Literature DB >> 33432459

Reduced postprandial bone resorption and greater rise in GLP-1 in overweight and obese individuals after an α-glucosidase inhibitor: a double-blinded randomized crossover trial.

A Kreitman1, S H Schneider2,3, L Hao1,3, Y Schlussel1, N T Bello3,4, S A Shapses5,6,7.   

Abstract

When taken with a meal, α-glucosidase inhibitors (α-GI) reduce the rise in postprandial glucose and increase glucagon-like peptide-1 (GLP-1), and this may lower bone turnover. In this study, a salacinol-type α-GI increased GLP-1 and markedly reduced postprandial bone resorption compared to placebo, suggesting it could have implications for bone health.
INTRODUCTION: Animal and clinical trials indicate that α-glucosidase inhibitors attenuate postprandial glycemic indices and increase secretion of GLP-1. In addition, GLP-1 acts on bone by inhibiting resorption. The goal in this study was to determine if a salacinol α-GI alters postprandial bone turnover and can be explained by changes in serum GLP-1.
METHODS: In this double-blind, placebo-controlled crossover study, healthy overweight/obese adults (body mass index 29.0 ± 3.8 kg/m2; 21-59 years; n = 21) received a fixed breakfast and, in random order, were administered Salacia chinensis (SC; 500 mg) or placebo. A fasting blood sample was taken before and at regular intervals for 3 h after the meal. Serum was measured for bone turnover markers, C-terminal telopeptide of type I collagen (CTX) and osteocalcin, and for glycemic indices and gut peptides.
RESULTS: Compared to placebo, SC attenuated the bone resorption marker, CTX, at 60, 90, and 120 min (p < 0.05) after the meal, and decreased osteocalcin, at 180 min (p < 0.05). As expected, SC attenuated the postprandial rise in glucose compared with placebo, whereas GLP-1 was increased at 60 min (p < 0.05) with SC. Serum GLP-1 explained 41% of the variance for change in postprandial CTX (p < 0.05).
CONCLUSION: This study indicates that attenuating postprandial glycemic indices, with an α-GI, markedly decreases postprandial bone resorption and can be explained by the rise in GLP-1. Future studies should determine whether longer term α-GI use benefits bone health.

Entities:  

Keywords:  Alpha-glucosidase inhibitor; Bone turnover; GLP-1; Mixed meal tolerance test; Salacia

Year:  2021        PMID: 33432459     DOI: 10.1007/s00198-020-05791-5

Source DB:  PubMed          Journal:  Osteoporos Int        ISSN: 0937-941X            Impact factor:   4.507


  4 in total

1.  Comparison of the hypoglycemic effect of acarbose monotherapy in patients with type 2 diabetes mellitus consuming an Eastern or Western diet: a systematic meta-analysis.

Authors:  Qibo Zhu; Yuzhen Tong; Taixiang Wu; Jieqing Li; Nanwei Tong
Journal:  Clin Ther       Date:  2013-04-18       Impact factor: 3.393

2.  Hydrophobic substituents increase the potency of salacinol, a potent α-glucosidase inhibitor from Ayurvedic traditional medicine 'Salacia'.

Authors:  Genzoh Tanabe; Weijia Xie; Gorre Balakishan; Mumen F A Amer; Nozomi Tsutsui; Haruka Takemura; Shinya Nakamura; Junji Akaki; Kiyofumi Ninomiya; Toshio Morikawa; Isao Nakanishi; Osamu Muraoka
Journal:  Bioorg Med Chem       Date:  2016-06-07       Impact factor: 3.641

3.  Salacia Extract Improves Postprandial Glucose and Insulin Response: A Randomized Double-Blind, Placebo Controlled, Crossover Study in Healthy Volunteers.

Authors:  Shankaranarayanan Jeykodi; Jayant Deshpande; Vijaya Juturu
Journal:  J Diabetes Res       Date:  2016-10-10       Impact factor: 4.011

4.  Postprandial metabolic responses of serum calcium, parathyroid hormone and C-telopeptide of type I collagen to three doses of calcium delivered in milk.

Authors:  Marlena C Kruger; Pamela R von Hurst; Christine L Booth; Barbara Kuhn-Sherlock; Joanne M Todd; Linda M Schollum
Journal:  J Nutr Sci       Date:  2014-04-30
  4 in total

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