Literature DB >> 33769176

What makes a good fragment in fragment-based drug discovery?

Zenon Konteatis1.   

Abstract

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Year:  2021        PMID： 33769176     DOI： 10.1080/17460441.2021.1905629

Source DB:  PubMed          Journal:  Expert Opin Drug Discov        ISSN： 1746-0441            Impact factor:   6.098


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  3 in total

1.  Comprehensive analysis of commercial fragment libraries.

Authors:  Julia Revillo Imbernon; Célien Jacquemard; Guillaume Bret; Gilles Marcou; Esther Kellenberger
Journal:  RSC Med Chem       Date:  2021-12-24

2.  Quadruple Target Evaluation of Diversity-Optimized Halogen-Enriched Fragments (HEFLibs) Reveals Substantial Ligand Efficiency for AP2-Associated Protein Kinase 1 (AAK1).

Authors:  Marcel Dammann; Markus Kramer; Markus O Zimmermann; Frank M Boeckler
Journal:  Front Chem       Date:  2022-02-02       Impact factor: 5.221

3.  Fragment Libraries Designed to Be Functionally Diverse Recover Protein Binding Information More Efficiently Than Standard Structurally Diverse Libraries.

Authors:  Anna Carbery; Rachael Skyner; Frank von Delft; Charlotte M Deane
Journal:  J Med Chem       Date:  2022-08-12       Impact factor: 8.039
  3 in total

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