Literature DB >> 33582070

Subtypes of EGFR- and HER2-Mutant Metastatic NSCLC Influence Response to Immune Checkpoint Inhibitors.

Sally C M Lau1, Aline Fusco Fares1, Lisa W Le2, Kate M Mackay1, Spencer Soberano1, Sze Wah Chan1, Elliot Smith1, Malcolm Ryan1, Ming Sound Tsao3, Penelope A Bradbury1, Prodipto Pal3, Frances A Shepherd1, Geoffrey Liu1, Natasha B Leighl1, Adrian G Sacher4.   

Abstract

INTRODUCTION: The efficacy of immune checkpoint inhibitors (ICIs) is low among EGFR-mutated non-small-cell lung cancer (NSCLC), although prolonged responses have occasionally been reported. We investigated the association between mutation subtypes and ICI outcomes among HER2- and EGFR-mutated NSCLC. PATIENTS AND METHODS: This retrospective single-center study analyzed patients with EGFR- and HER2-mutated advanced NSCLC who received at least 1 cycle of ICI between 2013 and 2019. Patient characteristics, mutation subtype, and ICI outcomes.
RESULTS: Among 48 patients with advanced NSCLC, 14 (29%) had HER2 mutations and 34 (71%) had EGFR mutations. EGFR mutations included 16 (47%) exon 19 deletion, 7 (21%) L858R, 5 (15%) uncommon, and 6 (18%) exon 20 insertion. Compared to EGFR-sensitizing mutations (ESMs), HER2 and EGFR exon 20 mutations were associated with a trend toward better response (respectively, ESM, HER2, and EGFR exon 20: 11%, 29%, and 50%; P = .07) and significantly better disease control rates (respectively, 18%, 57%, and 67%; P = .008). Compared to ESM, HER2 mutations (adjusted hazard ratio, 0.35; P = .02) and EGFR exon 20 mutations (adjusted hazard ratio, 0.37; P = .10 trend) were also associated with improved PFS. Programmed death ligand 1 (PD-L1) expression remained an independent predictor of PFS (adjusted hazard ratio, 0.42; 95% confidence interval, 0.23-0.76; P = .004). The 6-month PFS rates were 29% (HER2), 33% (EGFR exon 20), and 4% (ESM). ICIs were generally well tolerated in this population. Importantly, no immune-related toxicity was observed in 10 patients who received a tyrosine kinase inhibitor (TKI) as the immediate next line treatment after ICI.
CONCLUSION: HER2 and EGFR exon 20 mutations derive greater benefit from ICIs with comparable PFS to wild-type historical second/third-line unselected cohorts. ICIs remain a treatment option for this genomic subgroup, given the absence of approved targeted therapies for these rare mutations.
Copyright © 2021 Elsevier Inc. All rights reserved.

Entities:  

Keywords:  Driver mutations; Immunotherapy; Oncogene addiction; PD-1 inhibitors; PD-L1

Mesh:

Substances:

Year:  2021        PMID: 33582070     DOI: 10.1016/j.cllc.2020.12.015

Source DB:  PubMed          Journal:  Clin Lung Cancer        ISSN: 1525-7304            Impact factor:   4.785


  18 in total

1.  Real-world progression-free survival (rwPFS) and the impact of PD-L1 and smoking in driver-mutated non-small cell lung cancer (NSCLC) treated with immunotherapy.

Authors:  J Nicholas Bodor; Jessica R Bauman; Elizabeth A Handorf; Eric A Ross; Margie L Clapper; Joseph Treat
Journal:  J Cancer Res Clin Oncol       Date:  2022-06-16       Impact factor: 4.322

Review 2.  Non-small Cell Lung Cancer with EGFR or HER2 Exon 20 Insertion Mutations: Diagnosis and Treatment Options.

Authors:  Danielle Brazel; Gianna Kroening; Misako Nagasaka
Journal:  BioDrugs       Date:  2022-10-18       Impact factor: 7.744

3.  Sensitivity to Immune Checkpoint Blockade in Advanced Non-Small Cell Lung Cancer Patients with EGFR Exon 20 Insertion Mutations.

Authors:  Giulio Metro; Sara Baglivo; Guido Bellezza; Martina Mandarano; Alessio Gili; Giovanni Marchetti; Marco Toraldo; Carmen Molica; Maria Sole Reda; Francesca Romana Tofanetti; Annamaria Siggillino; Enrico Prosperi; Antonella Giglietti; Bruna Di Girolamo; Miriam Garaffa; Francesca Marasciulo; Vincenzo Minotti; Marco Gunnellini; Annalisa Guida; Monica Sassi; Angelo Sidoni; Fausto Roila; Vienna Ludovini
Journal:  Genes (Basel)       Date:  2021-04-30       Impact factor: 4.096

4.  Therapeutic exploration of uncommon EGFR exon 20 insertion mutations in advanced non-small cell lung cancer: breaking through brambles and thorns.

Authors:  Rilan Bai; Xiao Chen; Wei Song; Huimin Tian; Jiuwei Cui
Journal:  J Cancer Res Clin Oncol       Date:  2021-10-26       Impact factor: 4.553

Review 5.  EGFR and HER2 exon 20 insertions in solid tumours: from biology to treatment.

Authors:  Alex Friedlaender; Vivek Subbiah; Alessandro Russo; Giuseppe Luigi Banna; Umberto Malapelle; Christian Rolfo; Alfredo Addeo
Journal:  Nat Rev Clin Oncol       Date:  2021-09-24       Impact factor: 66.675

Review 6.  Comparative Analysis of Predictive Biomarkers for PD-1/PD-L1 Inhibitors in Cancers: Developments and Challenges.

Authors:  Fang Yang; Jacqueline F Wang; Yucai Wang; Baorui Liu; Julian R Molina
Journal:  Cancers (Basel)       Date:  2021-12-27       Impact factor: 6.639

7.  Case Report: Tumor Microenvironment Characteristics in a Patient With HER2 Mutant Lung Squamous Cell Carcinoma Harboring High PD-L1 Expression Who Presented Hyperprogressive Disease.

Authors:  Lixia Xia; Yinghui Yu; Fen Lan; Junrong Yan; Jinfan Li; Wen Li; Yang Xia
Journal:  Front Oncol       Date:  2021-12-24       Impact factor: 6.244

Review 8.  Anti-PD1/PD-L1 Immunotherapy for Non-Small Cell Lung Cancer with Actionable Oncogenic Driver Mutations.

Authors:  Edouard Dantoing; Nicolas Piton; Mathieu Salaün; Luc Thiberville; Florian Guisier
Journal:  Int J Mol Sci       Date:  2021-06-11       Impact factor: 5.923

Review 9.  HER2 Aberrations in Non-Small Cell Lung Cancer: From Pathophysiology to Targeted Therapy.

Authors:  Ioannis A Vathiotis; Andriani Charpidou; Niki Gavrielatou; Konstantinos N Syrigos
Journal:  Pharmaceuticals (Basel)       Date:  2021-12-14

Review 10.  Discovery, Development, Inventions, and Patent Trends on Mobocertinib Succinate: The First-in-Class Oral Treatment for NSCLC with EGFR Exon 20 Insertions.

Authors:  Mohd Imran; Shah Alam Khan; Mohammed Kanan Alshammari; Meshal Ayedh Alreshidi; Abeer Abdullah Alreshidi; Rawan Sulaiman Alghonaim; Fayez Aboud Alanazi; Sultan Alshehri; Mohammed M Ghoneim; Faiyaz Shakeel
Journal:  Biomedicines       Date:  2021-12-17
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