Literature DB >> 32081463

Phase Ib study of mirvetuximab soravtansine, a folate receptor alpha (FRα)-targeting antibody-drug conjugate (ADC), in combination with bevacizumab in patients with platinum-resistant ovarian cancer.

David M O'Malley1, Ursula A Matulonis2, Michael J Birrer3, Cesar M Castro4, Lucy Gilbert5, Ignace Vergote6, Lainie P Martin7, Gina M Mantia-Smaldone8, Antonio González Martin9, Raquel Bratos10, Richard T Penson11, Karim Malek12, Kathleen N Moore13.   

Abstract

PURPOSE: To evaluate the safety and clinical activity of mirvetuximab soravtansine, an antibody-drug conjugate comprising a humanized anti-folate receptor alpha (FRα) monoclonal antibody, cleavable linker, and the maytansinoid DM4, a potent tubulin-targeting agent, in combination with bevacizumab in patients with FRα-positive, platinum-resistant ovarian cancer.
METHODS: Patients with platinum-resistant epithelial ovarian, fallopian tube, or primary peritoneal cancer were administered mirvetuximab soravtansine (6 mg/kg, adjusted ideal body weight) and bevacizumab (15 mg/kg) once every 3 weeks. Eligibility included FRα positivity by immunochemistry and prior bevacizumab exposure was permitted. Adverse events, tumor response, and progression-free survival (PFS) were determined.
RESULTS: Sixty-six patients, with a median of 3 prior lines of therapy (range, 1-8), received the combination of mirvetuximab soravtansine and bevacizumab at full dosing during the escalation and expansion stages of the study. Adverse events were generally mild-to-moderate (≤grade 2) with diarrhea, blurred vision, nausea, and fatigue being the most common treatment-related toxicities. Six cases of pneumonitis (9%; all grade 1 or 2), an adverse event of special interest, were observed. The confirmed objective response rate (ORR) was 39%, including 5 complete responses and 21 partial responses, and the median PFS was 6.9 months. The combination was particularly active in the subset of patients (n = 16) who were bevacizumab-naïve, less heavily pretreated (1-2 prior lines), and whose tumors exhibited medium/high FRα expression (ORR, 56% with a median duration of response of 12 months; PFS, 9.9 months).
CONCLUSION: The combination of mirvetuximab soravtansine with bevacizumab is well tolerated in patients with platinum-resistant, recurrent ovarian cancer. The encouraging efficacy measures compare favorably to reported outcomes for bevacizumab combined with standard chemotherapy in similar patient populations.
Copyright © 2020 Elsevier Inc. All rights reserved.

Entities:  

Year:  2020        PMID: 32081463     DOI: 10.1016/j.ygyno.2020.01.037

Source DB:  PubMed          Journal:  Gynecol Oncol        ISSN: 0090-8258            Impact factor:   5.482


  22 in total

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2.  Identification of CD8+ T Cell Related Biomarkers in Ovarian Cancer.

Authors:  Ling Li; Dian Chen; Xiaolin Luo; Zhengkun Wang; Hanjie Yu; Weicheng Gao; Weiqiang Zhong
Journal:  Front Genet       Date:  2022-05-27       Impact factor: 4.772

3.  Phase II trial of bevacizumab and sorafenib in recurrent ovarian cancer patients with or without prior-bevacizumab treatment.

Authors:  Jung-Min Lee; Christina M Annunziata; John L Hays; Liang Cao; Peter Choyke; Minshu Yu; Daniel An; Ismail Baris Turkbey; Lori M Minasian; Seth M Steinberg; Helen Chen; John Wright; Elise C Kohn
Journal:  Gynecol Oncol       Date:  2020-08-01       Impact factor: 5.482

Review 4.  Novel antibody-drug conjugates: current and future roles in gynecologic oncology.

Authors:  Joan Tymon-Rosario; Burak Zeybek; Alessandro D Santin
Journal:  Curr Opin Obstet Gynecol       Date:  2021-02-01       Impact factor: 1.927

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Journal:  Nat Rev Clin Oncol       Date:  2021-02-08       Impact factor: 65.011

Review 6.  Cancer of the ovary, fallopian tube, and peritoneum: 2021 update.

Authors:  Jonathan S Berek; Malte Renz; Sean Kehoe; Lalit Kumar; Michael Friedlander
Journal:  Int J Gynaecol Obstet       Date:  2021-10       Impact factor: 4.447

7.  Corneal Epithelial Findings in Patients with Multiple Myeloma Treated with Antibody-Drug Conjugate Belantamab Mafodotin in the Pivotal, Randomized, DREAMM-2 Study.

Authors:  Asim V Farooq; Simona Degli Esposti; Rakesh Popat; Praneetha Thulasi; Sagar Lonial; Ajay K Nooka; Andrzej Jakubowiak; Douglas Sborov; Brian E Zaugg; Ashraf Z Badros; Bennie H Jeng; Natalie S Callander; Joanna Opalinska; January Baron; Trisha Piontek; Julie Byrne; Ira Gupta; Kathryn Colby
Journal:  Ophthalmol Ther       Date:  2020-07-25

Review 8.  Progress in Gynecologic Cancers with Antibody Drug Conjugates.

Authors:  David M O'Malley; Corinne A Calo
Journal:  Curr Oncol Rep       Date:  2021-06-14       Impact factor: 5.075

Review 9.  Stepping forward in antibody-drug conjugate development.

Authors:  Yiming Jin; Megan A Schladetsch; Xueting Huang; Marcy J Balunas; Andrew J Wiemer
Journal:  Pharmacol Ther       Date:  2021-06-24       Impact factor: 12.310

Review 10.  The promising role of antibody drug conjugate in cancer therapy: Combining targeting ability with cytotoxicity effectively.

Authors:  Wen-Qian Li; Han-Fei Guo; Ling-Yu Li; Yong-Fei Zhang; Jiu-Wei Cui
Journal:  Cancer Med       Date:  2021-06-24       Impact factor: 4.452

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