Literature DB >> 31967355

PET Molecular Imaging of Phosphodiesterase 10A: An Early Biomarker of Huntington's Disease Progression.

Patrik Fazio1, Cheryl J Fitzer-Attas2, Ladislav Mrzljak2, Juliana Bronzova3, Sangram Nag1, John H Warner2, Bernhard Landwehrmeyer3, Nabil Al-Tawil4, Christer Halldin1, Anton Forsberg1, Jennifer Ware2, Valentina Dilda2, Andrew Wood2, Cristina Sampaio2, Andrea Varrone1.   

Abstract

BACKGROUND: Changes in phosphodiesterase 10A enzyme levels may be a suitable biomarker of disease progression in Huntington's disease.
OBJECTIVES: To evaluate phosphodiesterase 10A PET imaging as a biomarker of HD progression using the radioligand, [18 F]MNI-659.
METHODS: The cross-sectional study (NCT02061722) included 45 Huntington's disease gene-expansion carriers stratified into four disease stages (early and late premanifest and Huntington's disease stages 1 and 2) and 45 age- and sex-matched healthy controls. The primary analysis compared striatal and pallidal phosphodiesterase 10A availability between Huntington's disease gene-expansion carriers and healthy controls as assessed by [18 F]MNI-659 binding. We assessed changes in phosphodiesterase 10A expression using several PET methodologies and compared with previously proposed measures of Huntington's disease progression (PET imaging of D2/3 receptors and anatomical volume loss on MRI). The longitudinal follow-up study (NCT02956148) continued evaluation of phosphodiesterase 10A availability in 35 Huntington's disease gene-expansion carriers at a mean of 18 months from baseline of the cross-sectional study.
RESULTS: Primary analyses revealed that phosphodiesterase 10A availability in caudate, putamen, and globus pallidus was significantly lower in Huntington's disease gene-expansion carriers versus healthy controls across all stages. Striatal and pallidal phosphodiesterase 10A availability progressively declined in the premanifest stages and appeared to plateau between stages 1 and 2. The percentage decline of phosphodiesterase 10A availability measured cross-sectionally between Huntington's disease gene-expansion carriers and healthy controls was greater than that demonstrated by D2/3 receptor availability or volumetric changes. Annualized rates of phosphodiesterase 10A change showed a statistically significant decline between the cross-sectional study and follow-up.
CONCLUSIONS: [18 F]MNI-659 PET imaging is a biologically plausible biomarker of Huntington's disease progression that is more sensitive than the dopamine-receptor and volumetric methods currently used.
© 2020 International Parkinson and Movement Disorder Society. © 2020 International Parkinson and Movement Disorder Society.

Entities:  

Keywords:  Huntington's disease; PDE10A; biomarker; imaging

Mesh:

Substances:

Year:  2020        PMID: 31967355     DOI: 10.1002/mds.27963

Source DB:  PubMed          Journal:  Mov Disord        ISSN: 0885-3185            Impact factor:   10.338


  7 in total

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Authors:  Sarah J Tabrizi; Carlos Estevez-Fraga; Willeke M C van Roon-Mom; Michael D Flower; Rachael I Scahill; Edward J Wild; Ignacio Muñoz-Sanjuan; Cristina Sampaio; Anne E Rosser; Blair R Leavitt
Journal:  Lancet Neurol       Date:  2022-07       Impact factor: 59.935

Review 2.  A Glimpse of Molecular Biomarkers in Huntington's Disease.

Authors:  Silvia Martí-Martínez; Luis M Valor
Journal:  Int J Mol Sci       Date:  2022-05-12       Impact factor: 6.208

3.  Exome sequencing revealed PDE11A as a novel candidate gene for early-onset Alzheimer's disease.

Authors:  Wei Qin; Aihong Zhou; Xiumei Zuo; Longfei Jia; Fangyu Li; Qi Wang; Ying Li; Yiping Wei; Hongmei Jin; Carlos Cruchaga; Bruno A Benitez; Jianping Jia
Journal:  Hum Mol Genet       Date:  2021-05-28       Impact factor: 5.121

Review 4.  Challenges on Cyclic Nucleotide Phosphodiesterases Imaging with Positron Emission Tomography: Novel Radioligands and (Pre-)Clinical Insights since 2016.

Authors:  Susann Schröder; Matthias Scheunemann; Barbara Wenzel; Peter Brust
Journal:  Int J Mol Sci       Date:  2021-04-07       Impact factor: 5.923

5.  Inhibition of PDE10A-Rescued TBI-Induced Neuroinflammation and Apoptosis through the cAMP/PKA/NLRP3 Pathway.

Authors:  Jin Huang; Dang Tang; Yiqiang Cao; Yonggang Wang; Jiang Long; Lin Wei; Hai Song
Journal:  Evid Based Complement Alternat Med       Date:  2022-04-12       Impact factor: 2.650

Review 6.  Drugging DNA Damage Repair Pathways for Trinucleotide Repeat Expansion Diseases.

Authors:  Caroline L Benn; Karl R Gibson; David S Reynolds
Journal:  J Huntingtons Dis       Date:  2021

Review 7.  The Use, Standardization, and Interpretation of Brain Imaging Data in Clinical Trials of Neurodegenerative Disorders.

Authors:  Adam J Schwarz
Journal:  Neurotherapeutics       Date:  2021-04-12       Impact factor: 7.620

  7 in total

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