Literature DB >> 31659377

PSPH-D-18-00526: Effect of a dual orexin receptor antagonist (DORA-12) on sleep and event-related oscillations in rats exposed to ethanol vapor during adolescence.

Cindy L Ehlers1, Jessica Benedict2, Derek Wills2, Manuel Sanchez-Alavez2.   

Abstract

RATIONALE: Sleep difficulties are one of the problems associated with adolescent binge drinking. However, the mechanisms underlying adolescent alcohol-associated sleep disturbances and potential targets for therapy remain under investigated. Orexin receptor antagonists may have therapeutic value in the treatment of insomnia, yet the use of this class of drugs in the treatment of sleep disturbances following adolescent alcohol exposure has not been studied.
OBJECTIVES: This study employed a model whereby ethanol vapor exposure occurred for 5 weeks during adolescence (AIE), and waking event-related oscillations (EROs) and EEG sleep were subsequently evaluated in young adult rats. The ability of two doses (10, 30 mg/kg PO) of a dual orexin receptor antagonist (DORA-12) to modify sleep, EEG, and EROs was investigated in AIE rats and controls.
RESULTS: Adolescent vapor exposure was found to produce a fragmentation of sleep, in young adults, that was partially ameliorated by DORA-12. DORA-12 also produced increases in delta and theta power in waking EROs recorded before sleep, and deeper sleep as indexed by increases in delta and theta power in the sleep EEG in both ethanol and control rats. Rats given DORA-12 also fell asleep faster than vehicle-treated rats as measured by a dose-dependent reduction in the latency to both the first slow wave and REM sleep episodes.
CONCLUSIONS: This study showed that DORA-12 can affect the sleep disturbance that is associated with a history of adolescent ethanol exposure and also has several other sleep-promoting effects that are equivalent in both ethanol and control rats.

Entities:  

Keywords:  Adolescence; Alcohol; DORA; EROs; Sleep

Year:  2019        PMID: 31659377      PMCID: PMC7186151          DOI: 10.1007/s00213-019-05371-4

Source DB:  PubMed          Journal:  Psychopharmacology (Berl)        ISSN: 0033-3158            Impact factor:   4.530


  84 in total

1.  Effect of Gabapentin on Sleep and Event-Related Oscillations (EROs) in Rats Exposed to Chronic Intermittent Ethanol Vapor and Protracted Withdrawal.

Authors:  Manuel Sanchez-Alavez; Derek N Wills; Leslie Amodeo; Cindy L Ehlers
Journal:  Alcohol Clin Exp Res       Date:  2018-01-31       Impact factor: 3.455

2.  Age at first drink and the first incidence of adult-onset DSM-IV alcohol use disorders.

Authors:  Deborah A Dawson; Risë B Goldstein; S Patricia Chou; W June Ruan; Bridget F Grant
Journal:  Alcohol Clin Exp Res       Date:  2008-09-30       Impact factor: 3.455

3.  Effects of adolescent ethanol exposure on sleep in adult rats.

Authors:  José R Criado; Derek N Wills; Brendan M Walker; Cindy L Ehlers
Journal:  Alcohol       Date:  2008-10-14       Impact factor: 2.405

4.  A randomized double-blind pilot trial of gabapentin versus placebo to treat alcohol dependence and comorbid insomnia.

Authors:  Kirk J Brower; Hyungjin Myra Kim; Stephen Strobbe; Maher A Karam-Hage; Flavia Consens; Robert A Zucker
Journal:  Alcohol Clin Exp Res       Date:  2008-06-06       Impact factor: 3.455

Review 5.  Orexin receptors: multi-functional therapeutic targets for sleeping disorders, eating disorders, drug addiction, cancers and other physiological disorders.

Authors:  Tian-Rui Xu; Yang Yang; Richard Ward; Linghuan Gao; Ying Liu
Journal:  Cell Signal       Date:  2013-08-01       Impact factor: 4.315

Review 6.  Suvorexant: scientifically interesting, utility uncertain.

Authors:  Nicholas A Keks; Judy Hope; Simone Keogh
Journal:  Australas Psychiatry       Date:  2017-10-10       Impact factor: 1.369

7.  An altered neural response to reward may contribute to alcohol problems among late adolescents with an evening chronotype.

Authors:  Brant P Hasler; Stephanie L Sitnick; Daniel S Shaw; Erika E Forbes
Journal:  Psychiatry Res       Date:  2013-10-18       Impact factor: 3.222

8.  Electrophysiological effects of dizocilpine (MK-801) in adult rats exposed to ethanol during adolescence.

Authors:  José R Criado; Derek N Wills; Brendan M Walker; Cindy L Ehlers
Journal:  Alcohol Clin Exp Res       Date:  2008-07-24       Impact factor: 3.455

9.  A longitudinal study of insomnia and other sleep complaints in adolescents with and without alcohol use disorders.

Authors:  Brant P Hasler; Christopher S Martin; D Scott Wood; Bedda Rosario; Duncan B Clark
Journal:  Alcohol Clin Exp Res       Date:  2014-06-27       Impact factor: 3.455

10.  Orexin-1 and orexin-2 receptor antagonists reduce ethanol self-administration in high-drinking rodent models.

Authors:  Rachel I Anderson; Howard C Becker; Benjamin L Adams; Cynthia D Jesudason; Linda M Rorick-Kehn
Journal:  Front Neurosci       Date:  2014-02-25       Impact factor: 4.677

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  2 in total

1.  Effects of an Orexin-2 Receptor Antagonist on Sleep and Event-Related Oscillations in Female Rats Exposed to Chronic Intermittent Ethanol During Adolescence.

Authors:  Leslie R Amodeo; Derek N Wills; Manuel Sanchez-Alavez; Cindy L Ehlers
Journal:  Alcohol Clin Exp Res       Date:  2020-06-12       Impact factor: 3.455

Review 2.  The role of sex in the persistent effects of adolescent alcohol exposure on behavior and neurobiology in rodents.

Authors:  Donita L Robinson; Leslie R Amodeo; L Judson Chandler; Fulton T Crews; Cindy L Ehlers; Alexander Gómez-A; Kati L Healey; Cynthia M Kuhn; Victoria A Macht; S Alexander Marshall; H Scott Swartzwelder; Elena I Varlinskaya; David F Werner
Journal:  Int Rev Neurobiol       Date:  2021-08-11       Impact factor: 4.280

  2 in total

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