Literature DB >> 32978826

Molecular determinants of enhanced response to somatostatin receptor ligands after debulking in large GH-producing adenomas.

Joan Gil1, Montserrat Marques-Pamies2, Mireia Jordà1, Carmen Fajardo-Montañana3, Araceli García-Martínez4,5, Miguel Sampedro5,6, Guillermo Serra7, Isabel Salinas2, Alberto Blanco8, Elena Valassi9, Gemma Sesmilo10, Cristina Carrato11, Rosa Cámara12, Cristina Lamas13, Paula Casano-Sancho5,14, Clara V Alvarez15, Ignacio Bernabéu16, Susan M Webb9, Antonio Picó5,17, Mónica Marazuela5,6, Manel Puig-Domingo1,2,5,17.   

Abstract

OBJECTIVE: Large somatotrophic adenomas depict poor response to somatostatin receptor ligands (SRLs). Debulking has shown to enhance SRLs effect in some but not all cases and tumour volume reduction has been proposed as the main predictor of response. No biological studies have been performed so far in this matter. We aimed to identify molecular markers of response to SRLs after surgical debulking in GH-secreting adenomas.
DESIGN: We performed a multicenter retrospective study. PATIENTS: 24 patients bearing large GH-producing tumours. MEASUREMENTS: Clinical data and SRLs response both before and after surgical debulking were collected, and 21 molecular biomarkers of SRLs response were studied in tumour samples by gene expression.
RESULTS: From the 21 molecular markers studied, only two of them predicted enhanced SRLs response after surgery. Tumours with improved response to SRLs after surgical debulking showed lower levels of Ki-67 (MKI67, FC = 0.17 and P = .008) and higher levels of RAR-related orphan receptor C (RORC) (FC = 3.1 and P ˂ .001). When a cut-off of no detectable expression was used for Ki-67, the model provided a sensitivity of 100% and a specificity of 52.6% with an area under the curve of 65.8%. Using a cut-off of 2 units of relative expression of RORC, the prediction model showed 100% of sensitivity and specificity.
CONCLUSIONS: High levels of RORC and low levels of Ki-67 identify improved SRLs response after surgical debulking in large somatotropic adenomas. To determine their expression would facilitate medical treatment decision-making after surgery.
© 2020 John Wiley & Sons Ltd.

Entities:  

Keywords:  zzm321990RORCzzm321990; Ki-67; acromegaly; somatostatin analogs; somatostatin receptor ligands; transsphenoidal surgery

Year:  2021        PMID: 32978826     DOI: 10.1111/cen.14339

Source DB:  PubMed          Journal:  Clin Endocrinol (Oxf)        ISSN: 0300-0664            Impact factor:   3.478


  4 in total

1.  Implications of Heterogeneity of Epithelial-Mesenchymal States in Acromegaly Therapeutic Pharmacologic Response.

Authors:  Joan Gil; Montserrat Marques-Pamies; Elena Valassi; Araceli García-Martínez; Guillermo Serra; Cristina Hostalot; Carmen Fajardo-Montañana; Cristina Carrato; Ignacio Bernabeu; Mónica Marazuela; Helena Rodríguez-Lloveras; Rosa Cámara; Isabel Salinas; Cristina Lamas; Betina Biagetti; Andreu Simó-Servat; Susan M Webb; Antonio Picó; Mireia Jordà; Manel Puig-Domingo
Journal:  Biomedicines       Date:  2022-02-16

2.  Data mining analyses for precision medicine in acromegaly: a proof of concept.

Authors:  Joan Gil; Montserrat Marques-Pamies; Miguel Sampedro; Susan M Webb; Guillermo Serra; Isabel Salinas; Alberto Blanco; Elena Valassi; Cristina Carrato; Antonio Picó; Araceli García-Martínez; Luciana Martel-Duguech; Teresa Sardon; Andreu Simó-Servat; Betina Biagetti; Carles Villabona; Rosa Cámara; Carmen Fajardo-Montañana; Cristina Álvarez-Escolá; Cristina Lamas; Clara V Alvarez; Ignacio Bernabéu; Mónica Marazuela; Mireia Jordà; Manel Puig-Domingo
Journal:  Sci Rep       Date:  2022-05-28       Impact factor: 4.996

Review 3.  Pasireotide in the Personalized Treatment of Acromegaly.

Authors:  Manel Puig-Domingo; Ignacio Bernabéu; Antonio Picó; Betina Biagetti; Joan Gil; Cristina Alvarez-Escolá; Mireia Jordà; Montserrat Marques-Pamies; Berta Soldevila; María-Angeles Gálvez; Rosa Cámara; Javier Aller; Cristina Lamas; Mónica Marazuela
Journal:  Front Endocrinol (Lausanne)       Date:  2021-03-16       Impact factor: 5.555

4.  Epithelial-Mesenchymal Transition in the Resistance to Somatostatin Receptor Ligands in Acromegaly.

Authors:  Joan Gil; Mireia Jordà; Berta Soldevila; Manel Puig-Domingo
Journal:  Front Endocrinol (Lausanne)       Date:  2021-03-15       Impact factor: 5.555

  4 in total

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