Literature DB >> 31471861

Leuprolide Acetate, a GnRH Agonist, Improves the Neurogenic Bowel in Ovariectomized Rats with Spinal Cord Injury.

Moisés Altamira-Camacho1, Daniel Medina-Aguiñaga1, Yolanda Cruz2, Denisse Calderón-Vallejo3, Kalman Kovacs4, Fabio Rotondo4, J Luis Quintanar5.   

Abstract

BACKGROUND: Electromyographic studies have shown that external anal sphincter activity is modified in response to distension in animals with spinal cord injury. Gonadotropin-releasing hormone and its agonist leuprolide acetate have neurotrophic properties in animals with spinal cord injury. AIM: This study was to determine the effects of leuprolide acetate treatment on electromyographic activity of the external anal sphincter and anorectal manometry in ovariectomized rats with spinal cord injury.
METHODS: Adult ovariectomized rats were divided in three groups: (a) sham of spinal cord injury, (b) spinal cord injury treated with saline solution, and (c) spinal cord injury treated with leuprolide acetate. The spinal cord injury was induced by clamping at level T9. Leuprolide acetate dosage of 10 μg/kg was proctored intramuscular for 5 weeks, commencing the day after the lesion. Electromyography of the external anal sphincter, anorectal manometry, and volume of the cecum were evaluated in all groups.
RESULTS: The electromyographic study of the external anal sphincter activity showed a significant improvement in injured rats treated with leuprolide acetate. Manometric analysis and cecum volume data obtained in animals with leuprolide acetate were very similar to those found in the sham group.
CONCLUSIONS: These results demonstrate that leuprolide acetate treatment improves the neurogenic colon in ovariectomized rats with spinal cord injury.

Entities:  

Keywords:  Cecum; Electromyography; External anal sphincter; GnRH; Neuroregeneration; SCI

Year:  2019        PMID: 31471861     DOI: 10.1007/s10620-019-05783-4

Source DB:  PubMed          Journal:  Dig Dis Sci        ISSN: 0163-2116            Impact factor:   3.199


  25 in total

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Authors:  Piero Periti; Teresita Mazzei; Enrico Mini
Journal:  Clin Pharmacokinet       Date:  2002       Impact factor: 6.447

2.  Persistent suppression of the pituitary-gonadal system in female rats by three-month depot injectable microspheres of leuprorelin acetate.

Authors:  H Okada; Y Doken; Y Ogawa
Journal:  J Pharm Sci       Date:  1996-10       Impact factor: 3.534

Review 3.  Neurogenic bowel management after spinal cord injury: a systematic review of the evidence.

Authors:  A Krassioukov; J J Eng; G Claxton; B M Sakakibara; S Shum
Journal:  Spinal Cord       Date:  2010-03-09       Impact factor: 2.772

4.  A sensitive and reliable locomotor rating scale for open field testing in rats.

Authors:  D M Basso; M S Beattie; J C Bresnahan
Journal:  J Neurotrauma       Date:  1995-02       Impact factor: 5.269

5.  Gonadotropin-releasing hormone treatment improves locomotor activity, urinary function and neurofilament protein expression after spinal cord injury in ovariectomized rats.

Authors:  Denisse Calderón-Vallejo; J Luis Quintanar
Journal:  Neurosci Lett       Date:  2012-03-28       Impact factor: 3.046

6.  Neurotrophic effects of GnRH on neurite outgrowth and neurofilament protein expression in cultured cerebral cortical neurons of rat embryos.

Authors:  J Luis Quintanar; Eva Salinas
Journal:  Neurochem Res       Date:  2007-12-20       Impact factor: 3.996

7.  Gonadotropin-releasing hormone receptor in spinal cord neurons of embryos and adult rats.

Authors:  J Luis Quintanar; Eva Salinas; Rodolfo González
Journal:  Neurosci Lett       Date:  2009-06-17       Impact factor: 3.046

8.  Debilitating "functional" bowel disease controlled by leuprolide acetate, gonadotropin-releasing hormone (GnRH) analog.

Authors:  J R Mathias; K L Ferguson; M H Clench
Journal:  Dig Dis Sci       Date:  1989-05       Impact factor: 3.199

9.  Effect of leuprolide acetate in treatment of abdominal pain and nausea in premenopausal women with functional bowel disease: a double-blind, placebo-controlled, randomized study.

Authors:  J R Mathias; M H Clench; T L Abell; K L Koch; G Lehman; M Robinson; R Rothstein; W J Snape
Journal:  Dig Dis Sci       Date:  1998-06       Impact factor: 3.199

Review 10.  Gonadotropin-Releasing Hormone and Its Role in the Enteric Nervous System.

Authors:  Bodil Ohlsson
Journal:  Front Endocrinol (Lausanne)       Date:  2017-06-07       Impact factor: 5.555

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