Literature DB >> 31027702

From the beginning to resistance: Study of plasma monitoring and resistance mechanisms in a cohort of patients treated with osimertinib for advanced T790M-positive NSCLC.

Paola Bordi1, Marzia Del Re2, Roberta Minari3, Eleonora Rofi2, Sebastiano Buti1, Giuliana Restante2, Anna Squadrilli1, Stefania Crucitta2, Chiara Casartelli1, Letizia Gnetti4, Cinzia Azzoni4, Lorena Bottarelli4, Iacopo Petrini5, Agnese Cosenza1, Leonarda Ferri1, Elena Rapacchi1, Romano Danesi2, Marcello Tiseo6.   

Abstract

INTRODUCTION: Analysis of circulating tumor DNA (ctDNA) for the identification of T790M mutation in advanced EGFR-mutated NSCLC patients can replace tissue re-biopsy for resistance characterization and, being non-invasive, may be applied for disease monitoring. We analysed ctDNA during osimertinib treatment to correlate mutational levels with clinical outcome and to predict pattern of resistance.
MATERIALS AND METHODS: Forty patients with advanced NSCLC receiving osimertinib for T790M + disease after previous EGFR-TKI were enrolled in a pilot study to collect plasma at baseline and every 12 weeks until progression. Molecular analysis of ctDNA was performed by ddPCR and Therascreen®. When feasible at progression, tissue re-biopsy and NGS analysis were performed.
RESULTS: Thirty-eight patients had baseline plasma samples suitable for molecular analysis. Patients with low levels of the EGFR activating mutation in ctDNA [< 2200 copies/mL or allele frequency (AF) < 6.1%] showed better progression-free survival (17.8 or 17.8 months vs. 4.3 or 2.7, p = 0.022 or p = 0.018, respectively) and overall survival (23.6 or 23.6 vs. 7.7 or 7.3, p = 0.016 or p = 0.013, respectively) than patients with high levels (≥ 2200 copies/mL or AF ≥ 6.1%). Patients with detectable EGFR mutations in plasma (shedders) presented worse outcome than negative subjects (non-shedders). Low levels of T790M, higher T790M/activating mutation ratio and complete clearance after 2 months were associated with a trend towards better outcome. Tissue re-biopsy at resistance showed 3 patients with EGFR C797S, 1 with MET amplification, 1 with MYC amplification, 1 with PTEN loss, 3 with SCLC transformation.
CONCLUSIONS: The mutational analysis performed on plasma plays a significant role in prognostic stratification, especially for the EGFR activating mutation, since patients with absence or low levels of mutations presented a better outcome to osimertinib. At progression, tissue re-biopsy remains a crucial issue for the identification of resistance mechanisms.
Copyright © 2019 Elsevier B.V. All rights reserved.

Entities:  

Keywords:  EGFR mutation; Liquid biopsy; NSCLC; Osimertinib; T790M

Mesh:

Substances:

Year:  2019        PMID: 31027702     DOI: 10.1016/j.lungcan.2019.03.017

Source DB:  PubMed          Journal:  Lung Cancer        ISSN: 0169-5002            Impact factor:   5.705


  15 in total

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4.  The prognostic value of longitudinal circulating tumor DNA profiling during osimertinib treatment.

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Journal:  Transl Lung Cancer Res       Date:  2021-01

Review 5.  Liquid Biopsies: Applications for Cancer Diagnosis and Monitoring.

Authors:  Ivana Martins; Ilda Patrícia Ribeiro; Joana Jorge; Ana Cristina Gonçalves; Ana Bela Sarmento-Ribeiro; Joana Barbosa Melo; Isabel Marques Carreira
Journal:  Genes (Basel)       Date:  2021-02-27       Impact factor: 4.096

6.  Dynamic cfDNA Analysis by NGS in EGFR T790M-Positive Advanced NSCLC Patients Failed to the First-Generation EGFR-TKIs.

Authors:  Li Ma; Haoyang Li; Dongpo Wang; Ying Hu; Mengjun Yu; Quan Zhang; Na Qin; Xinyong Zhang; Xi Li; Hui Zhang; Yuhua Wu; Jialin Lv; Xinjie Yang; Ruoying Yu; Shucai Zhang; Jinghui Wang
Journal:  Front Oncol       Date:  2021-03-25       Impact factor: 6.244

7.  Targeting c-Myc to Overcome Acquired Resistance of EGFR Mutant NSCLC Cells to the Third-Generation EGFR Tyrosine Kinase Inhibitor, Osimertinib.

Authors:  Lei Zhu; Zhen Chen; Hongjing Zang; Songqing Fan; Jiajia Gu; Guojing Zhang; Kevin D-Y Sun; Qiming Wang; Yong He; Taofeek K Owonikoko; Suresh S Ramalingam; Shi-Yong Sun
Journal:  Cancer Res       Date:  2021-07-21       Impact factor: 12.701

8.  Neuropilin-2b facilitates resistance to tyrosine kinase inhibitors in non-small cell lung cancer.

Authors:  Anastasios Dimou; Cecile Nasarre; Yuri K Peterson; Rose Pagano; Monika Gooz; Patrick Nasarre; Harry A Drabkin; Kent E Armeson; Barry C Gibney; Robert M Gemmill; Chadrick E Denlinger
Journal:  J Thorac Cardiovasc Surg       Date:  2020-05-25       Impact factor: 6.439

9.  Concomitant genetic alterations are associated with response to EGFR targeted therapy in patients with lung adenocarcinoma.

Authors:  Hualin Chen; Meilian Liu; Zhiwei Dai; Shujun Li; Yiping Luo; Yongcun Wang; Wenmei Su; Weijing Cai; Donghong Yang; Jian Huang; Zhixiong Yang
Journal:  Transl Lung Cancer Res       Date:  2020-08

10.  Licochalcone A inhibits EGFR signalling and translationally suppresses survivin expression in human cancer cells.

Authors:  Feng Gao; Ming Li; Xinfang Yu; Wenbin Liu; Li Zhou; Wei Li
Journal:  J Cell Mol Med       Date:  2020-11-27       Impact factor: 5.295

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