Literature DB >> 32554060

pH-dependent ileocolonic drug delivery, part I: in vitro and clinical evaluation of novel systems.

Annemarie Broesder1, Herman J Woerdenbag1, Grietje H Prins1, Duong N Nguyen1, Henderik W Frijlink1, Wouter L J Hinrichs2.   

Abstract

After the pH dependency of novel pH-dependent ileocolonic drug delivery systems is confirmed in vitro, their performance should be evaluated in human volunteers.
Copyright © 2020 The Author(s). Published by Elsevier Ltd.. All rights reserved.

Entities:  

Year:  2020        PMID: 32554060     DOI: 10.1016/j.drudis.2020.06.011

Source DB:  PubMed          Journal:  Drug Discov Today        ISSN: 1359-6446            Impact factor:   7.851


  3 in total

1.  A novel bedtime pulsatile-release caffeine formula ameliorates sleep inertia symptoms immediately upon awakening.

Authors:  Dario A Dornbierer; Firat Yerlikaya; Rafael Wespi; Martina I Boxler; Clarissa D Voegel; Laura Schnider; Aslihan Arslan; Diego M Baur; Markus R Baumgartner; Tina Maria Binz; Thomas Kraemer; Hans-Peter Landolt
Journal:  Sci Rep       Date:  2021-10-05       Impact factor: 4.379

2.  Ileo-Colon Targeting of the Poorly Water-Soluble Drug Celecoxib Using a pH-Dependent Coating in Combination with Self-Emulsifying Drug Delivery or Solid Dispersion Systems.

Authors:  Annemarie Broesder; Julia M E Berends; Sophie M Scheepers; Duong N Nguyen; Henderik W Frijlink; Wouter L J Hinrichs
Journal:  Pharmaceutics       Date:  2021-05-15       Impact factor: 6.321

3.  Formulation and In Vitro Evaluation of Pellets Containing Sulfasalazine and Caffeine to Verify Ileo-Colonic Drug Delivery.

Authors:  Annemarie Broesder; Said Y Bircan; Anneko B de Waard; Anko C Eissens; Henderik W Frijlink; Wouter L J Hinrichs
Journal:  Pharmaceutics       Date:  2021-11-23       Impact factor: 6.321

  3 in total

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