Literature DB >> 3385722

N6-[2-(3,5-dimethoxyphenyl)-2-(2-methylphenyl)ethyl]adenosine and its uronamide derivatives. Novel adenosine agonists with both high affinity and high selectivity for the adenosine A2 receptor.

A J Bridges1, R F Bruns, D F Ortwine, S R Priebe, D L Szotek, B K Trivedi.   

Abstract

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Year:  1988        PMID： 3385722     DOI： 10.1021/jm00402a004

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  17 in total

1.  Docking studies of agonists and antagonists suggest an activation pathway of the A3 adenosine receptor.

Authors:  Soo-Kyung Kim; Zhan-Guo Gao; Lak Shin Jeong; Kenneth A Jacobson
Journal:  J Mol Graph Model       Date:  2006-05-09       Impact factor: 2.518

Review 2.  Adenosine receptors as therapeutic targets.

Authors:  Kenneth A Jacobson; Zhan-Guo Gao
Journal:  Nat Rev Drug Discov       Date:  2006-03       Impact factor: 84.694

3.  Adenosine promotes burst activity in guinea-pig geniculocortical neurones through two different ionic mechanisms.

Authors:  H C Pape
Journal:  J Physiol       Date:  1992-02       Impact factor: 5.182

4.  ATP and glutamate are released from separate neurones in the rat medial habenula nucleus: frequency dependence and adenosine-mediated inhibition of release.

Authors:  S J Robertson; F A Edwards
Journal:  J Physiol       Date:  1998-05-01       Impact factor: 5.182

5.  Adenosine-mediated presynaptic modulation of glutamatergic transmission in the laterodorsal tegmentum.

Authors:  E Arrigoni; D G Rainnie; R W McCarley; R W Greene
Journal:  J Neurosci       Date:  2001-02-01       Impact factor: 6.167

6.  Molecular modeling of adenosine receptors. The ligand binding site on the rat adenosine A2A receptor.

Authors:  A P IJzerman; E M van der Wenden; P J van Galen; K A Jacobson
Journal:  Eur J Pharmacol       Date:  1994-06-15       Impact factor: 4.432

7.  Agonist derived molecular probes for A2 adenosine receptors.

Authors:  K A Jacobson; L K Pannell; X D Ji; M F Jarvis; M Williams; A J Hutchison; W W Barrington; G L Stiles
Journal:  J Mol Recognit       Date:  1989-12       Impact factor: 2.137

8.  A comparison of A2 adenosine receptor-induced cyclic AMP generation in cerebral cortex and relaxation of pre-contracted aorta.

Authors:  S P Alexander; A Losinski; D A Kendall; S J Hill
Journal:  Br J Pharmacol       Date:  1994-01       Impact factor: 8.739

9.  Adenosine-induced hyperpolarization of the membrane voltage in rat mesangial cells in primary culture.

Authors:  H Pavenstädt; J Ruh; R Greger; P Schollmeyer
Journal:  Br J Pharmacol       Date:  1994-09       Impact factor: 8.739

10.  Characterization of the locomotor depression produced by an A2-selective adenosine agonist.

Authors:  O Nikodijević; J W Daly; K A Jacobson
Journal:  FEBS Lett       Date:  1990-02-12       Impact factor: 4.124
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