Literature DB >> 33142249

Dose dependent reduction in median effective concentration (EC50) of ropivacaine with adjuvant dexmedetomidine in labor epidural analgesia: An up-down sequential allocation study.

Lin Liu1, Dan Drzymalski2, Wenping Xu1, Wangping Zhang1, Lizhong Wang1, Fei Xiao3.   

Abstract

STUDY
OBJECTIVE: Adjuvant dexmedetomidine can be used to reduce the required concentration of ropivacaine for labor epidural analgesia. However, the potency of dexmedetomidine has not been fully studied. The purpose of this study was to determine the median effective concentration (EC50) of ropivacaine with adjuvant dexmedetomidine.
DESIGN: Prospective, double-blind, up-down sequential allocation study.
SETTING: Academic medical center specializing in the care of women and children. PATIENTS: One hundred and fifty healthy, term parturients requesting labor epidural analgesia were randomly assigned to 1 of 5 different concentrations of dexmedetomidine: 0 μg/ml, 0.3 μg/ml, 0.4 μg/ml, 0.5 μg/ml, or 0.6 μg/ml.
INTERVENTIONS: The study solution for the first patient in each group included the randomly assigned concentration of dexmedetomidine in 0.1% ropivacaine. Subsequent patients in each randomization group received the assigned concentration of dexmedetomidine in a new concentration of ropivacaine as determined by the up-down allocation methodology. Effective analgesia was defined as pain on the visual analogue scale of<3 at30 min after administration of local anesthetic. The up-down sequential allocation method and probit regression were used to calculate the EC50 of epidural ropivacaine. MEASUREMENTS: The primary outcome was pain 30 min after administration of local anesthetic via epidural catheter. Exploratory outcomes included side effects, neonatal outcomes, and obstetric outcomes. MAIN
RESULTS: The EC50 values for ropivacaine in dexmedetomidine 0.4 μg/ml, 0.5 μg/ml, and 0.6 μg/ml (0.044% [95% CI 0.036% to 0.045%], 0.035% [95% CI 0.031% to 0.041%], and 0.039% [95% CI 0.034% to 0.045%], respectively) were lower compared to ropivacaine in dexmedetomidine 0 μg/ml and 0.3 μg/ml (0.086% [95% CI 0.081% to 0.092%], and, 0.069% [95% CI 0.056% to 0.076%], respectively). Differences between EC50 values for ropivacaine in dexmedetomidine 0.4 μg/ml, 0.5 μg/ml, and 0.6 μg/ml were not statistically significant. Results of our exploratory analyses did not reveal differences in side effects, neonatal outcomes, or obstetric outcomes.
CONCLUSIONS: In this study, the lowest concentration of dexmedetomidine in ropivacaine with the greatest clinical effect was 0.4 μg/ml, which is important because there may be no additional analgesic benefit of dexmedetomidine greater than 0.4 μg/ml.
Copyright © 2020 Elsevier Inc. All rights reserved.

Entities:  

Keywords:  50% effective concentration; Dexmedetomidine; Dose-response; Epidural; Labor analgesia

Year:  2020        PMID: 33142249     DOI: 10.1016/j.jclinane.2020.110115

Source DB:  PubMed          Journal:  J Clin Anesth        ISSN: 0952-8180            Impact factor:   9.452


  5 in total

Review 1.  Effect of Epidural Dexmedetomidine as an Adjuvant to Local Anesthetics for Labor Analgesia: A Meta-Analysis of Randomized Controlled Trials.

Authors:  Nijuan Li; Li Hu; Chunping Li; Xuelin Pan; Yong Tang
Journal:  Evid Based Complement Alternat Med       Date:  2021-10-27       Impact factor: 2.629

2.  Effect of Dexmedetomidine Combined with Ropivacaine on Cognitive Dysfunction and Inflammatory Response in Patients Undergoing Craniocerebral Surgery.

Authors:  Yang Liu; Hongwei Zhang; Wenhua Zhang
Journal:  Biomed Res Int       Date:  2021-11-30       Impact factor: 3.411

3.  Determination of the Dose-Response Relationship of Epidural Dexmedetomidine Combined with Ropivacaine for Labor Analgesia.

Authors:  Zhong Mei; Jing Yu; Jian-Xin Ni; Jia-Li Feng; Sheng-Jie Yao; Li-Feng Ni; Shao-Bo Song; Cong-Zhong Song; Xiao-Wei Qian
Journal:  Drug Des Devel Ther       Date:  2022-03-06       Impact factor: 4.162

4.  Dexmedetomidine Can Enhance PINK1/Parkin-Mediated Mitophagy in MPTP-Induced PD Mice Model by Activating AMPK.

Authors:  Cheng Chen; Yaohua Chen; Tingting Liu; Dan Song; Di Ma; Oumei Cheng
Journal:  Oxid Med Cell Longev       Date:  2022-04-12       Impact factor: 7.310

5.  Adjuvant Sufentanil Decreased the EC50 of Epidural Ropivacaine for Labor Analgesia in Healthy Term Pregnancy.

Authors:  Bo Xiang; Jian Yang; Xiaofeng Lei; Jin Yu
Journal:  Drug Des Devel Ther       Date:  2021-05-18       Impact factor: 4.162

  5 in total

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