Literature DB >> 32984536

SEVERE HYPERTRIGLYCERIDEMIA ASSOCIATED WITH EVEROLIMUS TREATMENT AFTER HEART TRANSPLANTATION.

Phillip Lo1,2, Katherine Kearney1,2, Christopher A Muir2,3, Ning Song1,2, John A Eisman2,3,4,5, Peter S Macdonald1,2,6.   

Abstract

OBJECTIVE: Everolimus, a mammalian target-ofrapamycin (mTOR) inhibitor, is increasingly used post-transplantation due to favorable effects on renal function and malignancy risk when compared to other immunosuppressive treatments such as calcineurin inhibitors. However, it can confer adverse effects such as dyslipidemia, which is not underpinned by any long-term screening and management of dyslipidemia in heart transplant recipients treated with everolimus.
METHODS: We report a case of severe hypertriglyceridemia which developed after commencement of everolimus in a heart transplant recipient with a background of Dunnigan-type familial partial lipodystrophy.
RESULTS: The patient is a 36-year-old woman who underwent heart transplantation for dilated cardiomyopathy. About 11 weeks following commencement of everolimus as part of her antirejection medication regime, serum triglyceride level concentration peaked at 5,093 mg/dL (normal, 0.0 to 177.2 mg/dL). There were no clinical complications with triglycerides at this elevated level and it improved substantially following cessation of everolimus and initiation of a high dose intravenous insulin-dextrose infusion.
CONCLUSION: This case highlights dyslipidemia as a potential complication of everolimus treatment and that appropriate screening is important as lipid lowering medication can effectively control levels and minimize adverse outcomes.
Copyright © 2020 AACE.

Entities:  

Year:  2020        PMID: 32984536      PMCID: PMC7511100          DOI: 10.4158/ACCR-2020-0191

Source DB:  PubMed          Journal:  AACE Clin Case Rep        ISSN: 2376-0605


  16 in total

Review 1.  Strategies for the management of adverse events associated with mTOR inhibitors.

Authors:  Bruce Kaplan; Yasir Qazi; Jason R Wellen
Journal:  Transplant Rev (Orlando)       Date:  2014-03-12       Impact factor: 3.943

Review 2.  Clinical practice. Hypertriglyceridemia.

Authors:  John D Brunzell
Journal:  N Engl J Med       Date:  2007-09-06       Impact factor: 91.245

3.  Hypertriglyceridemia-induced acute pancreatitis treated with insulin and heparin.

Authors:  Jennifer D Twilla; Jimmie Mancell
Journal:  Am J Health Syst Pharm       Date:  2012-02-01       Impact factor: 2.637

Review 4.  Management of adverse events associated with the use of everolimus in patients with advanced renal cell carcinoma.

Authors:  Camillo Porta; Susanne Osanto; Alain Ravaud; Miguel-Angel Climent; Ulka Vaishampayan; Dorothy A White; Patricia Creel; Brenda Dickow; Patricia Fischer; Suzanne Sweeney Gornell; Federica Meloni; Robert J Motzer
Journal:  Eur J Cancer       Date:  2011-04-08       Impact factor: 9.162

5.  Factors associated with low compliance with lipid-lowering drugs in hyperlipidemic patients.

Authors:  D N Kiortsis; P Giral; E Bruckert; G Turpin
Journal:  J Clin Pharm Ther       Date:  2000-12       Impact factor: 2.512

6.  Chronic rapamycin treatment causes glucose intolerance and hyperlipidemia by upregulating hepatic gluconeogenesis and impairing lipid deposition in adipose tissue.

Authors:  Vanessa P Houde; Sophie Brûlé; William T Festuccia; Pierre-Gilles Blanchard; Kerstin Bellmann; Yves Deshaies; André Marette
Journal:  Diabetes       Date:  2010-03-18       Impact factor: 9.461

Review 7.  Hypertriglyceridemia: its etiology, effects and treatment.

Authors:  George Yuan; Khalid Z Al-Shali; Robert A Hegele
Journal:  CMAJ       Date:  2007-04-10       Impact factor: 8.262

8.  Everolimus causing severe hypertriglyceridemia and acute pancreatitis.

Authors:  Somasundaram Subramaniam; Jason A Zell; Pamela L Kunz
Journal:  J Natl Compr Canc Netw       Date:  2013-01-01       Impact factor: 11.908

Review 9.  Everolimus in heart transplantation: an update.

Authors:  Stephan W Hirt; Christoph Bara; Markus J Barten; Tobias Deuse; Andreas O Doesch; Ingo Kaczmarek; Uwe Schulz; Jörg Stypmann; Assad Haneya; Hans B Lehmkuhl
Journal:  J Transplant       Date:  2013-12-05

Review 10.  Nonadherence to statins: individualized intervention strategies outside the pill box.

Authors:  Peter Lansberg; Andre Lee; Zhen-Vin Lee; Kannan Subramaniam; Sajita Setia
Journal:  Vasc Health Risk Manag       Date:  2018-05-24
View more
  1 in total

1.  Evaluation of Pharmacogenetics of Drug-Metabolizing Enzymes and Drug Efflux Transporter in Renal Transplants Receiving Immunosuppressants.

Authors:  Kannan Sridharan; Shamik Shah; Anfal Jassim; Mona Hammad; Johaina Ebrahim Al Gadhban; Ola Al Segai
Journal:  J Pers Med       Date:  2022-05-19
  1 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.