Literature DB >> 32030406

The algorithm used for the interpretation of doravirine transmitted drug resistance strongly influences clinical practice and guideline recommendations.

Carlos Guerrero-Beltrán1, Javier Martínez-Sanz2, Marta Álvarez1, Julián Olalla3, Mónica García-Álvarez4, Jose Antonio Iribarren5, Mar Masiá6, Marta Montero7, Silvia García-Bujalance8, José Ramón Blanco9, María Rivero10, Lucio Jesús García-Fraile11, Núria Espinosa12, Carmen Rodríguez13, Antonio Aguilera14, María Carmen Vidal-Ampurdanes15, Marina Martínez16, Asunción Iborra17, Arkaitz Imaz18, Juan Luis Gómez-Sirvent19, Joaquim Peraire20, Joaquín Portilla21, Estrella Caballero22, Belén Alejos23, Federico García1, Santiago Moreno2.   

Abstract

OBJECTIVES: We report the results of the reverse transcriptase (RT)/protease (PR) transmitted drug resistance (TDR) prevalence study in 2018, focusing on doravirine resistance-associated mutations and the differences observed when Stanford or French National Agency for AIDS Research (ANRS)/Spanish Network of AIDS Research (RIS)/IAS-USA resistance interpretation algorithms are used to describe clinically relevant resistance.
METHODS: We used the WHO 2009 list to investigate the prevalence of NNRTI, NRTI and PI TDR, in treatment-naive HIV-1-infected patients, adding mutations E138A/G/K/Q/R, V106I, V108I, V179L, G190Q, H221Y, F227C/L/V, M230IDR, L234I, P236L and Y318F in RT. The prevalence of doravirine resistance-associated mutations, as described by Soulie et al. in 2019, was evaluated. Clinically relevant TDR was investigated using the latest versions of ANRS, RIS, IAS-USA and Stanford algorithms.
RESULTS: NNRTI mutations were detected in 82 of 606 (13.5%) patients. We found 18 patients (3.0%) with NRTI mutations and 5 patients (0.8%) with PI mutations. We detected 11 patients harbouring doravirine resistance-associated mutations (prevalence of 1.8%). Furthermore, we observed important differences in clinically relevant resistance to doravirine when ANRS/RIS (0.7%), IAS-USA (0.5%) or Stanford algorithms (5.0%) were used. V106I, which was detected in 3.8% of the patients, was the main mutation driving these differences. V106I detection was not associated with any of the clinical, demographic or virological characteristics of the patients.
CONCLUSIONS: The prevalence of NRTI and PI TDR remains constant in Spain. Doravirine TDR is very infrequent by RIS/ANRS/IAS-USA algorithms, in contrast with results using the Stanford algorithm. Further genotype-phenotype studies are necessary to elucidate the role of V106I in doravirine resistance.
© The Author(s) 2020. Published by Oxford University Press on behalf of the British Society for Antimicrobial Chemotherapy. All rights reserved. For permissions, please email: journals.permissions@oup.com.

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Year:  2020        PMID: 32030406     DOI: 10.1093/jac/dkaa009

Source DB:  PubMed          Journal:  J Antimicrob Chemother        ISSN: 0305-7453            Impact factor:   5.790


  5 in total

Review 1.  Doravirine and Its Potential in the Treatment of HIV: An Evidence-Based Review of the Emerging Data.

Authors:  Alexander E Rock; Jeremy Lerner; Melissa E Badowski
Journal:  HIV AIDS (Auckl)       Date:  2020-06-10

2.  Is there a role for doravirine in African HIV treatment programmes? A large observational resistance study in South Africa.

Authors:  Kim Steegen; Michelle Moorhouse; Annemarie Mj Wensing; Willem Df Venter; Lucia Hans
Journal:  J Int AIDS Soc       Date:  2021-05       Impact factor: 5.396

3.  High Prevalence of Doravirine Resistance in HIV-1-Infected Patients with Virological Failure to an NNRTI-Based Single-Tablet Regimen.

Authors:  Hung-Chin Tsai; I-Tzu Chen; Hui-Min Chang; Susan Shin-Jung Lee; Yao-Shen Chen
Journal:  Infect Drug Resist       Date:  2022-07-20       Impact factor: 4.177

4.  In vitro cross-resistance to doravirine in a panel of HIV-1 clones harbouring multiple NNRTI resistance mutations.

Authors:  Francesco Saladini; Federica Giammarino; Behnaz A Hosseini; Alessia Giannini; Adele Boccuto; Filippo Dragoni; Ilaria Vicenti; Robert W Shafer; Maurizio Zazzi
Journal:  J Antimicrob Chemother       Date:  2021-01-01       Impact factor: 5.790

5.  Impact of HIV-1 Resistance-Associated Mutations on Susceptibility to Doravirine: Analysis of Real-World Clinical Isolates.

Authors:  Ernest Asante-Appiah; Johnny Lai; Hong Wan; Dongmei Yang; Elizabeth Anne Martin; Peter Sklar; Daria Hazuda; Christos J Petropoulos; Charles Walworth; Jay A Grobler
Journal:  Antimicrob Agents Chemother       Date:  2021-09-27       Impact factor: 5.191

  5 in total

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