Literature DB >> 32007513

Serlopitant for psoriatic pruritus: A phase 2 randomized, double-blind, placebo-controlled clinical trial.

David M Pariser1, Jerry Bagel2, Mark Lebwohl3, Gil Yosipovitch4, Elaine Chien5, Mary C Spellman6.   

Abstract

BACKGROUND: Pruritus, a common symptom of psoriasis, negatively affects quality of life; however, treatment of lesional skin does not consistently alleviate psoriatic itch.
OBJECTIVE: To examine the effects of serlopitant, an oral, once-daily neurokinin 1 receptor antagonist, for treatment of psoriatic pruritus in a phase 2, randomized clinical trial (NCT03343639).
METHODS: Patients (n = 204) were randomized to receive serlopitant, 5 mg, or placebo daily for 8 weeks. Eligible adult patients had plaque psoriasis for ≥6 months, plaques covering ≤10% of body surface area, pruritus for ≥4 weeks, and Worst Itch Numeric Rating Scale (WI-NRS) score ≥7 at the initial screening.
RESULTS: Participants (54.2% women) had a mean age of 47.5 years and 85.2% were white. Mean baseline WI-NRS scores were 8.3 for serlopitant and 8.1 for placebo. The WI-NRS 4-point response rate at 8 weeks (primary end point) was 33.3% for serlopitant vs 21.1% for placebo (P = .028); at 4 weeks the rates were 20.8% for serlopitant vs 11.5% for placebo (P = .039). Treatment-related adverse events were reported for 4.9% of serlopitant-treated and 4.0% of placebo-treated patients. LIMITATIONS: This was a phase 2 study with a small study population. Patients with severe psoriasis were excluded.
CONCLUSION: Serlopitant significantly reduced pruritus associated with mild to moderate psoriasis, supporting continued development of serlopitant for this patient population.
Copyright © 2020. Published by Elsevier Inc.

Entities:  

Keywords:  clinical trial; neurokinin 1 receptor (NK(1)R); pruritus; psoriasis; serlopitant; substance P

Year:  2020        PMID: 32007513     DOI: 10.1016/j.jaad.2020.01.056

Source DB:  PubMed          Journal:  J Am Acad Dermatol        ISSN: 0190-9622            Impact factor:   11.527


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3.  Role of Mast Cells in the Pathogenesis of Pruritus in Mastocytosis.

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Authors:  Changxiong J Guo; Nathaniel S Grabinski; Qin Liu
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5.  The Neurokinin-1 Receptor is Expressed with Gastrin-Releasing Peptide Receptor in Spinal Interneurons and Modulates Itch.

Authors:  Tayler D Sheahan; Charles A Warwick; Louis G Fanien; Sarah E Ross
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Review 7.  New Frontiers in Psoriatic Disease Research, Part II: Comorbidities and Targeted Therapies.

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Review 8.  Molecular and Cellular Mechanisms of Itch in Psoriasis.

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Review 9.  Emerging Therapeutic Options for Chronic Pruritus.

Authors:  Radomir Reszke; Piotr Krajewski; Jacek C Szepietowski
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Review 10.  Molecular Aspects of Pruritus Pathogenesis in Psoriasis.

Authors:  Kamila Jaworecka; Joanna Muda-Urban; Marian Rzepko; Adam Reich
Journal:  Int J Mol Sci       Date:  2021-01-16       Impact factor: 5.923

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