Literature DB >> 32387417

Treatment with abiraterone and enzalutamide does not overcome poor outcome from metastatic castration-resistant prostate cancer in men with the germline homozygous HSD3B1 c.1245C genotype.

C Lu1, A Terbuch2, D Dolling3, J Yu1, H Wang4, Y Chen1, J Fountain1, C Bertan3, A Sharp5, S Carreira3, W B Isaacs6, E S Antonarakis6, J S De Bono5, J Luo7.   

Abstract

BACKGROUND: In men with castration-sensitive prostate cancer (CSPC), the HSD3B1 c.1245A>C variant has been reported to be associated with shorter responses to first-line androgen-deprivation therapy (ADT). Here, we evaluated the association between the inherited HSD3B1 c.1245A>C variant and outcomes from metastatic castration-resistant prostate cancer (mCRPC) after first-line treatment with abiraterone (Abi) or enzalutamide (Enza). PATIENTS AND METHODS: Patients with mCRPC (n = 266) were enrolled from two centers at the time of starting first-line Abi/Enza. Outcomes after Abi/Enza included best prostate-specific antigen (PSA) response, treatment duration, and overall survival (OS). Outcomes after first-line ADT were determined retrospectively, and included treatment duration and OS. As was prespecified, we compared patients with the homozygous variant HSD3B1 genotype (CC genotype) versus the combined group with the heterozygous (AC) and homozygous wild-type (AA) genotypes.
RESULTS: Among the 266 patients, 22 (8.3%) were homozygous for the HSD3B1 variant (CC). The CC genotype had no association with PSA response rate; the median Abi/Enza treatment duration was 7.1 months for the CC group and 10.3 months for the AA/AC group (log rank P = 0.34). Patients with the CC genotype had significantly worse OS, with median survival at 23.6 months for the CC group and 30.7 months for the AA/AC group (log rank P = 0.02). In multivariable analysis adjusting for age, Gleason score, PSA, prior chemotherapy, and M1 disease, the association between the CC genotype and OS remained significant (hazard ratio 1.78, 95% confidence interval 1.03-3.07, P = 0.04). Poor outcome after first-line ADT in the CC group was also observed when evaluating retrospective ADT duration data for the same combined cohort.
CONCLUSIONS: In this large two-center study evaluating the HSD3B1 c.1245 genotype and outcomes after first-line Abi/Enza, homozygous variant (CC) HSD3B1 genotype was associated with worse outcomes. Novel therapeutic strategies are needed to enable treatment selection based on this genetic marker.
Copyright © 2020 European Society for Medical Oncology. Published by Elsevier Ltd. All rights reserved.

Entities:  

Keywords:  HSD3B1; abiraterone; androgen-deprivation therapy; biomarker; enzalutamide; mCRPC

Mesh:

Substances:

Year:  2020        PMID: 32387417     DOI: 10.1016/j.annonc.2020.04.473

Source DB:  PubMed          Journal:  Ann Oncol        ISSN: 0923-7534            Impact factor:   32.976


  10 in total

1.  Circulating and Intratumoral Adrenal Androgens Correlate with Response to Abiraterone in Men with Castration-Resistant Prostate Cancer.

Authors:  Elahe A Mostaghel; Brett T Marck; Orpheus Kolokythas; Felix Chew; Evan Y Yu; Michael T Schweizer; Heather H Cheng; Phillip W Kantoff; Steven P Balk; Mary-Ellen Taplin; Nima Sharifi; Alvin M Matsumoto; Peter S Nelson; R Bruce Montgomery
Journal:  Clin Cancer Res       Date:  2021-08-18       Impact factor: 12.531

2.  Management of prostate cancer by targeting 3βHSD1 after enzalutamide and abiraterone treatment.

Authors:  Zejie Mei; Tao Yang; Ying Liu; Yuanyuan Gao; Zemin Hou; Qian Zhuang; Dongyin He; Xuebin Zhang; Qilong Tan; Xuyou Zhu; Yingyi Qin; Xi Chen; Chengdang Xu; Cuidong Bian; Xinan Wang; Chenyang Wang; Denglong Wu; Shengsong Huang; Zhenfei Li
Journal:  Cell Rep Med       Date:  2022-04-20

3.  Targeting backdoor androgen synthesis through AKR1C3 inhibition: A presurgical hormonal ablative neoadjuvant trial in high-risk localized prostate cancer.

Authors:  Laura S Graham; Lawrence D True; Roman Gulati; George R Schade; Jonathan Wright; Petros Grivas; Todd Yezefski; Katie Nega; Katerina Alexander; Wen-Min Hou; Evan Y Yu; Bruce Montgomery; Elahe A Mostaghel; Alvin A Matsumoto; Brett Marck; Nima Sharifi; William J Ellis; Nicholas P Reder; Daniel W Lin; Peter S Nelson; Michael T Schweizer
Journal:  Prostate       Date:  2021-03-23       Impact factor: 4.104

Review 4.  Hormonal Therapy for Prostate Cancer.

Authors:  Kunal Desai; Jeffrey M McManus; Nima Sharifi
Journal:  Endocr Rev       Date:  2021-05-25       Impact factor: 19.871

Review 5.  Clinical implications of genomic alterations in metastatic prostate cancer.

Authors:  Takayuki Sumiyoshi; Kim N Chi; Alexander W Wyatt
Journal:  Prostate Cancer Prostatic Dis       Date:  2021-01-15       Impact factor: 5.455

6.  Observational study on time on treatment with abiraterone and enzalutamide.

Authors:  Giuseppe Fallara; Ingela Franck Lissbrant; Johan Styrke; Francesco Montorsi; Hans Garmo; Pär Stattin
Journal:  PLoS One       Date:  2020-12-28       Impact factor: 3.240

7.  Inhibiting 3βHSD1 to eliminate the oncogenic effects of progesterone in prostate cancer.

Authors:  Zemin Hou; Shengsong Huang; Zejie Mei; Longlong Chen; Jiacheng Guo; Yuanyuan Gao; Qian Zhuang; Xuebin Zhang; Qilong Tan; Tao Yang; Ying Liu; Yongnan Chi; Lifengrong Qi; Ting Jiang; Xuefeng Shao; Yan Wu; Xiaojun Xu; Jun Qin; Ruobing Ren; Huiru Tang; Denglong Wu; Zhenfei Li
Journal:  Cell Rep Med       Date:  2022-03-15

8.  Association Between Adrenal-Restrictive HSD3B1 Inheritance and Hormone-Independent Subtypes of Endometrial and Breast Cancer.

Authors:  Jeffrey M McManus; Roberto Vargas; Peter S Bazeley; Fredrick R Schumacher; Nima Sharifi
Journal:  JNCI Cancer Spectr       Date:  2022-09-01

Review 9.  Germline HSD3B1 Genetics and Prostate Cancer Outcomes.

Authors:  Lewis Thomas; Nima Sharifi
Journal:  Urology       Date:  2020-08-28       Impact factor: 2.649

10.  Combined Longitudinal Clinical and Autopsy Phenomic Assessment in Lethal Metastatic Prostate Cancer: Recommendations for Advancing Precision Medicine.

Authors:  Juho Jasu; Teemu Tolonen; Emmanuel S Antonarakis; Himisha Beltran; Susan Halabi; Mario A Eisenberger; Michael A Carducci; Yohann Loriot; Kim Van der Eecken; Martijn Lolkema; Charles J Ryan; Sinja Taavitsainen; Silke Gillessen; Gunilla Högnäs; Timo Talvitie; Robert J Taylor; Antti Koskenalho; Piet Ost; Teemu J Murtola; Irina Rinta-Kiikka; Teuvo Tammela; Anssi Auvinen; Paula Kujala; Thomas J Smith; Pirkko-Liisa Kellokumpu-Lehtinen; William B Isaacs; Matti Nykter; Juha Kesseli; G Steven Bova
Journal:  Eur Urol Open Sci       Date:  2021-07-02
  10 in total

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