Literature DB >> 33296668

Response to Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors.

Andrea Angeli1, Fabrizio Carta1, Alessio Nocentini1, Jean-Yves Winum2, Raivis Zalubovskis3, Valentina Onnis4, Wagdy M Eldehna5, Clemente Capasso6, Simone Carradori7, William A Donald8, Shoukat Dedhar9, Claudiu T Supuran10.   

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Year:  2020        PMID： 33296668      PMCID： PMC7820713          DOI： 10.1016/j.bpj.2020.11.011

Source DB:  PubMed          Journal:  Biophys J        ISSN： 0006-3495            Impact factor:   4.033


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  32 in total

Review 1.  Carbonic anhydrases: novel therapeutic applications for inhibitors and activators.

Authors:  Claudiu T Supuran
Journal:  Nat Rev Drug Discov       Date:  2008-02       Impact factor: 84.694

2.  Ureido-substituted benzenesulfonamides potently inhibit carbonic anhydrase IX and show antimetastatic activity in a model of breast cancer metastasis.

Authors:  Fabio Pacchiano; Fabrizio Carta; Paul C McDonald; Yuanmei Lou; Daniela Vullo; Andrea Scozzafava; Shoukat Dedhar; Claudiu T Supuran
Journal:  J Med Chem       Date:  2011-03-01       Impact factor: 7.446

3.  Lead Development of Thiazolylsulfonamides with Carbonic Anhydrase Inhibitory Action.

Authors:  Fabrizio Carta; Alexander Birkmann; Tamara Pfaff; Helmut Buschmann; Wilfried Schwab; Holger Zimmermann; Alfonso Maresca; Claudiu T Supuran
Journal:  J Med Chem       Date:  2017-03-17       Impact factor: 7.446

4.  Targeting tumor hypoxia: suppression of breast tumor growth and metastasis by novel carbonic anhydrase IX inhibitors.

Authors:  Yuanmei Lou; Paul C McDonald; Arusha Oloumi; Stephen Chia; Christina Ostlund; Ardalan Ahmadi; Alastair Kyle; Ulrich Auf dem Keller; Samuel Leung; David Huntsman; Blaise Clarke; Brent W Sutherland; Dawn Waterhouse; Marcel Bally; Calvin Roskelley; Christopher M Overall; Andrew Minchinton; Fabio Pacchiano; Fabrizio Carta; Andrea Scozzafava; Nadia Touisni; Jean-Yves Winum; Claudiu T Supuran; Shoukat Dedhar
Journal:  Cancer Res       Date:  2011-03-17       Impact factor: 12.701

5.  Carbonic anhydrase inhibitors based on sorafenib scaffold: Design, synthesis, crystallographic investigation and effects on primary breast cancer cells.

Authors:  Murat Bozdag; Marta Ferraroni; Carol Ward; Fabrizio Carta; Silvia Bua; Andrea Angeli; Simon P Langdon; Ian H Kunkler; Abdul-Malek S Al-Tamimi; Claudiu T Supuran
Journal:  Eur J Med Chem       Date:  2019-08-07       Impact factor: 6.514

6.  Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides derived from 4-isothiocyanato-benzolamide.

Authors:  Alessandro Cecchi; Jean-Yves Winum; Alessio Innocenti; Daniela Vullo; Jean-Louis Montero; Andrea Scozzafava; Claudiu T Supuran
Journal:  Bioorg Med Chem Lett       Date:  2004-12-06       Impact factor: 2.823

7.  Carbonic anhydrase inhibitors. Interaction of indapamide and related diuretics with 12 mammalian isozymes and X-ray crystallographic studies for the indapamide-isozyme II adduct.

Authors:  Claudia Temperini; Alessandro Cecchi; Andrea Scozzafava; Claudiu T Supuran
Journal:  Bioorg Med Chem Lett       Date:  2008-03-20       Impact factor: 2.823

8.  1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors.

Authors:  Melissa D'Ascenzio; Daniela Secci; Simone Carradori; Susi Zara; Paolo Guglielmi; Roberto Cirilli; Marco Pierini; Giulio Poli; Tiziano Tuccinardi; Andrea Angeli; Claudiu T Supuran
Journal:  J Med Chem       Date:  2020-02-04       Impact factor: 7.446

9.  The effect of temperature on the binding of sulfonamides to carbonic anhydrase isoenzymes I, II, and IV.

Authors:  C W Conroy; T H Maren
Journal:  Mol Pharmacol       Date:  1995-09       Impact factor: 4.436

10.  Nanoscale Ion Emitters in Native Mass Spectrometry for Measuring Ligand-Protein Binding Affinities.

Authors:  Giang T H Nguyen; Thinh N Tran; Matthew N Podgorski; Stephen G Bell; Claudiu T Supuran; William A Donald
Journal:  ACS Cent Sci       Date:  2019-01-14       Impact factor: 14.553
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  7 in total

1.  4-(3-Alkyl/benzyl-guanidino)benzenesulfonamides as selective carbonic anhydrase VII inhibitors.

Authors:  Morteza Abdoli; Simone Giovannuzzi; Claudiu T Supuran; Raivis Žalubovskis
Journal:  J Enzyme Inhib Med Chem       Date:  2022-12       Impact factor: 5.756

2.  Comments to the Editor Due to the Response by the Supuran Group to Our Article.

Authors:  Bengt-Harald Jonsson; Anders Liljas
Journal:  Biophys J       Date:  2020-12-13       Impact factor: 4.033

3.  Effect of amino acids and amines on the activity of the recombinant ι-carbonic anhydrase from the Gram-negative bacterium Burkholderia territorii.

Authors:  Viviana De Luca; Andrea Petreni; Vincenzo Carginale; Andrea Scaloni; Claudiu T Supuran; Clemente Capasso
Journal:  J Enzyme Inhib Med Chem       Date:  2021-12       Impact factor: 5.051

4.  Nitrous anhydrase activity of carbonic anhydrase II: cysteine is required for nitric oxide (NO) dependent phosphorylation of VASP in human platelets.

Authors:  Dimitrios Tsikas; Stepan Gambaryan
Journal:  J Enzyme Inhib Med Chem       Date:  2021-12       Impact factor: 5.051

Review 5.  Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase.

Authors:  Alessio Nocentini; Andrea Angeli; Fabrizio Carta; Jean-Yves Winum; Raivis Zalubovskis; Simone Carradori; Clemente Capasso; William A Donald; Claudiu T Supuran
Journal:  J Enzyme Inhib Med Chem       Date:  2021-12       Impact factor: 5.051

6.  Inhibitory Effects of Sulfonamide Derivatives on the β-Carbonic Anhydrase (MpaCA) from Malassezia pachydermatis, a Commensal, Pathogenic Fungus Present in Domestic Animals.

Authors:  Viviana De Luca; Andrea Angeli; Valeria Mazzone; Claudia Adelfio; Fabrizio Carta; Silvia Selleri; Vincenzo Carginale; Andrea Scaloni; Claudiu T Supuran; Clemente Capasso
Journal:  Int J Mol Sci       Date:  2021-11-22       Impact factor: 5.923

Review 7.  Amine- and Amino Acid-Based Compounds as Carbonic Anhydrase Activators.

Authors:  Andrea Angeli; Emanuela Berrino; Simone Carradori; Claudiu T Supuran; Marzia Cirri; Fabrizio Carta; Gabriele Costantino
Journal:  Molecules       Date:  2021-12-02       Impact factor: 4.411
  7 in total

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