Literature DB >> 31098984

Superior Diagnostic Performance of the GLP-1 Receptor Agonist [Lys40(AhxHYNIC-[99mTc]/EDDA)NH2]-Exendin-4 over Conventional Imaging Modalities for Localization of Insulinoma.

Katra Senica1, Ales Tomazic2, Ales Skvarca3, Petra Kolenc Peitl1, Renata Mikolajczak4, Alicja Hubalewska-Dydejczyk5, Luka Lezaic6.   

Abstract

PURPOSE: Insulinomas are the most common functioning neuroendocrine neoplasms of the pancreas, typically diagnosed due to characteristic symptoms. In the vast majority, the treatment is surgical and curative, requiring accurate localization of the tumour; conventional imaging, including somatostatin receptor molecular imaging, is negative in up to 10 % of cases. Recently, labelled glucagon-like peptide receptor (GLP-1R) analogues were introduced as a sensitive diagnostic method for localization of insulinomas. The aim of this study was to assess the diagnostic accuracy of a Tc-99m-labelled GLP-1R agonist [Lys40(AhxHYNIC-[99mTc]EDDA)NH2]-exendin-4 for localization of occult insulinoma. PROCEDURES: Eight patients (all females; age range 35-75 years) with biochemically proven insulinoma and with negative or inconclusive conventional imaging (consisting of somatostatin receptor scintigraphy, computed tomography, endoscopic ultrasound and magnetic resonance imaging) were enrolled. Whole-body single-photon emission tomography/computed tomography (SPECT/CT) imaging was performed 4 h post-injection of 740 MBq of [Lys40(AhxHYNIC-[99mTc]EDDA)NH2]-exendin-4. Surgical treatment was performed based on imaging findings. Histology of the removed lesions and biochemical and clinical symptom resolution was considered as the gold standard for analysis of the imaging results.
RESULTS: Focal uptake of [Lys40(AhxHYNIC-[99mTc]EDDA)NH2]-exendin-4 was found in all patients, leading to successful removal of the offending lesion and complete biochemical and symptomatic resolution. Histological analysis confirmed insulinoma in all included patients.
CONCLUSIONS: [Lys40(AhxHYNIC-[99mTc]EDDA)NH2]-exendin-4 SPECT/CT appears to be an excellent molecular imaging method for preoperative localization of an occult insulinoma, surpassing conventional imaging methods. If routinely available, it could be considered as a method of choice due to its favorable combination of imaging characteristics.

Entities:  

Keywords:  Exendin; GLP-1; GLP-1 receptor; Insulinoma; SPECT; SPECT/CT; Scintigraphy

Year:  2020        PMID: 31098984     DOI: 10.1007/s11307-019-01372-z

Source DB:  PubMed          Journal:  Mol Imaging Biol        ISSN: 1536-1632            Impact factor:   3.488


  30 in total

Review 1.  Insulinoma.

Authors:  Kimberly Vanderveen; Clive Grant
Journal:  Cancer Treat Res       Date:  2010

Review 2.  Pancreatic endocrine tumors.

Authors:  Kjell Oberg
Journal:  Semin Oncol       Date:  2010-12       Impact factor: 4.929

3.  Localization of Insulinoma Using 68Ga-DOTATATE PET/CT Scan.

Authors:  Pavel Nockel; Bruna Babic; Corina Millo; Peter Herscovitch; Dhaval Patel; Naris Nilubol; Samira M Sadowski; Craig Cochran; Phillip Gorden; Electron Kebebew
Journal:  J Clin Endocrinol Metab       Date:  2017-01-01       Impact factor: 5.958

4.  The role of arterial stimulation and simultaneous venous sampling in addition to cross-sectional imaging for localisation of biochemically proven insulinoma.

Authors:  D L Morganstein; D H Lewis; J Jackson; A Isla; J Lynn; D Devendra; K Meeran; J F Todd
Journal:  Eur Radiol       Date:  2009-07-14       Impact factor: 5.315

5.  An intrapatient comparison of 99mTc-EDDA/HYNIC-TOC with 111In-DTPA-octreotide for diagnosis of somatostatin receptor-expressing tumors.

Authors:  Michael Gabriel; Clemens Decristoforo; Eveline Donnemiller; Hanno Ulmer; Christine Watfah Rychlinski; Stephen J Mather; Roy Moncayo
Journal:  J Nucl Med       Date:  2003-05       Impact factor: 10.057

6.  Somatostatin receptor based PET/CT imaging with 68Ga-DOTA-Nal3-octreotide for localization of clinically and biochemically suspected insulinoma.

Authors:  Punit Sharma; Saurabh Arora; Sellam Karunanithi; Rajesh Khadgawat; Prashant Durgapal; Raju Sharma; Devasenathipathy Kandasamy; Chandrasekhar Bal; Rakesh Kumar
Journal:  Q J Nucl Med Mol Imaging       Date:  2014-04-17       Impact factor: 2.346

7.  Glucagon-like peptide-1 receptor imaging for localization of insulinomas.

Authors:  Emanuel Christ; Damian Wild; Flavio Forrer; Michael Brändle; Rahel Sahli; Thomas Clerici; Beat Gloor; Ferdinand Martius; Helmut Maecke; Jean Claude Reubi
Journal:  J Clin Endocrinol Metab       Date:  2009-10-09       Impact factor: 5.958

8.  Glucagon-like peptide-1 receptor imaging for the localisation of insulinomas: a prospective multicentre imaging study.

Authors:  Emanuel Christ; Damian Wild; Susanne Ederer; Martin Béhé; Guillaume Nicolas; Martyn E Caplin; Michael Brändle; Thomas Clerici; Stefan Fischli; Christoph Stettler; Peter J Ell; Jochen Seufert; Beat Gloor; Aurel Perren; Jean Claude Reubi; Flavio Forrer
Journal:  Lancet Diabetes Endocrinol       Date:  2013-07-25       Impact factor: 32.069

9.  Localization of insulinomas to regions of the pancreas by intraarterial calcium stimulation: the NIH experience.

Authors:  Jean-Marc Guettier; Anthony Kam; Richard Chang; Monica C Skarulis; Craig Cochran; H Richard Alexander; Steven K Libutti; James F Pingpank; Phillip Gorden
Journal:  J Clin Endocrinol Metab       Date:  2009-02-03       Impact factor: 5.958

10.  (64)Cu labeled sarcophagine exendin-4 for microPET imaging of glucagon like peptide-1 receptor expression.

Authors:  Zhanhong Wu; Shuanglong Liu; Indu Nair; Keiko Omori; Stephen Scott; Ivan Todorov; John E Shively; Peter S Conti; Zibo Li; Fouad Kandeel
Journal:  Theranostics       Date:  2014-05-24       Impact factor: 11.556

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  2 in total

1.  Changing Insulinoma Management Due to Incidentally Discovered Metastasis: A Case Report.

Authors:  Riya Madan; Tetyana Mettler; Jerry Froelich; Lisa S Chow
Journal:  Am J Case Rep       Date:  2020-06-14

2.  Synthesis and in vivo behaviour of an exendin-4-based MRI probe capable of β-cell-dependent contrast enhancement in the pancreas.

Authors:  Thomas J Clough; Nicoleta Baxan; Emma J Coakley; Charlotte Rivas; Lan Zhao; Isabelle Leclerc; Aida Martinez-Sanchez; Guy A Rutter; Nicholas J Long
Journal:  Dalton Trans       Date:  2020-04-15       Impact factor: 4.390

  2 in total

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