Literature DB >> 31073972

Efficacy and safety of trifluridine/tipiracil in third-line and beyond for the treatment of patients with metastatic colorectal cancer in routine clinical practice: patterns of use and prognostic nomogram.

A Fernandez Montes1, F Vazquez Rivera2, N Martinez Lago3, M Covela Rúa4, A Cousillas Castiñeiras5, P Gonzalez Villarroel6, J de la Cámara Gómez7, J C Méndez Méndez8, M Salgado Fernández9, S Candamio Folgar2, M Reboredo López3, M Carmona Campos4, E Gallardo Martín10, M Jorge Fernández6, M L Pellón Augusto7, L París Bouzas8, J García Gómez11.   

Abstract

INTRODUCTION: Trifluridine/tipiracil combination has shown a benefit over placebo in the treatment of patients with chemorefractory metastatic colorectal cancer (mCRC). We evaluated the efficacy and safety of this combination in the real-life setting at eight Galician centers in Spain. PATIENTS AND METHODS: This is a retrospective study of a cohort of patients with mCRC in treatment with trifluridine/tipiracil within usual clinical practice who have been previously treated or are not considered candidates for treatment with available therapies.
RESULTS: A total of 160 mCRC patients were included. Our data showed that 11.9% of patients achieved disease control. Median progression-free survival was 2.75 months; at 5.66 months follow-up, median overall survival was 7.94 months. Asthenia and neutropenia (48.1% both) were the most frequent adverse events. Overall survival was lower in patients with ECOG 2, multiple metastatic sites, platelets count 350,000/µl, alkaline phosphatase > 500 IU/l, and carcinoembryonic antigen > 10 ng/ml.
CONCLUSION: The results of this study confirm the efficacy and safety of trifluridine/tipiracil in chemorefractory mCRC patients. However, patients in clinical practice differ from patients in clinical trials. Due to this, prognostic factors have special importance to offer the best therapeutic approach.

Entities:  

Keywords:  Metastatic colorectal cancer; Nomogram; Prognostic factors; Real-life; Refractory; Trifluridine/tipiracil

Mesh:

Substances:

Year:  2019        PMID: 31073972     DOI: 10.1007/s12094-019-02130-x

Source DB:  PubMed          Journal:  Clin Transl Oncol        ISSN: 1699-048X            Impact factor:   3.405


  25 in total

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Authors:  E Van Cutsem; A Cervantes; B Nordlinger; D Arnold
Journal:  Ann Oncol       Date:  2014-09-04       Impact factor: 32.976

2.  Structure and activity of specific inhibitors of thymidine phosphorylase to potentiate the function of antitumor 2'-deoxyribonucleosides.

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Journal:  Biochem Pharmacol       Date:  2000-05-15       Impact factor: 5.858

3.  Irinotecan plus fluorouracil and leucovorin for metastatic colorectal cancer. Irinotecan Study Group.

Authors:  L B Saltz; J V Cox; C Blanke; L S Rosen; L Fehrenbacher; M J Moore; J A Maroun; S P Ackland; P K Locker; N Pirotta; G L Elfring; L L Miller
Journal:  N Engl J Med       Date:  2000-09-28       Impact factor: 91.245

4.  Neutropenia as a Predictive Factor in Metastatic Colorectal Cancer Treated With TAS-102.

Authors:  Satoshi Hamauchi; Kentaro Yamazaki; Toshiki Masuishi; Yosuke Kito; Azusa Komori; Takahiro Tsushima; Yukiya Narita; Akiko Todaka; Makoto Ishihara; Tomoya Yokota; Tsutomu Tanaka; Nozomu Machida; Shigenori Kadowaki; Akira Fukutomi; Takashi Ura; Yusuke Onozawa; Masashi Ando; Masahiro Tajika; Kei Muro; Hirofumi Yasui; Keita Mori; Hiroya Taniguchi
Journal:  Clin Colorectal Cancer       Date:  2016-07-21       Impact factor: 4.481

5.  Fluorinated pyrimidines. XXXVII. Effects of 5-trifluoromethyl-2'-deoxyuridine on the synthesis of deoxyribonucleic acid of mammalian cells in culture.

Authors:  Y Fujiwara; T Oki; C Heidelberger
Journal:  Mol Pharmacol       Date:  1970-05       Impact factor: 4.436

6.  Cancer incidence and mortality patterns in Europe: estimates for 40 countries in 2012.

Authors:  J Ferlay; E Steliarova-Foucher; J Lortet-Tieulent; S Rosso; J W W Coebergh; H Comber; D Forman; F Bray
Journal:  Eur J Cancer       Date:  2013-02-26       Impact factor: 9.162

7.  Safety of an oral anticancer agent (trifluridine/tipiracil combination tablet) in patients with advanced and recurrent colorectal cancer.

Authors:  M Kimura; M Go; M Iwai; D Ito; H Asano; E Usami; H Teramachi; T Yoshimura
Journal:  Pharmazie       Date:  2016-04       Impact factor: 1.267

8.  Phase I clinical study of three times a day oral administration of TAS-102 in patients with solid tumors.

Authors:  Michael J Overman; Scott Kopetz; Gauri Varadhachary; Masakazu Fukushima; Keizo Kuwata; Akira Mita; Robert A Wolff; Paulo Hoff; Henry Xiong; James L Abbruzzese
Journal:  Cancer Invest       Date:  2008-10       Impact factor: 2.176

9.  Regorafenib monotherapy for previously treated metastatic colorectal cancer (CORRECT): an international, multicentre, randomised, placebo-controlled, phase 3 trial.

Authors:  Axel Grothey; Eric Van Cutsem; Alberto Sobrero; Salvatore Siena; Alfredo Falcone; Marc Ychou; Yves Humblet; Olivier Bouché; Laurent Mineur; Carlo Barone; Antoine Adenis; Josep Tabernero; Takayuki Yoshino; Heinz-Josef Lenz; Richard M Goldberg; Daniel J Sargent; Frank Cihon; Lisa Cupit; Andrea Wagner; Dirk Laurent
Journal:  Lancet       Date:  2012-11-22       Impact factor: 79.321

10.  Retrospective study of regorafenib and trifluridine/tipiracil efficacy as a third-line or later chemotherapy regimen for refractory metastatic colorectal cancer.

Authors:  Akira Tanaka; Sotaro Sadahiro; Toshiyuki Suzuki; Kazutake Okada; Gota Saito; Hiroshi Miyakita
Journal:  Oncol Lett       Date:  2018-09-07       Impact factor: 2.967

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  1 in total

Review 1.  TAS-102 Monotherapy and Combination Therapy with Bevacizumab for Metastatic Colorectal Cancer.

Authors:  Cheng-Jiang Liu; Ting Hu; Ping Shao; Wu-Yang Chu; Yu Cao; Feng Zhang
Journal:  Gastroenterol Res Pract       Date:  2021-12-20       Impact factor: 2.260

  1 in total

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