Murakami; Wataru Okamoto; Masami Yamauchi; Michio Imamura; Nami Mori; Shintaro Takaki; Keiji Tsuji; Keiichi Masaki; Yoji Honda; Hirotaka Kouno; Hiroshi Kohno; Takashi Moriya; Noriaki Naeshiro; Michihiro Nonaka; Hideyuki Hyogo; Yasuyuki Aisaka; Takahiro Azakami; Akira Hiramatsu; Hiroshi Aikata
Journal:  Cancers (Basel)       Date:  2022-01-10       Impact factor: 6.639

5.  Atezolizumab plus bevacizumab treatment for unresectable hepatocellular carcinoma: Early clinical experience.

Authors:  Atsushi Hiraoka; Takashi Kumada; Toshifumi Tada; Masashi Hirooka; Kazuya Kariyama; Joji Tani; Masanori Atsukawa; Koichi Takaguchi; Ei Itobayashi; Shinya Fukunishi; Kunihiko Tsuji; Toru Ishikawa; Kazuto Tajiri; Hironori Ochi; Satoshi Yasuda; Hidenori Toyoda; Chikara Ogawa; Takashi Nishimura; Takeshi Hatanaka; Hideko Ohama; Kazuhiro Nouso; Asahiro Morishita; Akemi Tsutsui; Takuya Nagano; Norio Itokawa; Tomomi Okubo; Taeang Arai; Michitaka Imai; Yohei Koizumi; Shinichiro Nakamura; Kouji Joko; Hiroko Iijima; Yoichi Hiasa; Masatoshi Kudo
Journal:  Cancer Rep (Hoboken)       Date:  2021-06-11
  5 in total

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