Literature DB >> 33839076

Levosimendan Improves Hemodynamics and Exercise Tolerance in PH-HFpEF: Results of the Randomized Placebo-Controlled HELP Trial.

Daniel Burkhoff1, Barry A Borlaug2, Sanjiv J Shah3, Ronald Zolty4, Ryan J Tedford5, Thenappan Thenappan6, Roham T Zamanian7, Jeremy A Mazurek8, Jonathan D Rich3, Marc A Simon9, Eugene S Chung10, Farhan Raza11, David T Majure12, Gregory D Lewis13, Ioana R Preston14, Stuart Rich3.   

Abstract

OBJECTIVES: The purpose of this study was to evaluate the effects of intravenous levosimendan on hemodynamics and 6-min walk distance (6MWD) in patients with pulmonary hypertension and heart failure with preserved ejection fraction (PH-HFpEF).
BACKGROUND: There are no proven effective treatments for patients with PH-HFpEF.
METHODS: Patients with mean pulmonary artery pressure (mPAP) ≥35 mm Hg, pulmonary capillary wedge pressure (PCWP) ≥20 mm Hg, and LVEF ≥40% underwent 6MWD and hemodynamic measurements at rest, during passive leg raise, and supine cycle exercise at baseline and after an open-label 24-h levosimendan infusion (0.1 μg/kg/min). Hemodynamic responders (those with ≥4 mm Hg reduction of exercise-PCWP) were randomized (double blind) to weekly levosimendan infusion (0.075 to 0.1 ug/kg/min for 24 h) or placebo for 5 additional weeks. The primary end point was exercise-PCWP, and key secondary end points included 6MWD and PCWP measured across all exercise stages.
RESULTS: Thirty-seven of 44 patients (84%) met responder criteria and were randomized to levosimendan (n = 18) or placebo (n = 19). Participants were 69 ± 9 years of age, 61% female, and with resting mPAP 41.0 ± 9.3 mm Hg and exercise-PCWP 36.8 ± 11.3 mm Hg. Compared with placebo, levosimendan did not significantly reduce the primary end point of exercise-PCWP at 6 weeks (-1.4 mm Hg; 95% confidence interval [CI]: -7.8 to 4.8; p = 0.65). However, levosimendan reduced PCWP measured across all exercise stages (-3.9 ± 2.0 mm Hg; p = 0.047). Levosimendan treatment resulted in a 29.3 m (95% CI: 2.5 to 56.1; p = 0.033) improvement in 6MWD compared with placebo.
CONCLUSIONS: Six weeks of once-weekly levosimendan infusion did not affect exercise-PCWP but did reduce PCWP incorporating data from rest and exercise, in tandem with increased 6MWD. Further study of levosimendan is warranted as a therapeutic option for PH-HFpEF. (Hemodynamic Evaluation of Levosimendan in Patients With PH-HFpEF [HELP]; NCT03541603).
Copyright © 2021 The Authors. Published by Elsevier Inc. All rights reserved.

Entities:  

Keywords:  exercise; heart failure with preserved ejection fraction (HFpEF); hemodynamics; levosimendan; pulmonary hypertension

Mesh:

Substances:

Year:  2021        PMID: 33839076     DOI: 10.1016/j.jchf.2021.01.015

Source DB:  PubMed          Journal:  JACC Heart Fail        ISSN: 2213-1779            Impact factor:   12.035


  13 in total

Review 1.  Pulmonary Hypertension in the Context of Heart Failure With Preserved Ejection Fraction.

Authors:  Chakradhari Inampudi; Daniel Silverman; Marc A Simon; Peter J Leary; Kavita Sharma; Brian A Houston; Jean-Luc Vachiéry; Francois Haddad; Ryan J Tedford
Journal:  Chest       Date:  2021-08-12       Impact factor: 9.410

Review 2.  Heart Failure with Preserved Ejection Fraction: Mechanisms and Treatment Strategies.

Authors:  Kazunori Omote; Frederik H Verbrugge; Barry A Borlaug
Journal:  Annu Rev Med       Date:  2021-08-11       Impact factor: 13.739

Review 3.  Targeting Preload in Heart Failure: Splanchnic Nerve Blockade and Beyond.

Authors:  Marat Fudim; Muhammad Shahzeb Khan; Anousheh Awais Paracha; Kenji Sunagawa; Daniel Burkhoff
Journal:  Circ Heart Fail       Date:  2022-03-15       Impact factor: 8.790

4.  Advances in the understanding of excitation-contraction coupling: the pulsing quest for drugs against heart failure and arrhythmias.

Authors:  Urna Kansakar; Fahimeh Varzideh; Stanislovas S Jankauskas; Jessica Gambardella; Bruno Trimarco; Gaetano Santulli
Journal:  Eur Heart J Cardiovasc Pharmacother       Date:  2021-11-03

Review 5.  Understanding the Pathobiology of Pulmonary Hypertension Due to Left Heart Disease.

Authors:  Jessica H Huston; Sanjiv J Shah
Journal:  Circ Res       Date:  2022-04-28       Impact factor: 23.213

Review 6.  Venous Tone and Stressed Blood Volume in Heart Failure: JACC Review Topic of the Week.

Authors:  Marat Fudim; David M Kaye; Barry A Borlaug; Sanjiv J Shah; Stuart Rich; Navin K Kapur; Maria Rosa Costanzo; Michael I Brener; Kenji Sunagawa; Daniel Burkhoff
Journal:  J Am Coll Cardiol       Date:  2022-05-10       Impact factor: 27.203

7.  Pulmonary vasodilator treatment in pulmonary hypertension due to left heart or lung disease: time for a high-definition picture?

Authors:  Lucilla Piccari; Roberto J Bernardo; Diego Rodríguez-Chiaradía; Patrizio Vitulo; S John Wort; Sandeep Sahay
Journal:  Pulm Circ       Date:  2021-05-29       Impact factor: 3.017

8.  The Adenylate Cyclase Activator Forskolin Potentiates the Positive Inotropic Effect of the Phosphodiesterase Inhibitor Milrinone But Not of the Calcium Sensitizer Levosimendan nor of Its Hemodynamically Active Metabolites: An Apparent Conundrum.

Authors:  Jouko Levijoki; Piero Pollesello; Elena Grossini; Zoltán Papp
Journal:  J Cardiovasc Pharmacol       Date:  2022-06-01       Impact factor: 3.271

9.  Pulmonary vascular distensibility with passive leg raise is comparable to exercise and predictive of clinical outcomes in pulmonary hypertension.

Authors:  Callyn J Kozitza; Naga Dharmavaram; Ran Tao; Diana M Tabima; Naomi C Chesler; Farhan Raza
Journal:  Pulm Circ       Date:  2022-01-12       Impact factor: 2.886

Review 10.  Levosimendan-induced venodilation is mediated by opening of potassium channels.

Authors:  Daniel Burkhoff; Stuart Rich; Piero Pollesello; Zoltán Papp
Journal:  ESC Heart Fail       Date:  2021-10-30
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