Literature DB >> 32938211

Bisubstrate inhibitors: the promise of a selective and potent chemical inhibition of epigenetic 'writers'.

Corentin Bon1, Ludovic Halby1, Paola Barbara Arimondo1.   

Abstract

Keywords:  DNA; DNMT; HMT; SAM analogues; bisubstrate inhibitors; epigenetics; histone; methyltransferases; substrate analogues

Year:  2020        PMID： 32938211     DOI： 10.2217/epi-2020-0203

Source DB:  PubMed          Journal:  Epigenomics        ISSN： 1750-192X            Impact factor:   4.778


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  1 in total

1.  Synthesis and Biological Activity of a Cytostatic Inhibitor of MLLr Leukemia Targeting the DOT1L Protein.

Authors:  Corentin Bon; Yang Si; Melanie Pernak; Magdalena Barbachowska; Eva Levi-Acobas; Veronique Cadet Daniel; Corinne Jallet; Dusan Ruzic; Nemanja Djokovic; Teodora Djikić; Katarina Nikolic; Ludovic Halby; Paola B Arimondo
Journal:  Molecules       Date:  2021-08-31       Impact factor: 4.411
  1 in total

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