Literature DB >> 33435617

Inhibition of MLKL Attenuates Necroptotic Cell Death in a Murine Cell Model of Ischaemia Injury.

Raji Baidya1,2, Jérémie Gautheron3,4, Darrell H G Crawford1,2, Haolu Wang2,5, Kim R Bridle1,2.   

Abstract

BACKGROUND: Steatosis in donor livers poses a major risk of organ dysfunction due to their susceptibility to ischaemia-reperfusion (I/R) injury during transplant. Necroptosis, a novel form of programmed cell death, is orchestrated by receptor-interacting protein kinase 1 (RIPK1), receptor-interacting protein kinase 3 (RIPK3) and mixed-lineage kinase domain-like pseudokinase (MLKL), has been implicated in I/R injury. Here we investigated the mechanisms of cell death pathways in an in vitro model of hepato-steatotic ischaemia.
METHODS: Free fatty acid (FFA) treated alpha mouse liver 12 (AML-12) cells were incubated in oxygen-glucose-deprivation (OGD) conditions as seen during ischaemia.
RESULTS: We found that OGD triggered upregulation of insoluble fraction of RIPK3 and MLKL in FFA + OGD cells compared to FFA control cells. We report that intervention with small interfering (si) MLKL and siRIPK3 significantly attenuated cell death in FFA + OGD cells. Absence of activated CASPASE8 and cleaved-CASPASE3, no change in the expression of CASPASE1 and prostaglandin-endoperoxide synthase 2 (Ptgs2) in FFA + OGD treated cells compared to FFA control cells indicated that apoptosis, pyroptosis and ferroptosis, respectively, are unlikely to be active in this model.
CONCLUSION: Our findings indicate that RIPK3-MLKL dependent necroptosis contributed to cell death in our in vitro model. Both MLKL and RIPK3 are promising therapeutic targets to inhibit necroptosis during ischaemic injury in fatty liver.

Entities:  

Keywords:  apoptosis; in vitro; ischaemia-reperfusion injury; liver transplantation; necroptosis; steatosis

Year:  2021        PMID: 33435617     DOI: 10.3390/jcm10020212

Source DB:  PubMed          Journal:  J Clin Med        ISSN: 2077-0383            Impact factor:   4.241


  4 in total

1.  Liver Ischemia and Reperfusion Induce Periportal Expression of Necroptosis Executor pMLKL Which Is Associated With Early Allograft Dysfunction After Transplantation.

Authors:  Shaojun Shi; Eliano Bonaccorsi-Riani; Ivo Schurink; Thierry van den Bosch; Michael Doukas; Karishma A Lila; Henk P Roest; Daela Xhema; Pierre Gianello; Jeroen de Jonge; Monique M A Verstegen; Luc J W van der Laan
Journal:  Front Immunol       Date:  2022-05-17       Impact factor: 8.786

2.  Custodiol® Supplemented with Synthetic Human Relaxin Decreases Ischemia-Reperfusion Injury after Porcine Kidney Transplantation.

Authors:  Augustinas Bausys; Juste Maneikyte; Bettina Leber; Jennifer Weber; Nicole Feldbacher; Kestutis Strupas; Thomas Bernd Dschietzig; Peter Schemmer; Philipp Stiegler
Journal:  Int J Mol Sci       Date:  2021-10-22       Impact factor: 5.923

3.  The necroptosis-inducing pseudokinase mixed lineage kinase domain-like regulates the adipogenic differentiation of pre-adipocytes.

Authors:  Julie Magusto; Carine Beaupère; Marta B Afonso; Martine Auclair; Jean-Louis Delaunay; Pierre-Antoine Soret; Gilles Courtois; Tounsia Aït-Slimane; Chantal Housset; Isabelle Jéru; Bruno Fève; Vlad Ratziu; Cecilia M P Rodrigues; Jérémie Gautheron
Journal:  iScience       Date:  2022-09-19

4.  PPARγ2 functions as a tumor suppressor in a translational mouse model of human prostate cancer.

Authors:  Fu-Lu Dong; Dong-Mei Liu; Ting-Ting Lu; Feng Li; Chong Zhang; Qun E; Yong-Hui Zhang
Journal:  Asian J Androl       Date:  2022 Jan-Feb       Impact factor: 3.285

  4 in total

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