Literature DB >> 31516029

Multi-target ABC transporter modulators: what next and where to go?

Sven Marcel Stefan1.   

Abstract

Keywords:  ABC transporter inhibition; ABCB1; ABCC1; ABCG2; Alzheimer's disease; BCRP; MRP1; P-gp; activation; activator; broad-spectrum inhibitor; modulation; modulator; multi-target; multidrug resistance

Year:  2019        PMID: 31516029     DOI: 10.4155/fmc-2019-0185

Source DB:  PubMed          Journal:  Future Med Chem        ISSN: 1756-8919            Impact factor:   3.808


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  15 in total

Review 1.  Research advances in the role and pharmaceuticals of ATP-binding cassette transporters in autoimmune diseases.

Authors:  Jun Yu; Hao Chen; Jiangmei Xu; Peng Zhou
Journal:  Mol Cell Biochem       Date:  2022-01-16       Impact factor: 3.396

2.  Strategies to gain novel Alzheimer's disease diagnostics and therapeutics using modulators of ABCA transporters.

Authors:  Jens Pahnke; Pablo Bascuñana; Mirjam Brackhan; Katja Stefan; Vigneshwaran Namasivayam; Radosveta Koldamova; Jingyun Wu; Luisa Möhle; Sven Marcel Stefan
Journal:  Free Neuropathol       Date:  2021-12-13

Review 3.  Unconventional Protein Secretion in Brain Tumors Biology: Enlightening the Mechanisms for Tumor Survival and Progression.

Authors:  Rebeca Piatniczka Iglesia; Mariana Brandão Prado; Rodrigo Nunes Alves; Maria Isabel Melo Escobar; Camila Felix de Lima Fernandes; Ailine Cibele Dos Santos Fortes; Maria Clara da Silva Souza; Jacqueline Marcia Boccacino; Giovanni Cangiano; Samuel Ribeiro Soares; João Pedro Alves de Araújo; Deanna Marie Tiek; Anshika Goenka; Xiao Song; Jack Ryan Keady; Bo Hu; Shi Yuan Cheng; Marilene Hohmuth Lopes
Journal:  Front Cell Dev Biol       Date:  2022-06-15

Review 4.  Overcoming Multidrug Resistance: Flavonoid and Terpenoid Nitrogen-Containing Derivatives as ABC Transporter Modulators.

Authors:  Bruno M F Gonçalves; David S P Cardoso; Maria-José U Ferreira
Journal:  Molecules       Date:  2020-07-24       Impact factor: 4.411

5.  C@PA: Computer-Aided Pattern Analysis to Predict Multitarget ABC Transporter Inhibitors.

Authors:  Vigneshwaran Namasivayam; Katja Silbermann; Michael Wiese; Jens Pahnke; Sven Marcel Stefan
Journal:  J Med Chem       Date:  2021-03-16       Impact factor: 7.446

6.  Structural feature-driven pattern analysis for multitarget modulator landscapes.

Authors:  Vigneshwaran Namasivayam; Katja Stefan; Katja Silbermann; Jens Pahnke; Michael Wiese; Sven Marcel Stefan
Journal:  Bioinformatics       Date:  2021-12-09       Impact factor: 6.937

Review 7.  Momordica balsamina: phytochemistry and pharmacological potential of a gifted species.

Authors:  Cátia Ramalhete; Bruno M F Gonçalves; Filipa Barbosa; Noélia Duarte; Maria-José U Ferreira
Journal:  Phytochem Rev       Date:  2022-02-08       Impact factor: 7.741

8.  Scaffold fragmentation and substructure hopping reveal potential, robustness, and limits of computer-aided pattern analysis (C@PA).

Authors:  Vigneshwaran Namasivayam; Katja Silbermann; Jens Pahnke; Michael Wiese; Sven Marcel Stefan
Journal:  Comput Struct Biotechnol J       Date:  2021-05-10       Impact factor: 7.271

9.  Combination of Inhibitors of USP7 and PLK1 has a Strong Synergism against Paclitaxel Resistance.

Authors:  Sol-Bi Shin; Chang-Hyeon Kim; Hay-Ran Jang; Hyungshin Yim
Journal:  Int J Mol Sci       Date:  2020-11-16       Impact factor: 5.923

10.  Cancer stem cells, epithelial-mesenchymal transition, ATP and their roles in drug resistance in cancer.

Authors:  Haiyun Zhang; Alexander Steed; Milo Co; Xiaozhuo Chen
Journal:  Cancer Drug Resist       Date:  2021-06-17
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