Literature DB >> 31829907

Randomized Phase III Study of Ganetespib, a Heat Shock Protein 90 Inhibitor, With Docetaxel Versus Docetaxel in Advanced Non-Small-Cell Lung Cancer (GALAXY-2).

Rathi N Pillai1, Dean A Fennell2, Vladimir Kovcin3, Tudor-Eliade Ciuleanu4, Rodryg Ramlau5, Dariusz Kowalski6, Michael Schenker7, Ilker Yalcin8, Florentina Teofilovici8, Vojo M Vukovic8, Suresh S Ramalingam1.   

Abstract

PURPOSE: Ganetespib, a highly potent heat shock protein 90 inhibitor, blocks multiple oncogenic pathways, resulting in antitumor activity. We evaluated the combination of ganetespib and docetaxel for second-line therapy of patients with advanced adenocarcinoma of the lung. PATIENTS AND METHODS: In this international phase III trial, patients with stage IIIB or IV adenocarcinoma diagnosed > 6 months before study entry and 1 prior systemic therapy were randomly assigned (1:1) to ganetespib 150 mg/m2 on days 1 and 15 with docetaxel 75 mg/m2 on day 1 of a 21-day cycle or to docetaxel alone. The primary end point was overall survival (OS).
RESULTS: Of 677 enrolled patients, 335 were randomly assigned to ganetespib and docetaxel and 337 were assigned to docetaxel. The trial was stopped early as a result of futility at a planned interim analysis. The median OS time was 10.9 months (95% CI, 9.0 to 12.3 months) in the ganetespib and docetaxel arm compared with 10.5 months (95% CI, 8.6 to 12.2 months) in docetaxel arm (hazard ratio [HR], 1.11; 95% CI, 0.899 to 1.372; P = .329). Median progression-free survival was 4.2 months in the ganetespib and docetaxel arm and 4.3 months in the docetaxel arm (HR, 1.16; 95% CI, 0.96 to 1.403; P = .119). The addition of ganetespib did not improve outcomes compared with docetaxel alone for any secondary end point, including survival in the elevated lactate dehydrogenase or EGFR and ALK wild-type populations. The most common grade 3 or 4 adverse event in both arms was neutropenia (30.9% with ganetespib and docetaxel v 25% with docetaxel).
CONCLUSION: The addition of ganetespib to docetaxel did not result in improved survival for salvage therapy of patients with advanced-stage lung adenocarcinoma.

Entities:  

Year:  2019        PMID: 31829907     DOI: 10.1200/JCO.19.00816

Source DB:  PubMed          Journal:  J Clin Oncol        ISSN: 0732-183X            Impact factor:   44.544


  12 in total

1.  Hsp90 Inhibitor STA9090 Sensitizes Hepatocellular Carcinoma to Hyperthermia-Induced DNA Damage by Suppressing DNA-PKcs Protein Stability and mRNA Transcription.

Authors:  Lixia Liu; Yaotang Deng; Zhenming Zheng; Zihao Deng; Jinxin Zhang; Jieyou Li; Manfeng Liang; Xueqiong Zhou; Wenchong Tan; Hongjun Yang; Leonard M Neckers; Fei Zou; Xuemei Chen
Journal:  Mol Cancer Ther       Date:  2021-08-10       Impact factor: 6.009

2.  Novel T7-Modified pH-Responsive Targeted Nanosystem for Co-Delivery of Docetaxel and Curcumin in the Treatment of Esophageal Cancer.

Authors:  Lian Deng; Xiongjie Zhu; Zhongjian Yu; Ying Li; Lingyu Qin; Zhile Liu; Longbao Feng; Rui Guo; Yanfang Zheng
Journal:  Int J Nanomedicine       Date:  2020-10-09

3.  HSP90 Inhibitor, 17-DMAG, Alone and in Combination with Lapatinib Attenuates Acquired Lapatinib-Resistance in ER-positive, HER2-Overexpressing Breast Cancer Cell Line.

Authors:  Hye Jin Lee; Seungho Shin; Jinho Kang; Ki-Cheol Han; Yeul Hong Kim; Jeoung-Won Bae; Kyong Hwa Park
Journal:  Cancers (Basel)       Date:  2020-09-15       Impact factor: 6.639

Review 4.  Oh, the Mutations You'll Acquire! A Systematic Overview of Cutaneous Squamous Cell Carcinoma.

Authors:  Stephenie Droll; Xiaomin Bao
Journal:  Cell Physiol Biochem       Date:  2021-09-22

5.  Potential predictive value of plasma heat shock protein 90α in lung cancer.

Authors:  Xiaoqian Li; Xuesong Tong; Bin Liu; Zeng Li; Jing Ding; Jiang Li; Min Zheng; Yuke Tian; Siyou Yan; Meiling Huang; Jun Ge
Journal:  J Int Med Res       Date:  2021-12       Impact factor: 1.671

6.  Impact of Value Frameworks on the Magnitude of Clinical Benefit: Evaluating a Decade of Randomized Trials for Systemic Therapy in Solid Malignancies.

Authors:  Ellen Cusano; Chelsea Wong; Eddy Taguedong; Marcus Vaska; Tasnima Abedin; Nancy Nixon; Safiya Karim; Patricia Tang; Daniel Y C Heng; Doreen Ezeife
Journal:  Curr Oncol       Date:  2021-11-21       Impact factor: 3.677

7.  Ganetespib selectively sensitizes cancer cells for proximal and distal spread-out Bragg peak proton irradiation.

Authors:  Simon Deycmar; Elisabeth Mara; Sylvia Kerschbaum-Gruber; Verena Waller; Dietmar Georg; Martin Pruschy
Journal:  Radiat Oncol       Date:  2022-04-11       Impact factor: 3.481

Review 8.  Targeting Heat-Shock Protein 90 in Cancer: An Update on Combination Therapy.

Authors:  Xiude Ren; Tao Li; Wei Zhang; Xuejun Yang
Journal:  Cells       Date:  2022-08-17       Impact factor: 7.666

Review 9.  KRAS oncogene may be another target conquered in non-small cell lung cancer (NSCLC).

Authors:  Hanxiao Chen; Jun Zhao
Journal:  Thorac Cancer       Date:  2020-10-06       Impact factor: 3.500

10.  Identification of Predictive Biomarkers of Response to HSP90 Inhibitors in Lung Adenocarcinoma.

Authors:  Ángela Marrugal; Irene Ferrer; David Gómez-Sánchez; Álvaro Quintanal-Villalonga; María Dolores Pastor; Laura Ojeda; Luis Paz-Ares; Sonia Molina-Pinelo
Journal:  Int J Mol Sci       Date:  2021-03-03       Impact factor: 5.923

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