Literature DB >> 31270529

Efficacy and safety of alirocumab and evolocumab: a systematic review and meta-analysis of randomized controlled trials.

Paul Guedeney1,2, Gennaro Giustino1, Sabato Sorrentino1,3, Bimmer E Claessen1, Anton Camaj1, Deborah N Kalkman1,4, Birgit Vogel1, Samantha Sartori1, Salvatore De Rosa3, Usman Baber1, Ciro Indolfi3, Gilles Montalescot2, George D Dangas1, Robert S Rosenson1, Stuart J Pocock5, Roxana Mehran1.   

Abstract

AIMS: The effect of low-density lipoprotein cholesterol-lowering therapy with alirocumab or evolocumab on individual clinical efficacy and safety endpoints remains unclear. We aimed to evaluate the efficacy and safety of alirocumab and evolocumab in patients with dyslipidaemia or atherosclerotic cardiovascular disease. METHODS AND
RESULTS: We performed a review of randomized controlled trials (RCTs) comparing treatment with alirocumab or evolocumab vs. placebo or other lipid-lowering therapies up to March 2018. Primary efficacy endpoints were all-cause death, cardiovascular death, myocardial infarction (MI), and stroke. We estimated risk ratios (RR) and 95% confidence intervals (CI) using random effect models. We included 39 RCTs comprising 66 478 patients of whom 35 896 were treated with proprotein convertase subtilisin-kexin type 9 (PCSK9) inhibitors (14 639 with alirocumab and 21 257 with evolocumab) and 30 582 with controls. Mean weighted follow-up time across trials was 2.3 years with an exposure time of 150 617 patient-years. Overall, the effects of PCSK9 inhibition on all-cause death and cardiovascular death were not statistically significant (P = 0.15 and P = 0.34, respectively). Proprotein convertase subtilisin-kexin type 9 inhibitors were associated with lower risk of MI (1.49 vs. 1.93 per 100 patient-year; RR 0.80, 95% CI 0.74-0.86; I2 = 0%; P < 0.0001), ischaemic stroke (0.44 vs. 0.58 per 100 patient-year; RR 0.78, 95% CI 0.67-0.89; I2 = 0%; P = 0.0005), and coronary revascularization (2.16 vs. 2.64 per 100 patient-year; RR 0.83, 95% CI 0.78-0.89; I2 = 0%; P < 0.0001), compared with the control group. Use of these PCSK9 inhibitors was not associated with increased risk of neurocognitive adverse events (P = 0.91), liver enzymes elevations (P = 0.34), rhabdomyolysis (P = 0.58), or new-onset diabetes mellitus (P = 0.97).
CONCLUSION: Proprotein convertase subtilisin-kexin type 9 inhibition with alirocumab or evolocumab was associated with lower risk of MI, stroke, and coronary revascularization, with favourable safety profile. Published on behalf of the European Society of Cardiology. All rights reserved.
© The Author(s) 2019. For permissions, please email: journals.permissions@oup.com.

Entities:  

Keywords:  Alirocumab; Cholesterol-lowering therapies; Evolocumab; PCSK9

Year:  2019        PMID: 31270529     DOI: 10.1093/eurheartj/ehz430

Source DB:  PubMed          Journal:  Eur Heart J        ISSN: 0195-668X            Impact factor:   29.983


  24 in total

1.  Musculoskeletal Adverse Events Associated with PCSK9 Inhibitors: Disproportionality Analysis of the FDA Adverse Event Reporting System.

Authors:  Lingqing Ding; Congqin Chen; Yongkuan Yang; Jie Fang; Longxing Cao; Yige Liu
Journal:  Cardiovasc Ther       Date:  2022-01-25       Impact factor: 3.023

2.  PCSK9 inhibitors for secondary prevention in patients with cardiovascular diseases: a bayesian network meta-analysis.

Authors:  Xing Wang; Dingke Wen; Yuqi Chen; Lu Ma; Chao You
Journal:  Cardiovasc Diabetol       Date:  2022-06-15       Impact factor: 8.949

Review 3.  The Use of Monoclonal Antibody-Based Proprotein Convertase Subtilisin-Kexin Type 9 (PCSK9) Inhibitors in the Treatment of Hypercholesterolemia.

Authors:  Riya R Parikh; Frank Breve; Peter Magnusson; Payam Behzadi; Joseph Pergolizzi
Journal:  Cureus       Date:  2022-06-03

4.  Serum Proprotein Convertase Subtilisin/Kexin Type 9 (PCSK9) is Independently Associated with Insulin Resistance, Triglycerides, Lipoprotein(a) Levels but not Low-Density Lipoprotein Cholesterol Levels in a General Population.

Authors:  Hitoshi Hamamura; Hisashi Adachi; Mika Enomoto; Ako Fukami; Sachiko Nakamura; Yume Nohara; Nagisa Morikawa; Akiko Sakaue; Kenta Toyomasu; Maki Yamamoto; Yoshihiro Fukumoto
Journal:  J Atheroscler Thromb       Date:  2020-07-04       Impact factor: 4.928

5.  Effectiveness of proprotein convertase subtilisin/kexin-9 monoclonal antibody treatment on plasma lipoprotein(a) concentrations in patients with elevated lipoprotein(a) attending a clinic.

Authors:  Anindita Chakraborty; Jing Pang; Dick C Chan; Wendy Barnett; Ann Marie Woodward; Mary Vorster; Gerald F Watts
Journal:  Clin Cardiol       Date:  2021-05-06       Impact factor: 3.287

6.  Guía de práctica clínica mexicana para el diagnóstico y tratamiento de las dislipidemias y enfermedad cardiovascular aterosclerótica.

Authors:  Abel A Pavía-López; Marco A Alcocer-Gamba; Edith D Ruiz-Gastelum; José L Mayorga-Butrón; Roopa Mehta; Filiberto A Díaz-Aragón; Jorge A Aldrete-Velasco; Nitzia López-Juárez; Ivette Cruz-Bautista; Adolfo Chávez-Mendoza; Nikos C Secchi-Nicolás; Francisco J Guerrero-Martínez; Jorge E Cossio-Aranda; Victoria Mendoza-Zubieta; Guillermo Fanghänel-Salmon; Martha Valdivia-Proa; Luis Olmos-Domínguez; Carlos A Aguilar-Salinas; Luis Dávila-Maldonado; Armando Vázquez-Rangel; Vanina Pavia-Aubry; María de Los A Nava-Hernández; Carlos A Hinojosa-Becerril; Juan C Anda-Garay; Manuel O de Los Ríos-Ibarra; Ana C Berni-Betancourt; Julio López-Cuellar; Diego Araiza-Garaygordobil; Romina Rivera-Reyes; Gabriela Borrayo-Sánchez; Mónica Tapia-Hernández; Claudia V Cano-Nigenda; Arturo Guerra-López; Josué Elías-López; Marco A Figueroa-Morales; Bertha B Montaño-Velázquez; Liliana Velasco-Hidalgo; Ana L Rodríguez-Lozano; Claudia Pimentel-Hernández; María M Baquero-Hoyos; Felipe Romero-Moreno; Mario Rodríguez-Vega
Journal:  Arch Cardiol Mex       Date:  2022

Review 7.  Early Aspirin Discontinuation Following Acute Coronary Syndrome or Percutaneous Coronary Intervention: A Systematic Review and Meta-Analysis of Randomized Controlled Trials.

Authors:  Paul Guedeney; Jules Mesnier; Sabato Sorrentino; Farouk Abcha; Michel Zeitouni; Benoit Lattuca; Johanne Silvain; Salvatore De Rosa; Ciro Indolfi; Jean-Philippe Collet; Mathieu Kerneis; Gilles Montalescot
Journal:  J Clin Med       Date:  2020-03-03       Impact factor: 4.241

Review 8.  What Lessons Have We Learned and What Remains to be Clarified for PCSK9 Inhibitors? A Review of FOURIER and ODYSSEY Outcomes Trials.

Authors:  Remo H M Furtado; Robert P Giugliano
Journal:  Cardiol Ther       Date:  2020-02-05

Review 9.  Antiplatelet Effects of PCSK9 Inhibitors in Primary Hypercholesterolemia.

Authors:  Piotr Pęczek; Mateusz Leśniewski; Tomasz Mazurek; Lukasz Szarpak; Krzysztof J Filipiak; Aleksandra Gąsecka
Journal:  Life (Basel)       Date:  2021-05-23

10.  Inclisiran for the treatment of hypercholesterolaemia: implications and unanswered questions from the ORION trials.

Authors:  Arjen J Cupido; John J P Kastelein
Journal:  Cardiovasc Res       Date:  2020-09-01       Impact factor: 10.787

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